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ethyl 2-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}pyridine-3-carboxylate
N-{5-[4-(4-methoxyphenyl)piperazine-1-carbonyl]-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl}furan-2-carboxamide
1-[(2-phenylpyrimidin-5-yl)methyl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
methyl[3-(1-methyl-1H-imidazol-2-yl)propyl]{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}amine
4-(4-{[3-(2-methylphenyl)phenyl]methyl}piperazin-1-yl)butan-1-ol
[(2S,6S)-4-(thiophen-3-ylmethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
6-(dimethylamino)-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]pyridine-3-carboxamide
(3S,4S)-4-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-1-methylpyrrolidin-3-ol
5-(2-cyclopentylacetamido)-1-methyl-N-[(5-methylfuran-2-yl)methyl]-2-(oxolan-2-yl)-1H-1,3-benzodiazole-7-carboxamide
2-(1-methyl-3-oxopiperazin-2-yl)-N-[2-(naphthalen-2-yl)ethyl]acetamide
(3S,4R)-1-{2-[(2-methoxyethyl)(methyl)amino]acetyl}-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
5-[1-(1-methyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]-3-(propan-2-yl)-1,2,4-oxadiazole
1-{1-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-1-oxopropan-2-yl}pyrrolidin-2-one
1-(6-fluoro-4-methylquinazolin-2-yl)-N-methyl-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)pyrrolidine-2-carboxamide
(3S,4R)-4-(3-methylthiophen-2-yl)-1-[4-(1H-pyrazol-3-yl)benzoyl]piperidin-3-ol
1-[5-(methoxymethyl)furan-2-carbonyl]-4-(thiophen-2-ylmethyl)-1,4-diazepane
2-(4-chlorophenyl)-4-[(1,2-dimethyl-1H-imidazol-4-yl)sulfonyl]morpholine
1-cyclohexyl-3-(cyclopropylmethyl)-N-[2-(dimethylamino)ethyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
(4aS,7aR)-4-[2-(dimethylamino)acetyl]-N-(furan-2-ylmethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
2,6-diamino-4-(1-methyl-1H-indol-2-yl)-5,6,7,8-tetrahydroquinoline-3-carbonitrile
2-(3,4-dichlorophenyl)-4-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]morpholine
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(trifluoromethyl)benzamide
2,3-dimethyl-6-{4-[2-(1H-pyrrol-1-yl)ethyl]piperazine-1-carbonyl}quinoxaline
2-[3-({[3-(2-ethyl-1H-imidazol-1-yl)propyl]amino}methyl)-2-methyl-1H-indol-1-yl]acetamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-{[(2-fluoro-4-methylphenyl)carbamoyl]methyl}acetamide
N,3,6-trimethyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
2-(1-{[1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
2-[2-oxo-5-(trifluoromethyl)-1,2-dihydropyridin-1-yl]-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}acetamide
1-methyl-3-[3-(pyridin-4-yl)propyl]-8-(thiophen-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
{4-[(4-methoxyphenyl)methyl]-1-(thiophene-3-sulfonyl)piperidin-4-yl}methanol
4-[(4-fluorophenyl)methyl]-1-(3-methylbenzoyl)-3-(propan-2-yl)-1,4-diazepan-5-one
methyl 3-{[1-(pyrimidin-2-yl)piperidin-3-yl]carbamoyl}propanoate
3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-(4-methoxyphenyl)propanamide
2-(2,2-dimethylpropanoyl)-N-(1-phenylethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
1-benzyl-5-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetyl)-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-(2-hydroxyphenoxy)-1-[2-(trifluoromethyl)morpholin-4-yl]ethan-1-one
N-(cyclohex-1-en-1-ylmethyl)-7-[(2-methyl-1,3-oxazol-4-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
5-[(4-hydroxypiperidin-1-yl)methyl]-N-methyl-N-[2-(2-methylpiperidin-1-yl)ethyl]-1,2-oxazole-3-carboxamide
N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-[3-(1,3-thiazol-4-yl)phenyl]piperidin-4-amine
(2E)-1-[3-(3-chlorobenzoyl)piperidin-1-yl]-3-(2-fluorophenyl)prop-2-en-1-one
N-(2-fluoroethyl)-4-(5-methylfuran-2-yl)benzamide
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
1-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
N-[(2-chlorophenyl)methyl]-3-[1-(furan-3-carbonyl)piperidin-3-yl]propanamide
methyl 5-[(3-hydroxy-3-methylbutan-2-yl)amino]-3-(oxolane-2-amido)-1-(2-phenylethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-[(3,5-difluorophenyl)methyl]-8-[(2R)-oxolane-2-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
3-{[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-2-methoxypyridine
5-benzyl-5-[1-(quinoxalin-5-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}-1-[4-(propan-2-yl)phenyl]-1H-pyrazole
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-2-(2-methylphenyl)acetamide