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5-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-3-(propan-2-yl)-1H-pyrazole
N-methyl-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]-N-(pyridin-3-ylmethyl)acetamide
2-ethyl-8-(5-ethyl-1,3,4-thiadiazol-2-yl)-2,8-diazaspiro[4.5]decan-3-one
(3S,4R)-1-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-N,N-dimethyl-4-(4-methylphenyl)pyrrolidin-3-amine
2-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
1-{3-[(dimethylsulfamoyl)amino]phenyl}-3-methyl-3-[(5-methylthiophen-2-yl)methyl]urea
(4-methyl-5-{[1-(9H-purin-6-yl)piperidin-4-yl]methyl}-4H-1,2,4-triazol-3-yl)methanol
1-(1-{[3-hydroxy-5-(hydroxymethyl)-2-methylpyridin-4-yl]methyl}piperidin-4-yl)pyrrolidin-2-one
3-[(cyclopentylamino)methyl]-1-(2,2-dimethylpropyl)-3-hydroxypiperidin-2-one
N-(2,4-dimethoxyphenyl)-3-[1-(1H-pyrrole-2-carbonyl)piperidin-4-yl]propanamide
1-(3-carbamoylpropanoyl)-N-[3-(3-methylphenyl)phenyl]pyrrolidine-2-carboxamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylpyridine-4-carboxamide
methyl 3-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]benzoate
N-ethyl-4-hydroxy-2-(4-methylphenyl)-N-(oxan-4-ylmethyl)pyrimidine-5-carboxamide
4-methyl-N-{3-[2-methyl-3-(1H-1,2,4-triazol-1-yl)propanamido]phenyl}benzamide
N-{1-[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]pyrrolidin-3-yl}acetamide
4-fluoro-N-(2-{7-[(3-phenoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
3-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]benzamide
N-ethyl-1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)pyrrolidine-3-carboxamide
N-{[5-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-[2-(4-fluorophenyl)ethyl]-5-methoxybenzamide
2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-[(4-fluorophenyl)methyl]-5-methoxy-N-methylbenzamide
5-[1-(4-methoxyphenyl)cyclopropanecarbonyl]-3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
3-cyclohexyl-N-[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]-1H-pyrazole-4-carboxamide
1-(azepan-1-yl)-3-[3-({[(2-fluorophenyl)methyl]amino}methyl)phenoxy]propan-2-ol
5-({3-[2,2-bis(prop-2-en-1-yl)pyrrolidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)isoquinoline
3-[2-(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)-1H-imidazol-1-yl]-2,3-dihydro-1λ6-thiophene-1,1-dione
5-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)-N-methylpyrimidin-2-amine
N-{[(3S,4S)-3-hydroxy-1-[2-(propan-2-ylsulfanyl)acetyl]piperidin-4-yl]methyl}furan-2-carboxamide
N-[2-({2,7-dimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)ethyl]methanesulfonamide
{2-fluoro-5-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]phenyl}methanol
(1S,5R)-3-benzyl-6-[2-(methylsulfanyl)pyrimidine-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
methyl 4-{[(4aR,8aS)-1-[4-(furan-2-yl)benzoyl]-decahydro-1,6-naphthyridin-6-yl]methyl}benzoate
4-[4-(8-fluoroquinoline-2-carbonyl)piperazin-1-yl]-6-methylpyrimidin-2-amine
2-({4-[4-(3-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)phenol
(1-ethyl-5-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
N-(1-benzofuran-2-ylmethyl)-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
N-(1-methyl-2-oxopyrrolidin-3-yl)-5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-2-fluorobenzamide
N-methyl-5-(3-methyl-1,2,4-oxadiazol-5-yl)-N-(1,2-oxazol-3-ylmethyl)pyridin-2-amine
(2R,3S,6R)-3-phenyl-5-(quinoxalin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-{[(2R,5S)-5-[(6-methylpyridin-3-yl)methyl]oxolan-2-yl]methyl}thiomorpholine
(2S,4S)-4-amino-N-[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)ethyl]-1-methylpyrrolidine-2-carboxamide
N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(4-methylpiperidine-1-carbonyl)benzene-1-sulfonamide
3-chloro-4-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]oxy}-N-[2-(dimethylamino)ethyl]benzamide
4-(2-methoxy-2-phenylacetyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
N-[2-(1-benzylpiperidin-2-yl)ethyl]-4-hydroxy-1-methylpiperidine-4-carboxamide
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-N'-(3-ethylphenyl)butanediamide
1-[(4-methoxyphenyl)methyl]-4-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one