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3-(3-hydroxy-3-methylbutyl)-N-{[1-(pyrrolidin-1-yl)cyclopentyl]methyl}benzamide
N-(piperidin-4-ylmethyl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-(5,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)-N,N-bis(propan-2-yl)benzamide
N-(4-chloronaphthalen-1-yl)-4-(3-methoxypropyl)piperazine-1-carboxamide
N-[4-(2-methyl-1,3-benzoxazol-5-yl)phenyl]methanesulfonamide
{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[(5-methyl-1H-pyrazol-3-yl)methyl]amine
3-{1-[2-(2,2,3,3-tetrafluoropropoxy)acetyl]piperidin-3-yl}benzoic acid
3,3,3-trifluoro-1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}propan-1-one
N,N-diethyl-1-[4-(trifluoromethyl)pyrimidin-2-yl]pyrrolidin-3-amine
methyl (2S,4S)-4-(3,5-dimethyl-1H-pyrazole-4-sulfonamido)-1-methylpyrrolidine-2-carboxylate
4-benzyl-3-ethyl-1-(pyridine-2-carbonyl)-1,4-diazepan-5-one
1-{7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}pent-4-en-1-one
5-ethyl-4-{9-oxa-2-azaspiro[5.5]undecan-2-yl}pyrimidin-2-amine
N-ethyl-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}-N-[2-(pyrrolidin-1-yl)ethyl]acetamide
N-(3-methylphenyl)-3-{1-[3-(1H-pyrazol-1-yl)propyl]piperidin-4-yl}propanamide
3-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-1-[3-(2-methoxyethoxy)phenyl]urea
2-(3-methyl-4-{[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}-1H-pyrazol-1-yl)ethan-1-ol
N-methyl-5-[2-(methylsulfanyl)phenoxymethyl]-N-(1,2-oxazol-5-ylmethyl)-1,2-oxazole-3-carboxamide
ethyl 1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-4-(2-phenylethyl)piperidine-4-carboxylate
N-{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N,1-dimethylpyrrolidin-3-amine
3-[3-(furan-2-yl)propanoyl]-9-methoxy-N-[(4-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-(2-phenylphenyl)-4H-1,2,4-triazole
3-(5-phenyl-1,3,4-oxadiazol-2-yl)-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]propanamide
6-(5,6-dimethylpyrimidin-4-yl)-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]methylamine
2-amino-4-(4-hydroxy-2-methoxyphenyl)-6-(2-methylpropyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
(3R,4S)-4-cyclopropyl-1-[2-methyl-5-(1H-pyrazol-1-yl)benzenesulfonyl]pyrrolidin-3-amine
3-{[1-(pyrrolidine-1-sulfonyl)piperidin-4-yl]methyl}benzoic acid
8-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
3-[(2-methylprop-2-en-1-yl)oxy]-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}benzamide
4-methoxy-6-[2-(3-methoxyphenoxy)ethyl]pyrimidine
2-amino-3-ethyl-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-[(1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-yl)methyl]acetamide
(1R,3S)-3-amino-N-(2-methoxyethyl)-N-[(4-methoxyphenyl)methyl]cyclohexane-1-carboxamide
N-cyclohexyl-1-cyclopropyl-4-oxo-5-(3-oxo-4-phenylpiperazine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
2-(3-methoxyphenoxymethyl)-N-(1-methylpiperidin-3-yl)-1,3-oxazole-4-carboxamide
9-(2-chloro-5-methylbenzoyl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-({2-[1-(1-methylpiperidine-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2,2,2-trifluoroethyl)acetamide
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-4-(2,4-dioxoimidazolidin-1-yl)benzamide
4-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidine-1-carbonyl]-6-(2-methylpropyl)-1,2-dihydropyrimidin-2-one
3-cyclohexyl-N-[(2-ethoxy-3-methoxyphenyl)methyl]-N-methyl-1H-pyrazole-4-carboxamide
5-methyl-2-phenyl-N-[1-(3-propyl-1,2,4-oxadiazol-5-yl)ethyl]furan-3-carboxamide
(1-{6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-4-yl)(1-methyl-1H-imidazol-2-yl)methanol
5-[(4aS,8aR)-1-(3-methoxypropyl)-2-oxo-decahydro-1,6-naphthyridine-6-carbonyl]-1-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(3S,4R)-1-[(2-chloro-4-hydroxyphenyl)methyl]-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
4-[({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-2-methoxyphenol
N-methyl-5-(5-methylfuran-2-yl)-N-[1-(1,2-oxazol-3-yl)ethyl]-1,2,4-triazin-3-amine
1-{1-[(5-methoxy-1H-indazol-3-yl)methyl]piperidin-4-yl}piperidin-4-ol
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-(pyridin-4-yl)quinoline-4-carboxamide