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1-[(3-methyl-1,2-benzoxazol-5-yl)methyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
1-(4-{4-[(1-propylcyclopropyl)amino]piperidin-1-yl}phenyl)pyrrolidin-2-one
2-(4-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}-1-(3-methylbutyl)piperazin-2-yl)ethan-1-ol
(1S,5R)-6-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
2-(3-chloro-4-hydroxyphenyl)-N-[(3R,4R)-3-hydroxypiperidin-4-yl]acetamide
3-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
3-{[4-(2-fluoro-4-methanesulfonylphenyl)piperazin-1-yl]methyl}pyrrolidin-3-ol
(1R,5R)-N,N-dimethyl-6-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
4-{1-[(4-methoxyphenyl)methyl]-1H-pyrazol-4-yl}pyridin-2-amine
(2R,3R,6R)-3-(3-methoxyphenyl)-5-(oxane-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(4-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}-1,4-oxazepan-6-yl)methanol
8-(1H-indol-3-ylmethyl)-1-(3-methylbutyl)-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{1-[1-(2-hydroxyethyl)-1H-1,3-benzodiazole-5-carbonyl]piperidin-3-yl}benzoic acid
1-{4-[4-(4-methoxybenzoyl)piperazin-1-yl]-4-oxobutyl}pyrrolidin-2-one
N,2-dimethyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]furan-3-carboxamide
1-(3-{3-[2-(methylsulfanyl)pyrimidin-4-yl]phenyl}-1H-pyrazol-1-yl)butan-2-ol
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-propyl-2-(pyrrolidin-3-yl)benzamide
8-[(4-ethoxyphenyl)methyl]-2-phenyl-1,3,8-triazaspiro[4.5]dec-1-en-4-one
2-amino-N-[1-(pyrimidin-2-yl)piperidin-3-yl]-5,6,7,8-tetrahydroquinazoline-4-carboxamide
4-[1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)piperidin-3-yl]benzoic acid
N-[(2-fluorophenyl)methyl]-2-{[(3-phenyl-1H-pyrazol-4-yl)methyl]amino}acetamide
1-[cyclohexyl(methyl)amino]-3-{2-methoxy-4-[({[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}amino)methyl]phenoxy}propan-2-ol
3-{2-[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]-2-oxoethyl}-4-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperazin-2-one
3-(1H-imidazol-1-ylmethyl)-1-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]piperidine
ethyl 5-[(diethylcarbamoyl)methyl]-1-[2-(4-methoxyphenyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}-N-[(2S)-pyrrolidin-2-ylmethyl]benzamide
N-{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}-N-methyloxolan-3-amine
N-(1,4-dioxan-2-ylmethyl)-2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-(4-butylpiperazine-1-carbonyl)-4-(1-methyl-1H-pyrrole-2-carbonyl)morpholine
3-(dimethyl-1,2-oxazol-4-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]propan-1-one
1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-6-methoxyhexan-1-one
1-(1H-imidazole-2-carbonyl)-4-(2-methoxyphenoxy)piperidine
2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(pyrazin-2-ylmethyl)acetamide
5-butyl-6-methyl-N4-[2-(1H-pyrazol-1-yl)ethyl]pyrimidine-2,4-diamine
5,5-dimethyl-3-{2-[4-(1-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-oxoethyl}-1,3-oxazolidine-2,4-dione
3-(3-cyclohexylpropanoyl)-9-methoxy-N-methyl-7-oxo-N-(1,3-thiazol-4-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-[(2E)-3-phenylprop-2-en-1-yl]-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
1-{2-[8-(cyclopropylmethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]-2-oxoethyl}-3,3-dimethylurea
1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-2-(1-propylpiperidin-4-yl)ethan-1-one
{[6-chloro-2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}[2-(1H-imidazol-1-yl)ethyl]amine
1-(3,4-dihydro-2H-1-benzopyran-2-carbonyl)-4-(1-methyl-1H-imidazol-2-yl)piperidine
3-[4-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]-1-[2-(pyridin-3-yloxy)propyl]urea
(2S)-N-{1-[(4-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-2-(methoxymethyl)pyrrolidine-1-carboxamide
4-{[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]methyl}benzoic acid
5-methyl-N-[(4-phenyloxan-4-yl)methyl]-6-(piperidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
3-{4-[(methylcarbamoyl)amino]phenyl}-N-(propan-2-yl)benzamide
(3R,4R)-4-(4-methylpiperazin-1-yl)-1-(quinolin-2-yl)piperidin-3-ol
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-3-(piperidin-3-yl)benzamide
1-(1,3-dihydro-2-benzofuran-5-yl)-3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]urea
5-[(furan-3-ylmethyl)amino]-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid