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N-(5-fluoro-2-methylphenyl)-2-({2-[(prop-2-en-1-yl)amino]phenyl}formamido)propanamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}acetamide
1-{2-[3-(2-ethylphenoxy)azetidin-1-yl]-2-oxoethyl}pyrrolidin-2-one
N-({1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)piperidine-1-carboxamide
3-{[(1-cyclohexyl-1H-1,2,4-triazol-5-yl)methyl](methyl)amino}-1λ6-thiolane-1,1-dione
2-{[1-(2-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}pyridine
2-(2-chloro-6-fluorophenyl)-N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}acetamide
N-(4-acetylphenyl)-3-oxo-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-2-(3-methyl-1,2-oxazol-5-yl)acetamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-3-(1H-pyrazol-4-yl)propanamide
N-(2-hydroxy-2-phenylethyl)-N-methyl-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
4-(1-{4-[6-(methoxymethyl)pyrimidin-4-yl]phenyl}ethyl)morpholine
6-cyclopentyl-N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
9-methoxy-N-[(3-methoxyphenyl)methyl]-3-(2-methylfuran-3-carbonyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-(1-{[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperidin-4-yl)-1,2,3,4-tetrahydroisoquinoline
(2S,4S)-4-amino-N-methyl-1-(4-methyl-2-phenylpyrimidine-5-carbonyl)pyrrolidine-2-carboxamide
N-[(1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)methyl]acetamide
8-fluoro-2-({[2-(pyrazin-2-yl)ethyl]amino}methyl)quinolin-4-ol
3-[1-(3-ethyl-4-methyl-1H-pyrazol-5-yl)-N-methylformamido]-N-methylbutanamide
1-amino-3-[1-(3-chloro-4-fluorophenyl)-1H-1,2,4-triazol-5-yl]propan-2-ol
1-methyl-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-1H-indole-6-carboxamide
[(3-chloropyridin-4-yl)methyl](methyl){[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}amine
5-{[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-N-methylfuran-2-carboxamide
N-{[1-(3,5-dimethylfuran-2-carbonyl)piperidin-3-yl]methyl}thiophene-2-sulfonamide
5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-3-methyl-1H-1,2,4-triazole
1-[1-methyl-5-({4-[(4-methylpiperazin-1-yl)methyl]piperidin-1-yl}methyl)-1H-pyrrol-3-yl]ethan-1-one
3-fluoro-N-[(4-{[(2-fluorophenyl)methyl]amino}-8-methylquinazolin-2-yl)methyl]benzene-1-sulfonamide
1-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]-3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]propan-1-one
1-{3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-[1-(propan-2-yl)-1H-imidazol-2-yl]-1H-imidazole
10-methoxy-5-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
3-methyl-7-[(3-methylquinoxalin-2-yl)methyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N-[(3S,4R)-4-propyl-1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}pyrrolidin-3-yl]methanesulfonamide
{5-[1-(1H-indazol-6-yl)-1H-imidazol-2-yl]furan-2-yl}methanol
2-methyl-7-({3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}methyl)-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
3-({[6-chloro-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}carbamoyl)pyridin-1-ium-1-olate
4-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrole-2-carbonyl]-8-chloro-2-(furan-2-yl)quinoline
7-methyl-11-[(4-methyl-1H-imidazol-2-yl)methyl]-3,7,11-triazaspiro[5.6]dodecane
N-{[4-(1H-1,3-benzodiazol-2-yl)cyclohexyl]methyl}-1-cyclopropyl-6-oxopiperidine-3-carboxamide
(1R,7S)-3-[4-(2-hydroxyethyl)phenyl]-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-[(4-chlorophenyl)methyl]-N-[1-(3-methoxyphenyl)ethyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
N-[5-(methoxymethyl)-1,3,4-thiadiazol-2-yl]-2-{2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidin-1-yl}acetamide
ethyl 4-(7-chloro-3-{[N-cyclopropyl-2-(thiophen-3-yl)acetamido]methyl}quinolin-2-yl)piperazine-1-carboxylate
3-(3-chloro-1H-1,2,4-triazol-5-yl)-1-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]propan-1-one
1-[4-({4-[(3-ethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-1-yl]ethan-1-one
ethyl 1-(6,7-dimethoxy-3-{[(1,2-oxazol-3-ylmethyl)amino]methyl}quinolin-2-yl)piperidine-3-carboxylate
N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanamide
2-[4-chloro-2-(6-methyl-1H-1,3-benzodiazol-2-yl)phenoxy]acetic acid
N-ethyl-2-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-N-methylacetamide