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N-ethyl-2-[4-(1-ethyl-1H-pyrazole-3-carbonyl)piperazin-1-yl]acetamide
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pentane-1,2-dione
1-[2-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-oxoethyl]-1,2-dihydropyrimidin-2-one
2-(pyridin-2-ylmethyl)-8-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
N-(propan-2-yl)-1-(1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperidin-4-yl)piperidine-4-carboxamide
N-{5-[(E)-2-phenylethenyl]pyridin-2-yl}methanesulfonamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
2-(propan-2-yl)-8-[4-(trifluoromethyl)pyrimidin-2-yl]-2,8-diazaspiro[5.5]undecan-3-one
N-[2-methoxy-2-(thiophen-2-yl)ethyl]-1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
5-oxo-1-(pyridin-4-ylmethyl)-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}pyrrolidine-3-carboxamide
3-cyclobutyl-4-(4-methoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(3S,9aR)-3-(hydroxymethyl)-2-methyl-8-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[(4-ethylphenyl)methyl]-N-(2-methoxyethyl)pyridazine-4-carboxamide
(1S,5R)-6-methyl-3-{3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]propanoyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{3-[(3aS,6aS)-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]benzenesulfonyl}-4-methylpiperazine
1-(3-{[(3-methylbutyl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
3-{2-[4-(2-hydroxyethyl)piperazin-1-yl]-2-oxoethyl}-4-(naphthalen-1-ylmethyl)piperazin-2-one
[(3R,5R)-5-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(quinoline-3-carbonyl)piperidin-3-yl]methanol
1-[2-(4-chlorophenyl)ethyl]-N-[3-(methylsulfanyl)propyl]-6-oxopiperidine-3-carboxamide
2-[5-(5-propyl-1,3,4-oxadiazole-2-carbonyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
N-(2-hydroxyethyl)-4-(pyrrolidin-1-ylmethyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]benzamide
2-amino-6-(pyridin-2-yl)-4-[2-(pyrrolidin-1-yl)pyrimidin-5-yl]pyridine-3-carbonitrile
3-{1-[3-(3,5-dimethylphenyl)propanoyl]piperidin-3-yl}-N-[(3-methoxyphenyl)methyl]propanamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-1-(5,6,7,8-tetrahydro-1,6-naphthyridin-6-yl)ethan-1-one
2-hydroxy-6-methyl-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)pyridine-3-carboxamide
2-[(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinolin-2-yl]-N,N,5-trimethylpyrimidin-4-amine
3-(4-ethylpiperazine-1-carbonyl)-N-[(5-methylthiophen-2-yl)methyl]aniline
2-(1H-indol-5-ylmethyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
ethyl 2,4-dimethyl-5-{methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]carbamoyl}-1H-pyrrole-3-carboxylate
2-methoxy-N-({5-[(1-methyl-1H-indol-6-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
4-{[(1S,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}benzamide
2-ethyl-5-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrimidine
2-(1-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethan-1-ol
3-{2-[2-(4-fluorophenyl)azetidin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
(2S)-N2-[(2-chlorophenyl)methyl]-N2-(2-methoxyethyl)pyrrolidine-1,2-dicarboxamide
2-(2-hydroxyphenyl)-1-[4-(4-methoxyphenoxy)piperidin-1-yl]ethan-1-one
methyl 1-(2-methoxyethyl)-5-[(2-methylbutyl)amino]-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(2H-1,2,3,4-tetrazol-2-yl)ethan-1-one
5-(3,5-dimethyl-1-benzofuran-2-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
2-cyclohexyl-N-{5-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl}acetamide
N-[2-(3-fluorophenyl)ethyl]-5-(4-methylpiperidine-1-carbonyl)-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
methyl[2-(oxan-4-yl)ethyl][(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}acetic acid
3-cyclopropyl-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)-1H-pyrazole-5-carboxamide
2-[4-(4-fluorophenyl)-2-[(4-methylpiperazin-1-yl)methyl]phenoxy]-N-(quinolin-3-ylmethyl)acetamide
(1-methoxypropan-2-yl)[2-(2-methyl-1H-indol-1-yl)ethyl]amine
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-amino-7-[2-(2,2,3,3-tetrafluoropropoxy)acetyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[(4aR,8aS)-1-[1-(4-chlorophenyl)cyclobutanecarbonyl]-decahydro-1,6-naphthyridin-6-yl]-2-(thiophen-2-yl)ethan-1-one
5-methyl-1'-{1,3,6-trimethyl-1H-pyrazolo[3,4-b]pyridine-4-carbonyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]