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2-cyclopentyl-9-{[2-(ethylamino)pyrimidin-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
2-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-N-(4-methylphenyl)-2-oxoacetamide
{2-[methyl({[1-(piperidin-1-yl)cyclohexyl]methyl})amino]-1,3-thiazol-4-yl}methanol
(2S)-2-amino-1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-phenylethan-1-one
2-methyl-7-[1-(pyrazine-2-carbonyl)piperidin-4-yl]-2,7-diazaspiro[4.5]decane
1-[1-(1-benzothiophen-2-ylmethyl)piperidin-3-yl]-N-(3-hydroxypropyl)-1H-1,2,3-triazole-4-carboxamide
5-chloro-N-methyl-2-oxo-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1,2-dihydropyridine-3-carboxamide
1,4-dimethyl 2-[(1-{4-[2-oxo-2-(pyrrolidin-1-yl)ethyl]phenyl}piperidin-4-yl)amino]butanedioate
1-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-methyl-3-(1H-pyrazol-1-yl)propan-1-one
3-{[(1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidin-4-yl)oxy]methyl}pyridine
1-[2-(4-methoxyphenyl)ethyl]-3,8-dimethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-cyclopropanecarbonyl-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
2-(dimethylamino)-2-(3-methylphenyl)-N-[2-(1H-pyrrol-1-yl)ethyl]acetamide
methyl 4-[(4-{[3-(1,3-thiazol-4-yl)phenyl]carbamoyl}piperidin-1-yl)methyl]benzoate
5-[1-(2-amino-6-methylpyrimidin-4-yl)piperidin-4-yl]-5-(pyridin-2-yl)imidazolidine-2,4-dione
{1-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]-3-(3-methylbut-2-en-1-yl)piperidin-3-yl}methanol
8-chloro-2-(thiomorpholin-4-ylmethyl)quinoline
2-{1-[(2-ethoxyphenyl)methyl]-4-[(4-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
2-(4-chloro-3-methyl-1H-pyrazol-1-yl)-1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
3-[3-(dimethylamino)pyrazin-2-yl]-5-[2-(piperidin-2-yl)ethyl]phenol
5-[3-(4-chlorophenyl)propyl]-3-methyl-1,2,4-oxadiazole
N,5-dimethyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-[4-(5-methyl-4-{[1-(thiophen-2-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carbonyl)piperazin-1-yl]ethan-1-ol
4-{4-[1-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)-1H-imidazol-2-yl]-1H-1,2,3-triazol-1-yl}piperidine
ethyl 2-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]-1,3-oxazole-4-carboxylate
N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]-2-(morpholin-3-yl)acetamide
cyclohexyl[4-(1-ethylpiperidine-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methanol
methyl 5-{[(3-ethoxy-4-methoxyphenyl)methyl]amino}-3-(oxolane-3-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-[1-cyclohexyl-4-(1H-indol-3-ylmethyl)piperazin-2-yl]ethan-1-ol
N-[(1s,4s)-4-aminocyclohexyl]-2,3-dihydro-1H-indene-1-carboxamide
4-(2,4-dioxoimidazolidin-1-yl)-N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]benzamide
2-methoxy-N-(2-{2-methyl-3-oxo-2,8-diazaspiro[4.5]decane-8-carbonyl}phenyl)acetamide
2-(3-fluorophenoxymethyl)-N-methyl-N-(3-methylbutan-2-yl)-1,3-oxazole-4-carboxamide
1-cyclobutanecarbonyl-4-[4-(propan-2-yl)pyrimidin-2-yl]-1,4-diazepane
6-(2-methylpropyl)-2-oxo-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}-1,2-dihydropyrimidine-4-carboxamide
(2S,4S)-4-amino-1-(2-benzyl-1,3-thiazole-4-carbonyl)-N-methylpyrrolidine-2-carboxamide
11-{[(2,6-difluorophenyl)methyl]amino}-4-[2-(pyridin-2-yl)ethyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-(3-methylpentan-3-yl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-methyl-2-[1-methyl-3-(1-phenylcyclopropyl)-1H-1,2,4-triazol-5-yl]azepane
4-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-2-amine
2-(3-{[(6-hydroxy-6-methylheptan-2-yl)amino]methyl}-2-methyl-1H-indol-1-yl)acetamide
3-hydroxy-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]propanamide
N-{2-[1-(5-fluoro-2-methylbenzenesulfonyl)piperidin-2-yl]ethyl}acetamide
methyl (2R)-2-({2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazol-4-yl}formamido)propanoate
(1R,5R)-6-{[6-(dimethylamino)pyridin-3-yl]methyl}-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
6-chloro-4-(2,4-dimethyl-1,4-diazepane-1-carbonyl)-2-(1-methyl-1H-pyrazol-4-yl)quinoline
4-[3-(azocane-1-carbonyl)phenoxy]-N,N-dimethylpiperidine-1-sulfonamide
2-ethoxy-6-({4-[4-(naphthalen-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol
(4S)-4-(methoxymethyl)-1-(6-methoxypyrimidin-4-yl)-3,3-dimethylpiperidin-4-ol