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2-(methoxymethyl)-6-methyl-4-oxo-1-(3-phenylpropyl)-N-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3-carboxamide
1-[1'-(6-aminopyridine-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
5-[(isoquinolin-5-yloxy)methyl]-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-1,2-oxazole-3-carboxamide
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-2-(1H-pyrazol-1-yl)butanamide
3-ethyl-N-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]methyl}-1,2-oxazole-5-carboxamide
(3R,4R)-4-ethyl-1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperidine-3,4-diol
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-[(4-fluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-cyclopropyl-N-[(4-ethoxyphenyl)methyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
1-tert-butyl-N-ethyl-N-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidine-3-carboxamide
3-methyl-1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidine-3-carbonitrile
3-benzyl-3-[3-(2,5-dihydro-1H-pyrrol-1-yl)-3-oxopropyl]-1-methyl-2,3-dihydro-1H-indol-2-one
1-[5-(methoxymethyl)thiophene-2-carbonyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
3-methoxy-N-[1-(7-{[4-(propan-2-yloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]benzamide
4-({[4-(4-methoxyphenyl)butan-2-yl]amino}methyl)hepta-1,6-dien-4-ol
{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)(thiophen-3-ylmethyl)amine
1-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}-3-(pyrrolidine-1-carbonyl)piperidine
2-{2-[1-(5-chloro-2-fluorobenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
1-(4-{3-[({[4-(propan-2-yl)phenyl]methyl}amino)methyl]pyridin-2-yl}piperazin-1-yl)ethan-1-one
1-[2-(naphthalen-1-ylmethyl)morpholin-4-yl]-3-(1,2-oxazolidin-2-yl)propan-1-one
5-[3-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]quinoxaline
N-ethyl-4-[(furan-2-ylmethyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
4-(3-{[(1,5-dimethyl-1H-indazol-3-yl)methyl]amino}butyl)phenol
ethyl 1-{[3-({1-[3-(2-oxoimidazolidin-1-yl)benzoyl]piperidin-4-yl}oxy)phenyl]methyl}piperidine-2-carboxylate
N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-1H-1,2,3-benzotriazole-5-carboxamide
N-[2-(dimethylamino)ethyl]-3-(1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)propanamide
5-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-2-amine
4-cyano-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]benzamide
4-{[2-(3-methoxyphenyl)ethyl]amino}-N,5-dimethyl-N-(oxolan-3-yl)thieno[2,3-d]pyrimidine-6-carboxamide
3-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-1-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}propan-1-one
{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)[(2-methyl-1,3-thiazol-4-yl)methyl]amine
3-cyclopentyl-5-(2-methanesulfonylethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
4-(2-methoxyphenoxy)-1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidine
(4aS,8aR)-6-[(6-methylpyridin-2-yl)methyl]-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
1-{3-[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-({4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)pyridine
N,N-diethyl-1-[1-(quinolin-8-ylmethyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
(1R,5R)-6-[2-(2-ethylphenoxy)ethyl]-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-{4-[1-(2-hydroxyethyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}-1-(2-methyl-2,3-dihydro-1H-indol-1-yl)ethan-1-one
1-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carboxamide
methyl 2-({4-[(1-cyclopentylpiperidin-4-yl)oxy]-3-methoxyphenyl}formamido)acetate
2-[(4-chlorophenyl)methyl]-8-(5-ethyl-1,3,4-thiadiazol-2-yl)-2,8-diazaspiro[4.5]decan-3-one
2-(2-methoxyethoxy)-1-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]ethan-1-one
4-phenyl-3-[1-(9H-purin-6-yl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(3R,4R)-1-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-3,4-dimethylpyrrolidin-3-ol
3-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-(8-methylquinolin-5-yl)urea
5-(1H-indol-1-ylmethyl)-N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1H-pyrazole-3-carboxamide
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-2-(4-fluorophenyl)-2-hydroxyacetamide
1-(4-{1-[(4-chlorophenyl)methyl]pyrrolidin-3-yl}piperidin-1-yl)-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
2-[({3-[3-(azepan-1-yl)-2-hydroxypropoxy]phenyl}methyl)(methyl)amino]-N-methylacetamide