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1-{[2-(4-fluorophenyl)-6-methylquinolin-3-yl]methyl}-2-methyl-1,4-diazepan-5-one
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-(1H-indazol-1-yl)acetamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2-cyclopropyl-4-hydroxy-N-methylpyrimidine-5-carboxamide
methyl 5-[(3-hydroxy-3-methylbutan-2-yl)amino]-3-(2-methoxyacetamido)-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1,5-bis(2-methylpropyl)-1H,4H-pyrazolo[3,4-d]imidazole
N-[(3S,4R)-1-(furan-2-ylmethyl)-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
1-[3-({10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)propyl]piperidin-4-ol
1-(pyridin-4-yl)-4-{4H-thieno[3,2-b]pyrrole-5-carbonyl}-1,4-diazepan-6-ol
N-(2-fluorophenyl)-4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
4-methyl-6-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
1-(cyclohexylmethyl)-N-(furan-3-ylmethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
ethyl 4-(5-cyclopropyl-3-methyl-1H-pyrazole-4-carbonyl)piperazine-1-carboxylate
N-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1-[(4-methylphenyl)amino]cyclopentane-1-carboxamide
1-methanesulfonyl-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]piperidin-4-amine
N-(carbamoylmethyl)-2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-(3-methyl-4-{3-oxo-2,8-diazaspiro[4.5]decane-8-carbonyl}phenyl)acetamide
N-cyclopropyl-1-[1-(3-methylbutanoyl)piperidin-4-yl]piperidine-3-carboxamide
2-methyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}imidazo[1,2-a]pyrimidine-3-carboxamide
8-methyl-5-{5-methylthieno[2,3-d]pyrimidin-4-yl}quinoline
1-{5-acetyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-3-(1-methyl-1H-pyrrol-2-yl)propan-1-one
2-[(4-chlorophenyl)methyl]-8-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[4.5]decan-3-one
1-(3-{[6-(2-ethylpiperidine-1-carbonyl)-5-methylthieno[2,3-d]pyrimidin-4-yl]amino}propyl)pyrrolidin-2-one
N-[(4-chlorophenyl)methyl]-3-ethyl-N-(3-hydroxypropyl)-4-methyl-1H-pyrazole-5-carboxamide
3-[5-(5-methyl-2H-1,2,3-triazol-4-yl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
2-amino-6-cyclobutyl-4-[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]pyridine-3-carbonitrile
3-[(3S,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-(2-methylpropyl)piperidin-3-yl]-N-(4-methylphenyl)propanamide
2-methoxy-N-{1-[1-(3-methoxybenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-phenylacetamide
3-(1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-4-methyl-1,2,5-oxadiazole
9-({2-[3-(dimethylamino)propoxy]phenyl}methyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
4-oxo-4-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]butanamide
4-[(3-fluorophenyl)methyl]-9-methoxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[3-cyclopropyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-4-(1H-pyrrol-1-yl)phenol
N-{3-methyl-1-[7-(thiophen-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]butyl}pyridine-3-carboxamide
2-{4-[(7-chloro-3-methyl-1H-indol-2-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
4-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-ylmethyl]-5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazole
1-(3-oxo-3-{3-[4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}propyl)pyrrolidin-2-one
1-{5-[(4-ethylphenyl)methyl]-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidin-3-ol
methyl({[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})(pyridin-3-ylmethyl)amine
2-[3-cyclopentyl-5-(5-cyclopropyl-1,3-oxazol-4-yl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
4-{5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-yl}morpholine
N-ethyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-(3-methyl-2-oxo-1,2-dihydroquinoxalin-1-yl)acetamide
3-[1-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-4-yl]-N-[2-(dimethylamino)ethyl]propanamide
N-{4-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]-2-methoxyphenyl}acetamide
N-cyclopentyl-2-(4,5-dimethyl-2-oxo-2,3-dihydro-1,3-oxazol-3-yl)butanamide
methyl (2S,4R)-1-[(2-chlorophenyl)methyl]-4-(2-phenylbenzamido)pyrrolidine-2-carboxylate
(2S,4S)-4-amino-N-methyl-1-(4-propylpyrimidine-5-carbonyl)pyrrolidine-2-carboxamide
1-(3-ethyl-1,2-oxazole-5-carbonyl)-4-(pyridin-4-yl)piperazine
N-(2,3-dihydro-1H-inden-1-yl)-5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
N-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl)({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)amine