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2-(dimethylamino)-2-(3-fluorophenyl)-1-[4-(6-methylpyridin-2-yl)piperazin-1-yl]ethan-1-one
N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-(3-hydroxy-3-methylbut-1-yn-1-yl)benzamide
2-methyl-5-(1,2-oxazol-5-yl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}benzene-1-sulfonamide
1-(2-hydroxyethyl)-N-[2-(2-oxo-1,3-oxazolidin-3-yl)phenyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carboxamide
4-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-4H-1,2,4-triazole
4-{4-[(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)amino]piperidin-1-yl}-N-[(3S)-2-oxoazepan-3-yl]benzamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-5-methyl-4-[(pyridin-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
2-[2-(1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}piperidin-3-yl)-1H-imidazol-1-yl]acetamide
[2-(3-{3-[cyclohexyl(methyl)amino]propyl}-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl)-2-oxoethyl]urea
N-cyclopropyl-N-[(4-ethoxyphenyl)methyl]-2-[ethyl(methyl)amino]propanamide
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-propyl-3-(1H-pyrazol-1-yl)benzamide
2-[4-(1H-indole-2-carbonyl)-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl]ethan-1-ol
2-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-ol
methyl 6-(oxolane-2-carbonyl)-2-[(2-phenylethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-{[7-methoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)-4-(1H-pyrazol-1-yl)benzamide
1-[6-methyl-3-({methyl[(2-methylpyridin-4-yl)methyl]amino}methyl)quinolin-2-yl]piperidin-3-ol
1-ethyl-8-[(3-methylthiophen-2-yl)methyl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-(3-acetyl-2-fluorophenyl)thiophene-2-carboxamide
(2S,4S)-1-[(4-chlorophenyl)methyl]-N,N-diethyl-4-{[(4-phenylphenyl)methyl]amino}pyrrolidine-2-carboxamide
8-{[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]amino}-2,6-dimethyloctan-2-ol
5-(4-chlorophenyl)-3-[4-(2-methoxyethyl)piperazin-1-yl]-1,2,4-triazine
5-[1-(1-methyl-1H-pyrazole-5-carbonyl)pyrrolidin-2-yl]-N-(1,2,3-thiadiazol-5-yl)thiophene-2-carboxamide
5-[(dimethylsulfamoyl)amino]-1-methyl-2-(2-methylpropyl)-N-[(3-methylpyridin-2-yl)methyl]-1H-1,3-benzodiazole-7-carboxamide
N-(butan-2-yl)-2-methyl-N-(pyridin-2-ylmethyl)-3-[(pyridin-3-ylmethyl)amino]benzamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N,2-dimethyl-1H-pyrrole-3-carboxamide
1-{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}piperidine-3-carboxamide
1-[(3-methyl-1-benzofuran-2-yl)methyl]-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
(1R,3S)-3-(2-aminoethoxy)-7-{[3-(cyclopentyloxy)phenyl]methyl}-7-azaspiro[3.5]nonan-1-ol
1-[1-(1H-imidazol-4-ylmethyl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine
(2S)-1-[6-(3-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]pyrrolidine-2-carboxamide
N-(3-chloro-4-fluorophenyl)-3-{1-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]piperidin-4-yl}propanamide
2-{4-[4-(4-fluorophenyl)piperazine-1-carbonyl]-5-(propan-2-yl)-1H-pyrazol-1-yl}-4-(thiophen-2-yl)pyrimidine
1-cyclohexyl-4-[5-(3-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]piperazine
5-acetamido-2-ethyl-1-(pyridin-3-ylmethyl)-N-{spiro[2.5]octan-1-ylmethyl}-1H-1,3-benzodiazole-7-carboxamide
{[2-(methoxymethyl)pyrimidin-5-yl]methyl}[(2-methoxyphenyl)methyl](pyridin-3-ylmethyl)amine
3-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1-(2-methyl-5-sulfamoylphenyl)urea
N-[(1-ethyl-1H-imidazol-5-yl)methyl]-2,6,8-trimethylquinoline-4-carboxamide
(2R)-4-[(4-cyclopentylpyrimidin-2-yl)amino]-2-methylbutan-1-ol
N-(1-{7-[(2,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)furan-3-carboxamide
N-(2,3-dihydroxypropyl)-N-methyl-4-(5-methylfuran-2-yl)benzamide
1-{1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]piperidin-4-yl}-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
methyl (2S,4S)-1-[(2-chloro-6-fluorophenyl)methyl]-4-{2-[4-(trifluoromethyl)phenyl]benzamido}pyrrolidine-2-carboxylate
3-cyclopentyl-5-[(4-fluorophenyl)methyl]-5-{1-[(4-hydroxy-3-methoxyphenyl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
4-[5-(2,3-dimethoxyphenyl)-3-(furan-2-yl)-1H-1,2,4-triazol-1-yl]-1-methylpiperidine
4-(2-phenylethyl)-1-[1-(1H-pyrazol-1-yl)propan-2-yl]-1H-1,2,3-triazole
9-[2,2-dimethyl-1-(thiophen-2-yl)cyclopropanecarbonyl]-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-[(2E)-3-phenylprop-2-en-1-yl]-decahydro-1,6-naphthyridin-2-one
2-[(4aS,7aR)-4-(cyclopropylmethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carbonyl]benzonitrile
N-{1-[1-(azetidine-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-chlorobenzamide
2-(azepan-1-yl)-1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]ethan-1-one