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6-{[2-(butan-2-yloxy)phenyl]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
5-cyclopropyl-1-[4-(2-fluorophenyl)pyrimidin-2-yl]-N-[2-(pyridin-3-yl)ethyl]-1H-pyrazole-4-carboxamide
N,N-dimethyl-2-{2-[2-(thiophen-2-yl)ethyl]piperidine-1-carbonyl}aniline
ethyl 4-(2-methoxyethyl)-1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidine-4-carboxylate
methyl (2S,4S)-1-(naphthalen-2-ylmethyl)-4-[4-(1H-pyrazol-1-yl)benzamido]pyrrolidine-2-carboxylate
3-[1-(1-benzylpiperidin-4-yl)-1H-1,2,3-triazol-4-yl]pyridine
1-[4-({[(2,6-difluorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]-3-(4-ethylpiperazin-1-yl)propan-2-ol
5-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-3-(2-methylpropyl)-1H-pyrazole
N'-(3-ethylphenyl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]butanediamide
3-(2-hydroxyphenyl)-N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-1H-pyrazole-5-carboxamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]quinoline-5-carboxamide
N3-methyl-N3-[3-(4-methylphenoxy)propyl]piperidine-1,3-dicarboxamide
7-(2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}acetyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-{[8-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
5-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
methyl 3-(4-methoxy-4-oxobutanoyl)-7-oxo-9-(thiophen-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-3-[3-methyl-1-(propan-2-yl)-1H-pyrazol-5-yl]urea
N-(butan-2-yl)-4-[5-(4-methoxybenzamido)-1H-pyrazol-1-yl]piperidine-1-carboxamide
N1,N1-dimethyl-N3-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)piperidine-1,3-dicarboxamide
methyl[(3-methyl-1,2-oxazol-5-yl)methyl]{[2-(propan-2-yl)pyrimidin-4-yl]methyl}amine
1-{[1-(2-methyl-1,3-benzothiazole-6-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
1-(3-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-3-oxopropyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(4-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl)ethan-1-ol
3-(cyclohexylamino)-5-(dimethylsulfamoyl)-N-[(1R)-1-(4-methoxyphenyl)ethyl]benzamide
2-({[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)amino)ethan-1-ol
N-[2-(4-methoxyphenyl)ethyl]-N-[(1-methylpiperidin-4-yl)methyl]cyclohex-3-ene-1-carboxamide
3-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidine-1-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
1-(3-benzoylpiperidin-1-yl)-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}ethan-1-one
5-(1,2-oxazinane-2-carbonyl)-1-(pyridin-2-ylmethyl)piperidin-2-one
3-(1-cyclopentyl-4-methyl-1H-pyrazol-5-yl)-1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}urea
4-(2,3-dimethylphenyl)-3-[(methylamino)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[(2-fluorophenyl)methyl]-1-[(4-methyl-1,3-thiazol-5-yl)methyl]piperidine
4-[4-(furan-2-ylmethyl)piperazin-1-yl]-2-[2-(1H-pyrazol-1-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
(4aR,7aS)-1-(2-methoxyethyl)-4-[(2-methyl-1,3-oxazol-4-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{1-ethyl-5-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-4-phenylpiperazine
(2-methoxyethyl)[(3-methylthiophen-2-yl)methyl]{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}amine
4-hydroxy-N-methyl-2-(4-methylphenyl)-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}pyrimidine-5-carboxamide
1-(1,4-dithiepan-6-yl)-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
ethyl 3-[(2-methylphenyl)methyl]-1-[(trimethyl-1H-pyrazol-4-yl)sulfonyl]piperidine-3-carboxylate
1-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(propylsulfanyl)ethan-1-one
5-{3-[(dimethylamino)methyl]-3-hydroxypyrrolidine-1-carbonyl}thiophene-2-carboxylic acid
1-(2-methoxyethyl)-8-[3-(5-methylfuran-2-yl)butyl]-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(4-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-1-yl)-N-(propan-2-yl)acetamide
2-cyclopropyl-N-[(5-methylfuran-2-yl)methyl]-1,3-benzoxazole-6-carboxamide
1-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-3-phenoxypropan-1-one
3-(1,3-thiazol-2-yl)-7-thia-2,4,5-triazatricyclo[6.4.0.02,6]dodeca-1(12),3,5,8,10-pentaene
ethyl 5-[(4-formylpiperazin-1-yl)methyl]-1-(4-phenyl-1,3-thiazol-2-yl)-1H-pyrazole-4-carboxylate
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}quinoxaline