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1-{[1-ethyl-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-4-methyl-1,4-diazepane
{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(3-methylpyridin-4-yl)methyl]amine
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-N-(furan-2-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
3-fluoro-N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]benzamide
1-{4-[(dimethylsulfamoyl)amino]phenyl}-N-[(1S)-1-phenylethyl]piperidin-4-amine
5-(4-fluorophenyl)-N-[(3-methylpyridin-4-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-amino-N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
1-(3-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-3-oxopropyl)pyrrolidin-2-one
7-fluoro-4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1,2-dihydroquinolin-2-one
N-[(3S,4R)-4-(4-methoxyphenyl)-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]pyrrolidin-3-yl]acetamide
[(1-benzylpyrrolidin-3-yl)methyl](methyl)(pyridin-3-ylmethyl)amine
3-[1-(3,4-dimethylbenzenesulfonyl)piperidin-3-yl]-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-{1-[(5-methylpyrazin-2-yl)methyl]-4-phenyl-1H-imidazol-5-yl}phenol
1-(2-methoxyethyl)-8-(1-methoxypropan-2-yl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-(2,3-dimethoxyphenyl)-4-phenyl-1-(prop-2-en-1-yl)-1H-imidazole
6-(2-aminoethyl)-N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N,2-dimethylpyrimidin-4-amine
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]butanamide
1-benzyl-4-(2,6-dimethoxyphenyl)-1H-pyrazole
1-[7-(5-chloropyridin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-4-methylpentane-1,2-dione
4-{[4-(pyridin-4-yl)piperazin-1-yl]methyl}-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraen-2-one
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-(4-ethenylbenzoyl)piperidin-3-amine
1-cyclopentyl-4-{6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carbonyl}piperazin-2-one
methyl 7-oxo-9-(pyridin-2-ylmethoxy)-3-[2-(thiophen-2-yl)acetyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
9-(6-aminopyridine-3-carbonyl)-2-benzyl-2,9-diazaspiro[5.5]undecan-3-one
6-cyclopropyl-N-[1-(thiophen-2-yl)propyl]pyrimidin-4-amine
(2S)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-methoxy-2-phenylacetamide
1-{4-[(cyclohexylamino)methyl]-2-methoxyphenoxy}-3-(diethylamino)propan-2-ol
ethyl 3-(3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}propanamido)propanoate
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-[(3S,4R)-1-benzyl-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanamide
(3S,4R)-1-(cyclopentylcarbamoyl)-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
[3-(cyclopropylmethyl)-1-[4-(difluoromethoxy)benzoyl]piperidin-3-yl]methanol
1-[2-(3-fluorophenyl)ethyl]-N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N-methyl-6-oxopiperidine-3-carboxamide
3-[5-(2-methyl-1H-pyrrole-3-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]-1-(morpholin-4-yl)propan-1-one
N-(5-chloro-2-methoxyphenyl)-3-{1-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]piperidin-3-yl}propanamide
N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
1-({2,4-dimethyl-5-[(4-methylpiperidin-1-yl)methyl]phenyl}methyl)azetidin-3-ol
1-(4-methyl-1,3-thiazole-5-carbonyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
N-(4-chloro-2-ethylphenyl)-4-(3-hydroxypiperidin-1-yl)piperidine-1-carboxamide
3-{5-[2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)ethyl]-1,2,4-oxadiazol-3-yl}pyridine
ethyl 1-(benzenesulfonyl)-4-[(4-methoxyphenyl)methyl]piperidine-4-carboxylate
2-({3-[5-(benzylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-6-methylpyridine
N3-cycloheptyl-1-cyclopropyl-4-oxo-N5-[1-(thiophen-3-yl)propan-2-yl]-1,4-dihydropyridine-3,5-dicarboxamide
N-{[1-(dimethyl-1,2-oxazole-4-carbonyl)piperidin-3-yl]methyl}thiophene-2-sulfonamide
4-ethoxy-N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]pyrimidin-2-amine
N-[(2R,3R)-2-methoxy-1'-[2-(2-oxopyrrolidin-1-yl)acetyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-2-carboxamide
1-[({1-[(3-methylphenyl)methyl]cyclopropyl}carbamoyl)methyl]piperidine-4-carboxamide
2-(2-fluorophenoxymethyl)-N-(propan-2-yl)-1,3-oxazole-4-carboxamide
3-[(3-methoxyphenyl)methyl]-1-(pyridin-3-ylmethyl)piperidine-3-carboxylic acid
1-[cyclohexyl(methyl)amino]-3-[2-methoxy-4-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)phenoxy]propan-2-ol