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4-(2,6-dimethylpyridin-3-yl)-N-(pyridin-4-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]acetamide
N-methyl-N-(pyrimidin-4-ylmethyl)-5-[3-(trifluoromethyl)phenoxymethyl]-1H-pyrazole-3-carboxamide
(2S,4S)-4-amino-1-[3-(1,3-benzothiazol-2-yl)propanoyl]-N-ethylpyrrolidine-2-carboxamide
N-{[(2S,4S)-4-fluoro-1-(1H-indazole-3-carbonyl)pyrrolidin-2-yl]methyl}piperidine-1-carboxamide
2-({[(1R,2R)-2-hydroxycyclohexyl]methyl}amino)-N-[2-methyl-6-(propan-2-yl)phenyl]acetamide
N-(cyclopropylmethyl)-2-(2-fluorophenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[1-(pyridin-3-yl)propan-2-yl]benzamide
4-(1H-1,3-benzodiazol-1-yl)-1-(5-cyanopyridin-2-yl)piperidine-4-carboxylic acid
2-amino-N-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)acetamide
N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-2-(1H-pyrazol-1-yl)butanamide
N-[(2R,3R)-1'-[(5-ethylfuran-2-yl)methyl]-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]benzamide
5-(2-{[(4-methoxyphenyl)methyl]amino}ethyl)-1-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]pyrrolidin-2-one
3-(2H-1,3-benzodioxol-5-ylmethyl)-6-fluoro-3,4-dihydroquinazolin-4-one
N-benzyl-1-(5-methoxy-1H-indole-2-carbonyl)-N-methylpiperidin-3-amine
N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-2-propyl-1,3-thiazole-4-carboxamide
2-amino-4-(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
1-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-3-methyl-3-[3-(1-methyl-1H-pyrazol-4-yl)propyl]urea
5-[bis(prop-2-en-1-yl)amino]-1-methyl-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
7-chloro-N,3,5-trimethyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-1-benzofuran-2-carboxamide
1-(3-fluorophenyl)-3-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}urea
(3aS,6aS)-2-acetyl-5-[4-(trifluoromethyl)pyrimidin-2-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
9-[5-(propan-2-yl)pyrimidin-4-yl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[2-oxo-8-(quinoxaline-5-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-3-yl]acetic acid
2-[(4-acetyl-6-hydroxy-1,4-diazepan-1-yl)methyl]-6-fluoro-1,4-dihydroquinolin-4-one
4-[2-(2-fluorophenyl)ethyl]-3-(furan-2-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(4aS,7aR)-1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-(2-methoxyacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3R,5S)-5-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}pyrrolidin-3-amine
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-6-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
[(3R,4R)-4-[(4-ethylpiperazin-1-yl)methyl]-1-(9H-purin-6-yl)pyrrolidin-3-yl]methanol
N-[(3-methylpyridin-2-yl)methyl]-3-(1H-pyrazol-4-yl)benzamide
2-{4-methyl-1-[5-(morpholine-4-carbonyl)furan-2-yl]-1H-1,3-benzodiazol-2-yl}ethan-1-ol
3-(1H-indazol-5-yl)-1-[3-(morpholin-4-yl)propyl]urea
(3aS,6aR)-3-(pyridin-2-ylmethyl)-5-(pyrrolidine-1-sulfonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
methyl 3-[(3S,4R)-1-[(2,4-dimethoxy-3-methylphenyl)methyl]-4-(dimethylamino)piperidin-3-yl]propanoate
2-[4-(2H-1,3-benzodioxol-5-yl)-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-(thiolan-3-yl)acetamide
2-{1-[(3-methoxyphenyl)methyl]-4-[(1-methyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
7-[(4-fluorophenyl)methyl]-2-[(5-methylfuran-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
(1R,2S)-N-butyl-2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-carbonyl]cyclohexane-1-carboxamide
N-{3-[3-(1H-imidazol-2-yl)piperidin-1-yl]-3-oxopropyl}-3-methoxybenzamide
2-methyl-N-{1-oxaspiro[4.4]nonan-3-yl}imidazo[1,2-a]pyridine-6-carboxamide
4-(3-hydroxy-3-methylbutyl)-N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}benzamide
3-{1-[(3,4-dimethoxyphenyl)methyl]-3-methyl-1H-pyrazol-5-yl}-1-[(5-methyl-1,2-oxazol-3-yl)methyl]urea
1-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)urea
(1S,3R)-3-amino-N-{[5-(2-chlorophenyl)furan-2-yl]methyl}cyclopentane-1-carboxamide
2-(1-{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}pyrrolidin-2-yl)pyridine
5-[4-methyl-2-(1H-pyrazol-1-yl)phenyl]pyrazin-2-amine
N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-(pyridin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-[5-(4,4-diphenylpiperidine-1-carbonyl)-1H-pyrazol-3-yl]ethan-1-one