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3-{imidazo[1,2-a]pyridin-2-yl}-5-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl]-1,2,4-oxadiazole
N-butyl-6-(2,5-dimethylfuran-3-yl)-N-ethyl-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
4-({4-methoxy-3-[2-(1-{2-[3-(trifluoromethyl)phenyl]acetyl}piperidin-2-yl)ethoxy]phenyl}methyl)piperazin-2-one
1-[(1S,5R)-6-(1,6-dimethyl-1H-indole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]({1-[(2-fluorophenyl)methyl]-2-methanesulfonyl-1H-imidazol-5-yl}methyl)methylamine
(2-{2-[1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
2-{1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]piperidin-2-yl}acetic acid
5-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidine-1-carbonyl]pyridine-2-carbonitrile
N-[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]-1-[2-(dimethylamino)ethyl]-6-oxopiperidine-3-carboxamide
7-[3-(3-hydroxy-3-methylbutyl)benzoyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}[3-(morpholin-4-yl)propyl]amine
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-methyl-N-[2-(oxan-2-yl)ethyl]-1,2-oxazole-3-carboxamide
ethyl 1-[6-(1-benzothiophen-3-yl)-3-{methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]carbamoyl}pyridin-2-yl]piperidine-3-carboxylate
1-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-3-(1-propyl-1H-1,2,3-triazol-4-yl)urea
4-ethyl-1-(4-methylpent-3-en-1-yl)-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(2R)-2-[(6-methoxypyrimidin-4-yl)amino]-3-phenylpropan-1-ol
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-1,9-dioxaspiro[5.5]undecan-4-amine
2-cyclopropyl-N-(1-methylpiperidin-4-yl)-6-oxo-N-(pyridin-4-ylmethyl)-1,6-dihydropyrimidine-5-carboxamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidine-4-carboxamide
[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl](methyl)[(5-methylthiophen-2-yl)methyl]amine
2-(3-{[2-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}phenoxy)acetamide
2-amino-7-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[(3-methoxyphenyl)methyl]-N-methyl-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
4-chloro-N,1-dimethyl-N-[1-(pyridin-3-yl)propyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
3-ethyl-3-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-1-[4-(oxan-2-ylmethoxy)phenyl]urea
N-(2-{7-[(2-chloro-3,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)pyridine-3-carboxamide
1-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl]-3-[4-(3-methylphenyl)piperazin-1-yl]propan-1-one
9-(1-methylpiperidine-2-carbonyl)-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-[1-(3-amino-1H-1,2,4-triazole-5-carbonyl)piperidin-4-yl]-4-benzyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-2-(4-phenylpiperidin-1-yl)acetamide
(3S,4R)-1-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
5-[2-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]-1,3,4-thiadiazol-2-amine
(1R,2R)-2-phenyl-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclopropane-1-carboxamide
N-[1,3-dihydroxy-2-(hydroxymethyl)propan-2-yl]-2,3-dihydro-1H-indene-1-carboxamide
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
2-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-amine
7-{[3-(dimethylamino)pyrrolidin-1-yl]sulfonyl}-N-ethyl-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
2-{3-oxo-9-[(2-phenylethyl)carbamoyl]-2,9-diazaspiro[5.5]undecan-2-yl}acetic acid
[(4-{[1-(2,3-dimethoxybenzoyl)piperidin-3-yl]methoxy}phenyl)methyl](methyl)(naphthalen-1-ylmethyl)amine
1-(1-benzothiophene-5-carbonyl)-4-[(3-methylpyridin-2-yl)methyl]piperazine
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-5-[(4-methylpiperidin-1-yl)methyl]furan-2-carboxamide
5-(4-chloro-2-methoxyphenoxymethyl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1,2-oxazole-3-carboxamide
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-3,5-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
N-(2-hydroxyethyl)-1-{1-[(4-methoxynaphthalen-1-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
2-(1-methyl-1H-pyrazol-3-yl)-1-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]piperidine
4-({[(2,4-dimethoxyphenyl)methyl]amino}methyl)-6,7-dimethyl-2H-chromen-2-one
4-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-methyl-5-propylpyrimidine
4-hydroxy-N-[2-(1H-imidazol-1-yl)propyl]-2-phenylpyrimidine-5-carboxamide
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}[1-(pyrimidin-4-yl)ethyl]amine