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1-{1-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}pyrrolidin-2-one
2-({5-[3-(methoxymethyl)piperidine-1-carbonyl]pyridin-2-yl}(methyl)amino)ethan-1-ol
5-butyl-1'-(5-phenyl-1,2,4-oxadiazol-3-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-(2-hydroxyethyl)-3-[(5-methylthiophen-2-yl)methyl]-1-[3-(piperidin-1-ylmethyl)phenyl]urea
N-(4-{[({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)(2-methylpropyl)amino]methyl}phenyl)acetamide
(3R,9aR)-8-(cyclohexylmethyl)-3-(hydroxymethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-{[3-(2-fluorophenoxy)azetidin-1-yl]methyl}-2-(methylsulfanyl)pyrimidine
N-(3,4-dimethylphenyl)-1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]piperidin-3-amine
1-[(2-chloro-6-fluorophenyl)methyl]-4-(4-methyl-5-{[2-(piperidin-1-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)piperidine
(2R,3S,6R)-3-(2-methoxyphenyl)-5-(morpholine-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
9-[3-(difluoromethoxy)benzoyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-methoxy-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]pyridine-4-carboxamide
3-[(3R,4S)-1-(3,6-dimethylpyrazin-2-yl)-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
[(5-{1-[(2,4-difluorophenyl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
N2-(4-cyclopentylpyrimidin-2-yl)-N1-(pyridin-3-yl)ethane-1,2-diamine
3,6-dimethyl-N-{1-oxaspiro[4.5]decan-3-yl}-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
4-(4-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}piperidine-1-carbonyl)pyridine
5-cyclopropyl-1-[4-(3-fluoro-4-methoxyphenyl)pyrimidin-2-yl]-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
4-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidine-1-carbonyl]-1-ethyl-1,2-dihydropyridin-2-one
(3S,5R)-N-(4-methylphenyl)-5-(3-oxopiperazine-1-carbonyl)piperidine-3-carboxamide
1-({1-[(3-fluoro-2,4-dimethylphenyl)methyl]pyrrolidin-3-yl}methyl)-3-(propan-2-yl)urea
4-{2-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]phenyl}-1λ6-thiomorpholine-1,1-dione
1-(1-benzofuran-2-carbonyl)-N-(4-methoxyphenyl)piperidin-3-amine
4-(4-chlorophenoxy)-1-[(2E)-3-phenylprop-2-en-1-yl]piperidine-4-carboxylic acid
1-{6-hydroxy-4-[2-(1H-pyrazol-4-yl)ethyl]-1,4-diazepan-1-yl}-2-(pyrrolidin-1-yl)ethan-1-one
[1-(2-chlorophenyl)ethyl]({[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl})amine
N-methyl-N-(1,2-oxazol-5-ylmethyl)-1-[4-(1,3-thiazol-4-yl)phenyl]piperidin-4-amine
methyl 4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
(1H-1,3-benzodiazol-2-ylmethyl)(furan-2-ylmethyl)(prop-2-en-1-yl)amine
5-({cyclopropyl[(3-ethoxyphenyl)methyl]amino}methyl)-2-methoxybenzoic acid
N-(1-{2-oxo-2-[2-(1,3-thiazol-2-yl)piperidin-1-yl]ethyl}-1H-pyrazol-4-yl)benzamide
3-{1-[3-(2-methoxyphenyl)propanoyl]piperidin-4-yl}-N-(3-methylphenyl)propanamide
4-{1-[2-(1H-imidazol-4-yl)-1H-imidazol-1-yl]ethyl}-2-methyl-1,3-thiazole
1-[1-(2-methoxyethyl)piperidine-4-carbonyl]spiro[azepane-4,2'-chromene]
5-[methyl(2-phenylethyl)amino]-2-[(1-methylpiperidin-2-yl)methyl]-2,3-dihydropyridazin-3-one
N-[2-(2-chlorophenoxy)ethyl]-N-ethyl-2-(1H-imidazol-2-yl)benzamide
N-[3-(2-methoxybenzamido)phenyl]-3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
2-{[2-(3-methylpyridin-2-yl)ethyl]amino}-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-(2,3-dihydro-1-benzofuran-5-carbonyl)-3-{[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
2-phenyl-N-{1-[1-(1,2,5-thiadiazole-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}acetamide
methyl[(3-{[1-(2,3,4,9-tetrahydro-1H-carbazole-6-carbonyl)piperidin-4-yl]oxy}phenyl)methyl](thiophen-2-ylmethyl)amine
3-{[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl}benzoic acid
4-methoxy-1-({3-[3-(trifluoromethyl)phenoxy]phenyl}methyl)piperidine
1-{2-[(2-chlorophenyl)methyl]morpholin-4-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one
methyl 2-({5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)acetate
1-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-3-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}urea
[(3,7-dimethyl-1H-indol-2-yl)methyl]({[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl})methylamine
5-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-N-[(5-methylfuran-2-yl)methyl]pyridin-2-amine
4-{[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methyl}morpholine
3-[(3S,4R)-4-(dimethylamino)-1-(naphthalen-2-ylmethyl)piperidin-3-yl]-N-[2-(1H-imidazol-4-yl)ethyl]propanamide