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4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-methyl-N-(thiophen-3-ylmethyl)benzamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[(2-ethoxypyridin-3-yl)methyl]propanamide
N-ethyl-5-{1-[1-(pyridin-4-yl)propyl]-1H-1,2,3-triazol-4-yl}pyrimidin-2-amine
2-(3-methylthiophen-2-yl)-1-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazole
1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-2-(thiophen-2-yl)ethan-1-one
1-(azocan-1-yl)-3-{2-methoxy-5-[({2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}amino)methyl]phenoxy}propan-2-ol
2-cyclopentyl-8-(1H-pyrrole-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(2,4-dimethylphenyl)-2-[4-(3-methoxybenzoyl)piperazin-1-yl]acetic acid
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-(thiophen-2-yl)propanamide
3-cyclopropyl-6-[2-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)ethyl]-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
1-{9-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl}-2-(1H-imidazol-4-yl)ethan-1-one
7-fluoro-2-methyl-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]quinoline-4-carboxamide
N-[2-(2-chlorophenyl)ethyl]-5-(4-methylpiperidine-1-carbonyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
7-{thieno[3,2-d]pyrimidin-4-yl}-2,7-diazaspiro[4.4]nonane-1,3-dione
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[7-methyl-2-(3-methylphenyl)quinolin-3-yl]methyl}thiophene-2-carboxamide
(1S,5R)-3-(2H-1,3-benzodioxol-5-ylmethyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
6-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
N-(2-chlorophenyl)-3-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]propanamide
4-[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-N-[2-(prop-2-en-1-yloxy)phenyl]piperidine-1-carboxamide
4-(1,3-benzothiazol-2-yl)-2-({[2-(diethylamino)ethyl](methyl)amino}methyl)phenol
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
2-({[(1-cyclopentylpiperidin-3-yl)methyl][2-(piperidin-1-yl)ethyl]amino}methyl)phenol
N-[4-(methylsulfanyl)phenyl]-6-[(2E)-3-phenylprop-2-enoyl]-6-azaspiro[2.5]octane-1-carboxamide
1-{1,9-dioxaspiro[5.5]undecan-4-yl}-4-{5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}piperazine
N-(2-chloro-4-{5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-6-yl}phenyl)-2-methoxyacetamide
(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)-N-(2-phenylethyl)pyrrolidine-1-carboxamide
N-{[7-(2H-1,3-benzodioxole-5-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-methoxy-2-phenylacetamide
(3S,4S)-1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4-(morpholin-4-yl)pyrrolidin-3-ol
1-(3-acetylphenyl)-3-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}urea
methyl 2-{[(3-chlorophenyl)methyl]sulfamoyl}-6-(2-methylbutanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-methoxy-N-[2-methyl-3-({[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]carbamoyl}amino)phenyl]acetamide
3-{[(4-cyclobutyl-6-methylpyrimidin-2-yl)amino]methyl}-6-ethyl-2-methoxy-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
1-{4-[hydroxy(phenyl)methyl]piperidin-1-yl}-3-(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propan-1-one
2,8-dimethyl-4-[3-(3-methylphenoxy)azetidine-1-carbonyl]quinoline
2-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]acetic acid
8-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-{5-methylimidazo[1,2-a]pyridin-2-yl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-(4-{[(1S,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}phenoxy)acetic acid
2-(pyridin-2-ylsulfanyl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]acetamide
2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-3-(trifluoromethyl)pyridine
9-(2-methoxyethyl)-1-methyl-4-(4-methyl-1H-imidazole-2-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(2-methyl-1H-imidazol-1-yl)-1-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)ethan-1-one
1-[1-(2-{1-oxa-8-azaspiro[4.5]decan-8-yl}-2-oxoethyl)-1H-indol-3-yl]butan-1-one
3-[1-(1,3-benzothiazol-2-ylmethyl)piperidin-4-yl]-N-[2-(dimethylamino)ethyl]propanamide
1-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
2-{4-[(dimethylamino)methyl]phenyl}-N-(1-methyl-1H-indazol-6-yl)pyrrolidine-1-carboxamide
4-[4-(4-methylphenyl)-2-{[2-(pyrazin-2-yl)ethyl]amino}pyrimidin-5-yl]phenol
3-(2H-1,3-benzodioxol-5-yl)-N-(3-methylbutyl)-3-phenylpropanamide
4-[(2,3-difluoro-6-methoxyphenyl)methyl]-1-(3-methoxyphenyl)piperazin-2-one