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3,4,7-trimethyl-2-{4-[1-(morpholin-4-yl)ethyl]piperidine-1-carbonyl}-1H-indole
2-(3-methyl-5-oxo-1-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl)-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}acetamide
(1S,5R)-3-benzyl-6-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
(2S,4R)-4-amino-N-(propan-2-yl)-1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}pyrrolidine-2-carboxamide
3-{[methyl({[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl})amino]methyl}pyrrolidin-3-ol
2-[(3,5-difluorophenyl)methyl]-8-methanesulfonyl-2,8-diazaspiro[4.5]decan-3-one
1-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-3-(3-ethyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)urea
N-[3-(4-{methyl[1-(4-methyl-1,3-thiazol-2-yl)ethyl]amino}piperidin-1-yl)phenyl]-4-phenylbutanamide
N-cyclopentyl-2-(2,3-difluorophenoxymethyl)-N-propyl-1,3-oxazole-4-carboxamide
6-amino-N-[(3S,5S)-1-[(2E)-but-2-en-1-yl]-5-(ethylcarbamoyl)pyrrolidin-3-yl]pyridine-3-carboxamide
N-[(5-phenyl-1H-pyrazol-3-yl)methyl]-N-(propan-2-yl)-2,8-diazaspiro[4.5]decane-3-carboxamide
7-(cyclohexylmethyl)-2-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decane
N-(2,6-difluorophenyl)-3-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)benzamide
N-[(2S,4R,6S)-2-benzyl-6-(1-methyl-1H-imidazol-5-yl)oxan-4-yl]acetamide
2-[(1-cyclooctylpiperidin-4-yl)oxy]-N-cyclopropyl-4-methoxybenzamide
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N,N-bis(prop-2-en-1-yl)piperidine-3-carboxamide
1-(thiophene-2-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
4-[1-(2,3-dihydro-1-benzofuran-7-carbonyl)pyrrolidin-2-yl]-3,5-dimethyl-1,2-oxazole
4-(4-methoxyphenoxymethyl)-1-[(2-methyl-1H-imidazol-4-yl)methyl]piperidine
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
N-[(1S)-1-carbamoyl-3-methylbutyl]-N'-(4-methylphenyl)propanediamide
N-[3-(2-methoxyphenyl)propyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
[(3R,4R)-1-(5-chloro-2-methylbenzoyl)-4-{[ethyl(methyl)amino]methyl}pyrrolidin-3-yl]methanol
(3aR,5R,6S,7aS)-2-[(2-methoxypyrimidin-5-yl)methyl]-octahydro-1H-isoindole-5,6-diol
(3S,4S)-1-(1H-1,3-benzodiazol-2-ylmethyl)-4-(4-fluorophenyl)piperidin-3-ol
4-[4-(4-fluorophenyl)benzoyl]-6-methoxy-1-[3-(2-oxopyrrolidin-1-yl)propyl]-1,4-diazepan-2-one
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl]methanol
3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-8-[4-(methylsulfanyl)benzoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[7-(pyridin-2-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-2,3-dihydro-1H-isoindole
3-[(3,3-difluoropyrrolidin-1-yl)methyl]-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
methyl 1-[2-hydroxy-3-(4-{[(prop-2-en-1-yl)amino]methyl}phenoxy)propyl]piperidine-4-carboxylate
2-chloro-N-({3,5-dimethoxy-4-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]benzene-1-sulfonamide
2-[4-(hydroxymethyl)-4-(3-phenylpropyl)piperidin-1-yl]pyridine-3-carboxamide
1-cyclopentyl-N3-methyl-N3-(2-methylpropyl)-4-oxo-N5-{[3-(trifluoromethoxy)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-3-propyl-1H-pyrazole-5-carboxamide
N4-[(3-propyl-1,2-oxazol-5-yl)methyl]-5,6,7,8-tetrahydroquinazoline-2,4-diamine
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)({2-phenylimidazo[1,2-a]pyridin-3-yl}methyl)amine
6-(2-chlorophenyl)-2-[(3S)-3-hydroxypyrrolidine-1-carbonyl]-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
5-[(3-hydroxypropyl)(naphthalen-1-ylmethyl)carbamoyl]-1H-imidazole-4-carboxylic acid
({4-ethyl-5-[1-(pyridine-3-sulfonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
1-[3-(2-oxo-1,2-dihydropyridin-1-yl)propanoyl]-3-propylpiperidine-3-carboxylic acid
N-[2-(1H-imidazol-1-yl)ethyl]-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-amine
2-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-N,N-dimethylaniline
4-(3-methylphenyl)-3-[1-(propan-2-yloxy)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(2-phenoxyethyl)-4-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperazine
1-{3-[4-(quinolin-2-yl)-1H-1,2,3-triazol-1-yl]propyl}pyrrolidin-2-one
2-(2-cyclopropylpyrimidin-5-yl)-4-(3,3-dimethylpyrrolidine-1-carbonyl)-8-methylquinoline
8-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
3-({[(2,4-difluorophenyl)methyl]amino}methyl)-3-hydroxy-1-(3-phenylpropyl)piperidin-2-one
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-(2-fluorophenyl)propanamide