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3-(but-2-yn-1-yl)-5-{1-[(2-methylphenyl)methyl]piperidin-4-yl}-5-(2-phenylethyl)imidazolidine-2,4-dione
4-fluoro-3-{3-methyl-5-[(methylsulfanyl)methyl]-1H-1,2,4-triazol-1-yl}benzene-1-sulfonamide
1-tert-butyl-N-[3-(1H-indazol-1-yl)propyl]-5-oxopyrrolidine-3-carboxamide
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-(pyridin-4-ylmethyl)acetamide
2-(3-hydroxypropyl)-8-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
5-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]-3,4-dihydropyrimidin-4-one
N,3,5-trimethyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-1H-indole-2-carboxamide
5-[(2S)-2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-4-ethyl-1,3-thiazol-2-amine
3-(hydroxymethyl)-1-[6-(4-hydroxypiperidin-1-yl)pyrimidin-4-yl]piperidin-3-ol
1-[2-(dimethylamino)ethyl]-3-(2-fluorophenyl)-3-{2-[3-(methoxymethyl)piperidin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
2-(5-fluoro-2-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
5-[2-(3-methoxyphenyl)piperidine-1-carbonyl]-N,N,4-trimethylpyrimidin-2-amine
2-(2-ethoxyphenyl)-5-methyl-4-{[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methyl}-1,3-oxazole
N-(1-{2-[4-(1,3-benzoxazol-2-yl)piperidin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-2H-1,3-benzodioxole-5-carboxamide
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-[2-(4-methoxyphenyl)ethyl]piperidine
(2S,4S)-4-amino-N-[2-(5-cyano-2-methyl-1H-indol-3-yl)ethyl]-1-methylpyrrolidine-2-carboxamide
6-{2-[(2-methoxyphenyl)methoxy]phenyl}-N,N-dimethylpyridine-3-carboxamide
N,N-dimethyl-6-[2-(trifluoromethyl)morpholin-4-yl]pyridine-3-carboxamide
1-(1H-indazol-5-yl)-4-[(3R)-1,2,3,4-tetrahydroisoquinoline-3-carbonyl]piperazin-2-one
4-(5-{[3-(2,6-dimethylphenoxy)azetidin-1-yl]methyl}pyrimidin-2-yl)morpholine
N-methyl-N-[2-(2-methyl-1H-indol-1-yl)ethyl]-3-(pyridin-4-yl)propanamide
2-(3-methoxyphenoxy)-1-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
(1R,7S)-N-methyl-N-(1,2-oxazol-3-ylmethyl)-4-oxo-3-(pentan-3-yl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N,4,6-trimethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]quinolin-2-amine
(1S,9S)-11-[(6-chloro-4-{[3-(propan-2-yloxy)propyl]amino}quinazolin-2-yl)methyl]-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
1-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]azetidin-3-yl}-3,5-dimethyl-1H-pyrazole
4-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-1,2-dihydroquinolin-2-one
2,8-dimethyl-4-[4-(propan-2-yl)piperazine-1-carbonyl]quinoline
3-[methyl(1-methylpyrrolidin-3-yl)amino]-1-[4-(4-methylphenoxy)piperidin-1-yl]propan-1-one
3-fluoro-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]pyridine-4-carboxamide
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-[5-(1H-indol-2-yl)-4-phenyl-1H-imidazol-1-yl]-1-(pyrrolidin-1-yl)propan-1-one
methyl 3-[(5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)amino]propanoate
N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-2-(pyridin-3-yloxy)acetamide
5-fluoro-1-methyl-2-{[4-(3-methylpyridin-2-yl)piperazin-1-yl]methyl}-1H-indole
N1-phenyl-N2-{2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}ethane-1,2-diamine
N-{3-[4-(5-chloropyridin-2-yl)piperazine-1-carbonyl]phenyl}-2-methoxyacetamide
2-{[({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)amino]methyl}-6-methoxyphenol
3-methyl-N-[3-(methylsulfanyl)propyl]-4-oxo-3,4-dihydrophthalazine-1-carboxamide
4-{[5-(1,3-dimethyl-1H-pyrazol-5-yl)-1H,4H-pyrazolo[3,4-d]imidazol-1-yl]methyl}pyridine
N-(3,3-diphenylpropyl)-6-[(3-ethoxy-4-hydroxyphenyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
3-[2-(naphthalen-1-yl)-1H-imidazol-1-yl]pyridine
2-methyl-4-[3-(trifluoromethoxy)phenyl]-1H-imidazole
(1S,5R)-6-(cyclobutylmethyl)-N-(2-methoxyphenyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
3-[(3-methyl-1H-pyrazol-5-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
7-methyl-3-(1,3-thiazol-4-ylmethyl)-3,7,11-triazaspiro[5.6]dodecan-12-one
2-{[4-(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)-1H-1,2,3-triazol-1-yl]methyl}-4-methanesulfonylmorpholine
4-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-7-(2-methylphenyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-phenoxy-N-[1-({[1-(thiophen-3-yl)propan-2-yl]carbamoyl}methyl)-1H-pyrazol-4-yl]propanamide
ethyl 2-oxo-5-{[(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amino]methyl}-2,3-dihydro-1H-imidazole-4-carboxylate