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N-(1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-3-yl)acetamide
1-(5-phenoxyfuran-2-carbonyl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
({4-cyclopropyl-5-[1-(4-methyl-1H-imidazole-2-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
2-(ethoxymethyl)-N-[2-(furan-2-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-({[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(2-hydroxyethyl)amino)ethan-1-ol
1,6-dimethyl-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}benzonitrile
2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-N-(oxan-4-ylmethyl)-1,3-oxazole-4-carboxamide
5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-(pyridin-4-ylmethyl)pyridin-2-amine
1-(5-phenyl-1,2,4-oxadiazol-3-yl)-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}[(1R)-1-(4-methoxyphenyl)ethyl]amine
N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cycloheptanamine
N-(2,1,3-benzoxadiazol-4-ylmethyl)-N-[(2-ethoxyphenyl)methyl]cyclopropanamine
6-(1H-indol-5-yl)pyrazine-2-carboxylic acid
[(2,5-dimethoxyphenyl)methyl][1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine
6,7-dimethoxy-1-[(4-methylphenyl)methyl]-3-{[(pyridin-3-ylmethyl)amino]methyl}-1,2-dihydroquinolin-2-one
3-(1-{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)propan-1-ol
{1-[(6-fluoroquinolin-2-yl)methyl]-3-(2-phenylethyl)piperidin-3-yl}methanol
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-1-[3-(2-methylphenoxy)azetidin-1-yl]ethan-1-one
1-(4-{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)ethan-1-one
N-(4-chlorophenyl)-3-[1-(3-methylthiophene-2-carbonyl)piperidin-3-yl]propanamide
2-(5-amino-1,3,4-thiadiazol-2-yl)-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]acetamide
1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-3-(2-methoxyphenyl)propan-1-one
N-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-6-oxo-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-N-(prop-2-yn-1-yl)cyclohexanamine
2-methoxy-N-(3-{4-[4-(pyrazin-2-yl)piperazin-1-yl]piperidin-1-yl}phenyl)benzamide
(1S,2R)-N1-[2-(7-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-N2-(prop-2-en-1-yl)cyclohexane-1,2-dicarboxamide
2-{4-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]pyrimidin-5-yl}acetic acid
(1S,2S)-2-[4-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]cyclohexan-1-ol
1-{2-amino-6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}-4-(1H-1,2,3-triazol-4-ylmethyl)-1,4-diazepan-6-ol
3-(1-methyl-1H-pyrazol-5-yl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
3-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}phenol
N-ethyl-1-[(3-methoxyphenyl)methyl]-5-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
3-[2-(2,6-difluorophenyl)ethyl]-1-(1H-pyrazole-3-carbonyl)piperidine
methyl 4-(5-{[4-(acetamidomethyl)piperidin-1-yl]methyl}furan-2-yl)benzoate
3-[7-(3,4-dimethoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]-5,6-dimethyl-1,2-dihydropyridin-2-one
(3aR,6aS)-5-[5-(hydroxymethyl)furan-2-carbonyl]-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-methyl-3-{1-[(3-methyl-1-benzofuran-2-yl)methyl]pyrrolidin-2-yl}-1,2-oxazole
methyl 2-{[(2-fluorophenyl)methyl]sulfamoyl}-6-(4-methyl-2-oxopentanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-(2-phenylethyl)-1-{1-[3-(1H-pyrazol-1-yl)propyl]piperidin-4-yl}piperidine-4-carboxamide
3-{2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-1-yl}-N-(1,3-thiazol-2-yl)propanamide
N-(3-ethoxypropyl)-6-methyl-4-oxo-2-(2-phenylethyl)-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
3-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-5-(propan-2-yl)-1,2-oxazole
N-(2-benzylphenyl)-4-[2-(methylsulfanyl)ethyl]piperazine-1-carboxamide
(1S,9aR)-1-{2-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]ethyl}-octahydro-1H-quinolizine
1-[2-amino-4-(4-fluoropiperidin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-3-methylbut-2-en-1-one
3-(1H-1,2,4-triazol-1-yl)-1-{4-[3-(trifluoromethyl)phenoxy]piperidin-1-yl}propan-1-one
N,1-dimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1H-pyrrole-2-carboxamide
5-[(3-cyclohexylpyrrolidin-1-yl)methyl]-N-methyl-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide