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N-(dimethyl-1,2-oxazol-4-yl)-4-{[3-(N-ethylacetamido)pyrrolidin-1-yl]methyl}benzamide
3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-[2-(3-methylpyridin-2-yl)ethyl]propanamide
2-{[3-(2-hydroxyethyl)-4-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-1-yl]methyl}-5-methoxyphenol
1-[1-(3-fluoro-4-methoxyphenyl)ethyl]-3-(2,4,6-trimethylpyridin-3-yl)urea
1-{2-[6-hydroxy-4-(pyridin-4-yl)-1,4-diazepan-1-yl]-2-oxoethyl}pyrrolidin-2-one
2-{4-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-1,4-diazepan-1-yl}-1,3-benzothiazole
(3R,4R)-4-{methyl[2-(pyridin-2-yl)ethyl]amino}-1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-3-ol
4-[3-(1H-imidazol-1-yl)propyl]-2-(6-methoxynaphthalen-2-yl)morpholine
3-[2-(methylsulfanyl)benzoyl]-1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperidine
2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(1r,4r)-4-hydroxycyclohexyl]acetamide
1-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(methylamino)ethan-1-one
N-[3-(6-methyl-1,3-benzoxazol-2-yl)propyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
3-[5-({3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}methyl)-1,3,4-oxadiazol-2-yl]pyridine
N-(1,4-dioxan-2-ylmethyl)-N-methyl-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
5-(1-ethylpyrrolidine-3-carbonyl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
[2-ethoxy-5-({1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}methyl)phenyl]methanol
2-[(3,5-difluorophenyl)methyl]-8-(pyridine-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
2-[(1-butyl-2-cyclobutylmethanesulfonyl-1H-imidazol-5-yl)methyl]-1,2-oxazolidine
(3R,4R)-4-(hydroxymethyl)-1-(quinolin-2-ylmethyl)piperidin-3-ol
4-{3-[3-(dimethylamino)piperidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
2-{[1-(cyclohexylmethyl)piperidin-4-yl]oxy}-N-cyclopropyl-4-methoxybenzamide
1-[5-(2,3-dimethylphenoxymethyl)-1H-1,2,4-triazol-1-yl]butan-2-ol
1-{1-azabicyclo[2.2.2]octan-3-yl}-3-[5-(5-ethyl-1,3,4-oxadiazol-2-yl)-2-methoxyphenyl]urea
methyl({[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl})(propan-2-yl)amine
3-(1-methyl-1H-pyrrol-2-yl)-N-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]-1H-pyrazole-5-carboxamide
4-[3-(2,3-dihydro-1H-isoindole-2-carbonyl)phenyl]-2-methylbutan-2-ol
6-[(diethylamino)methyl]-N-(2-methoxy-5-methylphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-[2-(dimethylamino)ethyl]-N-[(5-methylthiophen-2-yl)methyl]-2-(pyrrolidin-3-yl)acetamide
(1R,5R)-6-[2-(2-methoxy-4-methylphenoxy)ethyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
3-[1-(2H-1,3-benzodioxol-4-ylmethyl)piperidin-3-yl]-N-[(2,4-dimethoxyphenyl)methyl]propanamide
5-(2-chloro-4-methoxyphenoxymethyl)-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-1,2-oxazole-3-carboxamide
5-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidine-1-carbonyl]pyrazin-2-ol
7-[(2-methylprop-2-en-1-yl)oxy]-4-[2-(methylsulfanyl)ethyl]-1,2,3,4-tetrahydroquinolin-2-one
1-[1'-(3-fluorobenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-N-[(4-fluorophenyl)methyl]-N-methylpyridin-2-amine
(2S,4S)-4-amino-N-ethyl-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]pyrrolidine-2-carboxamide
1,3-dimethyl-2,6-dioxo-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-({[5-(2-cyanophenyl)furan-2-yl]methyl}(methyl)amino)-N,N-dimethylpropanamide
N-{3-[(furan-2-ylmethyl)sulfanyl]propyl}-4-(trifluoromethyl)pyrimidin-2-amine
{4-[({[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)methyl]oxan-4-yl}methanol
[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]({[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl})methylamine
4-{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-2-ethyl-1-(propan-2-yl)piperazine
N-[(1S,2R)-1-hydroxy-1-(4-hydroxyphenyl)propan-2-yl]-4-(piperidin-1-yl)butanamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(2-methoxypyrimidine-5-carbonyl)piperidin-3-ol
3-benzyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
[1-(2-methoxyphenyl)ethyl](methyl)[(4-methyl-1H-imidazol-5-yl)methyl]amine
N-(2,3-dihydro-1H-inden-2-yl)-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
N-{1-[5-(3-methoxyphenyl)furan-2-carbonyl]piperidin-3-yl}acetamide
N-{2-[(2R)-2-aminopropanoyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}-4-(trifluoromethyl)benzamide
N-cyclohexyl-2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide