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methyl 1-[6-(2-methoxyphenyl)pyridazin-3-yl]piperidine-4-carboxylate
N-{[2-(dimethylamino)-7-(methylsulfanyl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-2,3,4-trimethoxybenzamide
N-(2-ethoxyphenyl)-N'-{2-[(pyridin-3-yl)amino]ethyl}propanediamide
1-(4-methylpiperazin-1-yl)-3-{1-[2-(pyridin-4-ylsulfanyl)acetyl]piperidin-3-yl}propan-1-one
3-{1-[2-(1H-imidazol-4-yl)acetyl]piperidin-3-yl}-N-(4-methoxy-2-methylphenyl)propanamide
N,N-diethyl-1-{1-[(4-hydroxy-3-methoxyphenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
(3S)-3-({[7-fluoro-2-(3-methoxyphenyl)quinolin-3-yl]methyl}amino)azepan-2-one
1-{5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1H-pyrazole-3-carbonyl}piperidin-3-ol
4-{2-[1-butyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]phenyl}morpholine
ethyl 1-(1-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-4-yl)piperidine-4-carboxylate
4-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
2-{[(1-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)oxy]methyl}pyridine
3-(1-methylpiperidin-4-yl)-N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-4-ylmethyl)propanamide
1-[cyclohexyl(methyl)amino]-3-[2-methoxy-4-({methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
2-{4-[2-amino-6-(methylamino)pyrimidin-4-yl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
N-(1-ethyl-1H-1,2,4-triazol-3-yl)-10-azabicyclo[4.3.1]decane-10-carboxamide
3-(dimethyl-1,2-oxazol-4-yl)-1-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]urea
4-methyl-N-({4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)benzamide
5-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]-2,1,3-benzoxadiazol-1-ium-1-olate
N-methyl-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)-N-[1-(pyridin-3-yl)pentyl]benzamide
5-[(1-cyclohexyl-1H-1,2,4-triazol-5-yl)methyl]-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-[5-(2-chlorophenyl)furan-2-carbonyl]-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
2-[1-(dimethyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]-4-methyl-1H-1,3-benzodiazole
2-[(1S,5R)-3-[3-(1H-1,3-benzodiazol-2-yl)propanoyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
2-(3-methoxypropyl)-1-{[4-(1,2-oxazol-5-yl)thiophen-2-yl]sulfonyl}piperidine
1-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]-3-[1-methyl-3-(pyridin-2-yl)-1H-pyrazol-5-yl]urea
1-methyl-4-(2-phenyl-1,3-thiazol-4-yl)-3-(pyridin-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(3S,4R)-1-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
6-(methoxymethyl)-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)pyrimidin-4-amine
2-[2-(3-chlorophenoxy)acetyl]-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
8-(3-hydroxypropyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-phenyl-1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperidin-3-amine
1-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-4-yl)-2-(3,4-dimethoxyphenyl)-1H-1,3-benzodiazole
methyl({[1-(2-methylpropyl)-2-(oxolan-2-ylmethanesulfonyl)-1H-imidazol-5-yl]methyl})(2-phenoxyethyl)amine
(3S,9aR)-3-(hydroxymethyl)-8-(4-methylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-{[1-(1,4-oxazepan-4-yl)hex-5-en-2-yl]oxy}pyridine-4-carbonitrile
(1S,3R)-3-[3-(4-chloro-1H-pyrazol-1-yl)propanamido]-N-(3,5-dimethylphenyl)cyclopentane-1-carboxamide
1'-(4-chlorobenzoyl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N-(1H-indazol-4-yl)-4-{[(propan-2-yl)carbamoyl]methyl}piperazine-1-carboxamide
2-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]morpholine
2-(2,4-difluorophenyl)-4-{[2-(3-methoxyphenyl)pyrrolidin-1-yl]methyl}-5-methyl-1,3-oxazole
3-methyl-N-(oxolan-2-ylmethyl)-N-({4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)thiophene-2-carboxamide
3-[1-(7-methoxy-1,2,3,4-tetrahydronaphthalen-2-yl)piperidin-4-yl]-1-(morpholin-4-yl)propan-1-one
N-[1-(7-{[4-(diethylamino)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-2-methylpropanamide
3-{1-[5-(2-chloro-4-methoxyphenoxymethyl)-1H-pyrazol-3-yl]-N-methylformamido}propanamide
(2S,4R)-N-ethyl-4-[(1-ethylpiperidin-4-yl)amino]-1-(naphthalen-2-ylmethyl)pyrrolidine-2-carboxamide
2-[(4-methoxyphenyl)methyl]-N-methyl-N-[2-(oxan-4-yl)ethyl]-1,3-benzoxazole-6-carboxamide
3-{1-[(2-chloro-4-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide