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2-(3-hydroxypropyl)-9-[(2-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-butyl-N-[(3-methoxyphenyl)methyl]-1-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
(2R)-1-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-2-cyclohexyl-2-hydroxyethan-1-one
7-(2-methoxyacetamido)-N-[(1R)-1-(4-methoxyphenyl)ethyl]-1-methyl-2-(pyridin-3-yl)-1H-1,3-benzodiazole-5-carboxamide
N-cyclobutyl-7-(cyclopropylmethyl)-8-oxo-6-(thiophen-2-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2,4-dimethyl-N-[(4-sulfamoylphenyl)methyl]pyrimidine-5-carboxamide
[(3R,4R)-1-[(3-chloro-4-fluorophenyl)methyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-[3-(1H-indol-1-yl)propyl]-2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)thiophene-2-sulfonamide
(5S,9aS,9bS)-5-(2,1,3-benzoxadiazol-4-yl)-2-(2-phenylethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
8-[(3-fluoro-4-methylphenyl)methyl]-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
1-(3-{[(8-fluoro-4-hydroxyquinolin-2-yl)methyl]amino}propyl)pyrrolidin-2-one
1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-2-(thiophen-3-yl)ethan-1-one
methyl 3-chloro-4-[(3-acetamidopyrrolidine-1-carbonyl)amino]benzoate
{[(3S,4R)-1-(2,4-difluorobenzoyl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
4-{[2-(difluoromethoxy)phenyl]methyl}-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-{[1-(hydroxymethyl)cyclobutyl]methyl}-N-methylacetamide
diethyl({2-ethyl-5-[2-(trifluoromethyl)morpholine-4-carbonyl]furan-3-yl}methyl)amine
N-(pyrazin-2-yl)-2-{[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]amino}acetamide
N-methyl-N-phenyl-2-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
N,N-diethyl-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
(3aS,6aS)-2-acetyl-5-[(4-chlorophenyl)methanesulfonyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(3R,5S)-1-cyclobutanecarbonyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]pyrazine-2-carboxamide
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-3-(3-methoxyphenyl)-N-methyl-1H-pyrazole-4-carboxamide
ethyl 4-{[2-methyl-3-(1H-pyrrol-1-yl)phenyl]carbamoyl}piperazine-1-carboxylate
N,6-dimethyl-4-(4-methyl-1H-imidazol-5-yl)-2-oxo-N-[(5-propyl-1H-pyrazol-3-yl)methyl]-1,2,3,4-tetrahydropyrimidine-5-carboxamide
5-chloro-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]thiophene-2-carboxamide
2-(4-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}piperazin-1-yl)-N,N-dimethylacetamide
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-1-ethyl-1H-pyrazole-5-carboxamide
9-[(5-fluoro-2-methoxyphenyl)methyl]-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(2-{1-[(6-fluoroquinolin-2-yl)methyl]piperidin-2-yl}ethyl)pyrrolidin-2-one
1-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-methyl-N-[3-(phenylsulfanyl)propyl]acetamide
methyl 4-{[3-(2-hydroxyethyl)-4-(thiophen-3-ylmethyl)piperazin-1-yl]methyl}benzoate
3-(hydroxymethyl)-3-(2-methoxyethyl)-N-(2-phenylethyl)piperidine-1-carboxamide
1-[4-(furan-2-yl)pyrimidin-2-yl]-N,5-dimethyl-N-(2-phenylethyl)-1H-pyrazole-4-carboxamide
4-[(1S,3R)-3-aminocyclopentaneamido]-2-(pyrrolidin-1-yl)benzamide
2-methanesulfonyl-N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]acetamide
1-[7-(1-benzothiophen-3-yl)-9-[2-(pyridin-2-yl)ethoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methoxyethan-1-one
ethyl 1-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-imidazole-2-carboxylate
5-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(but-3-enoyl)-N-[3-(1H-indol-2-yl)phenyl]piperidine-4-carboxamide
4-ethyl-3-{[3-(2-methoxyethyl)-1-[(4-methylphenyl)methyl]-1H-1,2,4-triazol-5-yl]methyl}piperazin-2-one
3-{[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}phenol
N-cyclopropyl-N-({3-[(1-methoxypropan-2-yl)oxy]phenyl}methyl)thiophene-2-carboxamide
3-(5-{3-[5-(4-fluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]propyl}-1,2,4-oxadiazol-3-yl)pyridazine
3-{[(2S)-1-hydroxypropan-2-yl]sulfamoyl}-N-[3-(pyridin-3-yl)propyl]benzamide
(4aS,8aR)-6-[(3-methyl-1,2-oxazol-5-yl)methyl]-1-(2-phenylethyl)-decahydro-1,6-naphthyridin-2-one
N-[3-(1H-indol-1-yl)propyl]-2,4-dimethylpyrimidine-5-carboxamide
N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N,4,6-trimethylpyrimidin-2-amine