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2-hydroxy-N-(isoquinolin-5-ylmethyl)-N-methyl-6-(trifluoromethyl)pyridine-3-carboxamide
(3aR,6aS)-5-{[2-(cyclopentyloxy)phenyl]methyl}-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[2-oxo-2-(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)ethyl]pyrrolidin-2-one
N-methyl-2-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyridine-3-carboxamide
1-(6-chloro-2-methylpyridin-3-yl)-3-[2-(pyrrolidine-1-sulfonyl)ethyl]urea
ethyl 4-(1-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}piperidin-3-yl)piperazine-1-carboxylate
2-(4-fluorophenyl)-2-{[2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}ethan-1-ol
N-(cyclohexylmethyl)-3-oxo-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
7-(3,6-dimethylpyrazin-2-yl)-4-(oxolan-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-ethyl-3-methyl-N-[(6-oxo-1,6-dihydropyrimidin-4-yl)methyl]piperidine-3-carboxamide
N-methyl-2-phenyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
methyl 5-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[2-(piperidin-1-yl)ethyl]benzamide
2-[4-cyclohexyl-1-(propan-2-yl)piperazin-2-yl]ethan-1-ol
(3R,4R)-1-[(2-fluorophenyl)methyl]-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
N-(1H-indol-2-ylmethyl)-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-(4-{furo[3,2-c]pyridin-4-yl}-1H-pyrazol-1-yl)-N-(1-methyl-1H-indazol-3-yl)acetamide
N-[(3R,5S)-1-[(3-ethenylphenyl)methyl]-5-(ethylcarbamoyl)pyrrolidin-3-yl]-1H-imidazole-2-carboxamide
6-(4-ethoxypiperidin-1-yl)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(15),3(8),6,11,13-pentaen-4-one
1-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}-3-(pyridin-3-yl)propan-1-one
N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-{4-[1-(2H-1,3-benzodioxol-5-ylmethyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}-N,N-dimethylacetamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[4-(trifluoromethyl)pyrimidin-2-yl]piperidin-3-ol
4-phenyl-3-(piperidin-3-yl)-1-[2-(1H-1,2,4-triazol-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[3-(1H-indol-2-yl)phenyl]-1-propylpiperidine-3-carboxamide
N-{1-[1-(2-methoxyphenyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide
methyl 5-[(1-ethyl-1H-imidazol-5-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
1-methyl-6-({2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}methyl)-1H-indole
3-cyclohexyl-N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
1-[(3-chlorophenyl)methyl]-N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
6-ethyl-N-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}pyrimidin-4-amine
3-{4-[(2-cyclohexylpyrimidin-5-yl)methyl]piperazin-1-yl}-2,5-dimethylpyrazine
methyl 2-(ethylsulfamoyl)-6-[(2-methylphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-(3-methylphenoxy)-1-[2-(4-methylpiperazine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]ethan-1-one
3-[(2R,3R,6R)-5-(4-fluorobenzoyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
(4-{5-[(pyridin-2-ylsulfanyl)methyl]-1,2,4-oxadiazol-3-yl}phenyl)methanol
(5S,9aS,9bS)-2-phenyl-5-[1-(pyridin-3-yl)-1H-pyrrol-2-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-(1-ethylpiperidine-2-carbonyl)-1-(oxan-4-ylmethyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
3-methyl-7-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
3-{2-[4-(4-hydroxyphenyl)piperazin-1-yl]-2-oxoethyl}-4-(2-methylpropyl)piperazin-2-one
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-(3-methyl-5-oxo-1-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl)acetamide
2-(azocan-1-yl)-1-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-one
4-(1H-indazol-6-yl)-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
4-(2,2-dimethylpropyl)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
3-(2-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-2-oxoethyl)-1,3-thiazolidine-2,4-dione
7-[(4-fluorophenyl)methyl]-2-[(trimethylpyrazin-2-yl)methyl]-2,7-diazaspiro[4.5]decane
{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]amine
1-(1,3-benzothiazol-2-yl)-N-[3-(methylsulfanyl)propyl]piperidin-3-amine
3-(2-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-oxoethyl)imidazolidine-2,4-dione
N-[4-(methylsulfanyl)phenyl]-3-(4-phenylpiperazin-1-yl)piperidine-1-carboxamide