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5-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1H-1,3-benzodiazole
1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(piperidine-1-carbonyl)piperidine
N-ethyl-6-{4-[1-(2-methylpropyl)piperidin-4-yl]piperazin-1-yl}pyridine-3-carboxamide
3-[(3-ethoxyphenyl)methyl]-9-methoxy-N-[(2-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
6-[3-(2-methoxyphenoxy)propyl]pyridine-2-carbonitrile
2-[4-(1-benzofuran-2-ylmethyl)-1-[(2-methylphenyl)methyl]piperazin-2-yl]ethan-1-ol
2-[1-cyclopentyl-4-(pyridin-3-ylmethyl)piperazin-2-yl]ethan-1-ol
5-[(2-chloro-6-fluorophenyl)methyl]-8-ethoxy-2-(3,4,5-trimethoxyphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
N-[3-(3-chlorophenyl)phenyl]-1-(oxolane-2-carbonyl)piperidine-4-carboxamide
N-(pentan-3-yl)-N-(2-phenylethyl)-6-azaspiro[2.5]octane-1-carboxamide
3-(3-cyclopentyl-1-methyl-1H-1,2,4-triazol-5-yl)-N,N-dimethylpropanamide
(4aS,7aR)-1-(1H-imidazol-4-ylmethyl)-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[4-(2-chlorophenyl)piperidin-4-yl]-N-(furan-2-ylmethyl)-N-methylpyrimidin-2-amine
4-(2-acetylbenzoyl)-6-[(3-fluorophenyl)methoxy]-1-(2-methylpropyl)-1,4-diazepan-2-one
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-2-(2,2,3,3-tetrafluoropropoxy)acetamide
N-{[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-3-yl]methyl}-2,2-dimethylpropanamide
4-methyl-N-[3-({5-methylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propyl]benzene-1-sulfonamide
1-(4-{[(5-methyl-1H-pyrazol-3-yl)methyl]amino}-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
5-(oxolan-2-yl)-3-[2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)ethyl]-1,2,4-oxadiazole
ethyl 1-[1-(cyclohexylmethyl)-6-oxopiperidine-3-carbonyl]piperidine-4-carboxylate
(1R,7S)-3-(2-methoxyethyl)-N-methyl-4-oxo-N-(1,3-thiazol-2-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
4-{2-methoxy-4-[3-(methoxymethyl)piperidine-1-carbonyl]phenoxy}-1-methylpiperidine
4-(3-fluoropyridin-4-yl)-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
6-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-N-ethylpyridine-3-carboxamide
6-[(3-methoxyphenyl)methoxy]-1-(pyridin-2-ylmethyl)-4-(1,3-thiazole-5-carbonyl)-1,4-diazepan-2-one
[2-methoxy-2-(thiophen-2-yl)ethyl]({[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl})amine
N-methyl-2-[3-methyl-5-oxo-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-[1-(1,2-oxazol-3-yl)ethyl]acetamide
1-[(5-ethylfuran-2-yl)methyl]-4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
(3R,4R)-1-[2-(benzyloxy)ethyl]-4-cyclobutyl-3-methylpiperidin-4-ol
4-[(4-phenyl-4H-1,2,4-triazol-3-yl)methyl]phenol
(5S,9aS,9bS)-5-(5-chloro-2,3-dimethoxyphenyl)-2-(pyridin-3-ylmethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
methyl 1-(2-methoxyethyl)-5-{[4-(4-methoxyphenyl)butan-2-yl]amino}-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-5-(4-methoxyphenyl)furan-2-carboxamide
methyl 2-[(oxolan-2-ylmethyl)sulfamoyl]-6-[(2,4,5-trimethylphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-[4-(2-chlorophenyl)piperidin-4-yl]-N,N-dimethylpyrimidin-2-amine
1-[2-(dimethylamino)ethyl]-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-6-oxopiperidine-3-carboxamide
N-[(4-chlorophenyl)(pyridin-4-yl)methyl]-6-oxo-1,6-dihydropyridine-2-carboxamide
5-butyl-1-(2-methoxyphenyl)-4-(5-methyl-1,3-oxazole-4-carbonyl)piperazin-2-one
ethyl 4-(3-phenylpropyl)-1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]piperidine-4-carboxylate
N,N-dimethyl-3-[(3-phenylpiperidin-1-yl)sulfonyl]benzamide
1-ethyl-5-({[(propan-2-yl)carbamoyl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-methyl-2-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonan-3-yl]-N-(2-phenylethyl)acetamide
2-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
5-(2-chlorophenyl)-N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}furan-2-carboxamide
N-({1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]piperidin-3-yl}methyl)-1-phenylmethanesulfonamide
N,N-dimethyl-5-{[5-methyl-5-(4-methylpent-3-en-1-yl)-2-oxopiperidin-1-yl]methyl}furan-2-carboxamide
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidine
2-methyl-9-(4-methylpiperazine-1-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecane
N-cyclopropyl-3-{1-[3-(trifluoromethyl)benzenesulfonyl]piperidin-4-yl}propanamide
3-{[methyl({[2-(methylamino)pyrimidin-5-yl]methyl})amino]methyl}piperidin-3-ol