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N-[2-(dimethylamino)ethyl]-N-(oxolan-2-ylmethyl)-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(1,4-dithiepan-6-yl)pyrrolidine-3-carboxylic acid
4-benzyl-1-(1-methylpiperidin-4-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-3-(furan-2-yl)propanamide
1-[4-(2-{3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl}-2-oxoethyl)phenyl]imidazolidin-2-one
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-3-(2-phenylethyl)-1,2-oxazole-5-carboxamide
1-(2,4-difluorophenyl)-5-(5-methoxypentyl)-1H-1,2,4-triazole
methyl 3-(furan-2-amido)-1-(2-methoxyethyl)-5-[(4-phenylbutan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-({9-oxo-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)benzonitrile
2-[3-(1-cyclohexyl-1H-1,2,3-triazol-4-yl)phenoxymethyl]pyridine
4-(2H-1,3-benzodioxol-5-yl)-3-(methoxymethyl)-1-[2-oxo-2-(pyrrolidin-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
14-(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)-5-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
1-[1-(3-phenylphenyl)piperidin-4-yl]piperidine-4-carbonitrile
methyl 6-(naphthalen-1-ylmethyl)-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-1-[(2R,6S)-2,6-dimethylmorpholin-4-yl]ethan-1-one
4-(2-chloro-4,5-difluorobenzoyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-8-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
6-(2-methoxypyrimidin-5-yl)-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(methylsulfanyl)ethan-1-one
4-(2-ethylpyridine-4-carbonyl)-1-(2-methoxyphenyl)piperazin-2-one
ethyl 4-(3-phenylpropyl)-1-(thiophene-3-sulfonyl)piperidine-4-carboxylate
4-({1-[(2-butyl-1H-imidazol-4-yl)methyl]piperidin-4-yl}oxy)-3-chloro-N-(2-methoxyethyl)benzamide
6-[(3-methoxyphenyl)methoxy]-1-(2-methylpropyl)-4-(1,3-thiazole-5-carbonyl)-1,4-diazepan-2-one
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
2-methyl-6-(piperidin-4-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrimidin-4-amine
1-[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]-3-(pyridin-2-yl)propan-1-one
1-methyl-2-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]azepane
1-{[2-(butan-2-ylsulfanyl)pyrimidin-5-yl]methyl}-4-(pyridin-3-yl)piperidin-4-ol
1,3-dimethyl-N-[(5-methylpyrazin-2-yl)methyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
ethyl 4-[1-(2-cyclooctyl-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl)piperidine-4-amido]piperidine-1-carboxylate
2-{4-[4-(ethylamino)pyrimidin-2-yl]piperazin-1-yl}phenol
(1s,4s)-4-[4-(4-phenyl-1,4-diazepane-1-carbonyl)-1H-1,2,3-triazol-1-yl]cyclohexan-1-amine
5-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-2-methyl-4-phenylpyrimidine
2-(2-methoxyethyl)-N-[2-(pyridin-3-yloxy)propyl]-1,3-benzoxazole-6-carboxamide
N-{[7-({4-[methyl(phenyl)amino]phenyl}methyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-2-phenylacetamide
2-(4-propanoylphenoxy)-N-[2-(pyridin-3-yloxy)propyl]acetamide
7-(2-methoxyethyl)-2-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
2-methanesulfonyl-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-6-one
1-cyclopentyl-4-({[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]amino}methyl)pyrrolidin-2-one
(4aS,8aS)-2-[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-decahydroisoquinolin-4a-ol
6-(benzyloxy)-1-(2-methylpropyl)-4-(thiolan-3-yl)-1,4-diazepan-2-one
1-[(4-methoxyphenyl)methyl]-4-(3-methoxypyrazin-2-yl)piperazin-2-one
2-methoxy-6-({methyl[1-(pyridin-2-yl)propan-2-yl]amino}methyl)phenol
N-{4-[({2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}carbamoyl)methyl]phenyl}butanamide
N-[2-(1H-indol-3-yl)ethyl]-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
6-(benzyloxy)-1-cyclohexyl-4-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-1,4-diazepan-2-one
8-benzoyl-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
1-{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-methoxypiperidine
4-[5-(3-chlorophenyl)-4-phenyl-1H-imidazol-1-yl]-1-methylpiperidine
1,2-dimethyl-4-[(2-phenyl-1H-imidazol-4-yl)methyl]piperazine