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N-(1-cyclopropanecarbonylpiperidin-3-yl)-3-(3-hydroxy-3-methylbutyl)benzamide
3-(4-methyl-1,3-thiazol-5-yl)-1-[2-(pyridin-3-yl)pyrrolidin-1-yl]propan-1-one
3-[3-(dimethylamino)propyl]-5-{1-[(2E)-2-methylbut-2-enoyl]piperidin-4-yl}-5-[(2-methylphenyl)methyl]imidazolidine-2,4-dione
N-benzyl-2-[4-(4-fluorophenyl)-2-[(4-methylpiperazin-1-yl)methyl]phenoxy]-N-methylacetamide
2-ethyl-N-[1-(4-methyl-1H-imidazol-2-yl)propyl]pyrimidine-5-carboxamide
5-(6-aminopyridin-3-yl)-4-(4-methylphenyl)-N-[(5-methylpyrazin-2-yl)methyl]pyrimidin-2-amine
2-[4-(propan-2-yl)phenyl]-5-(1H-1,2,3,4-tetrazol-1-yl)-1H-1,3-benzodiazole
methyl[(2-phenyl-1,3-oxazol-4-yl)methyl][1-(pyrazin-2-yl)propan-2-yl]amine
4-(dimethylamino)-N-[4-(furan-2-yl)phenyl]azepane-1-carboxamide
14-(1H-indol-4-yl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
2-(3-fluorophenyl)-1-(1-methyl-3-phenyl-1H-pyrazole-5-carbonyl)piperidine
6-[3-(propan-2-yl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-4-(3-methylpyridin-2-yl)piperazine
2-(2-aminoethyl)-N-{imidazo[1,2-a]pyridin-3-ylmethyl}-5,6-dimethylthieno[2,3-d]pyrimidin-4-amine
2-(3-hydroxypropyl)-9-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
4-(1-butyl-1H-imidazol-2-yl)-1-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)piperidine
N-[(3R,4S)-4-cyclopropyl-1-[2-(pyridin-2-yl)ethyl]pyrrolidin-3-yl]methanesulfonamide
(4-{[1-(2-fluoro-5-methylbenzenesulfonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[(5-ethylfuran-2-yl)methyl]pyrrolidine-3-carboxylic acid
(2E)-3-(3,4-difluorophenyl)-1-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)prop-2-en-1-one
1-[(3R,5S)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]-2-(1H-imidazol-1-yl)ethan-1-one
3-acetamido-N-(2-methoxyphenyl)-5-{[(quinolin-7-ylmethyl)amino]methyl}benzamide
5,8-dimethyl-2-{[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}quinolin-4-ol
ethyl 1-(1H-1,3-benzodiazol-2-ylmethyl)-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
(2S)-5-oxo-N-[(2-phenoxypyridin-3-yl)methyl]pyrrolidine-2-carboxamide
1-({4-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]phenyl}methyl)piperidine
N-cyclopropyl-4-[(8-methoxy-2H-chromen-3-yl)methyl]piperazine-2-carboxamide
1-[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidin-1-yl]-2-(4-methyl-1H-pyrazol-1-yl)ethan-1-one
1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N-[4-(1H-pyrazol-5-yl)phenyl]piperidine-3-carboxamide
methyl 3-({5-[1-(4-chlorophenyl)cyclopropanecarbonyl]-1-(cyclopropylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}formamido)propanoate
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-methyl-1H-pyrazole-5-carboxamide
N-[2-(1H-imidazol-4-yl)ethyl]-2-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)butanamide
3-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-3-methyl-1-(4-methyl-2-oxo-2H-chromen-7-yl)urea
N-cyclopropyl-4-(1H-indol-2-ylmethyl)piperazine-2-carboxamide
2-{2-[(2-methylpyrrolidin-1-yl)methyl]phenyl}-6-(phenoxymethyl)-3,4-dihydropyrimidin-4-one
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
(3S,7S)-5-[3-(6-oxo-1,6-dihydropyridazin-3-yl)propanoyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
7-[2-(morpholin-4-yl)propanoyl]-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2,2-diphenyl-1-(4-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)ethan-1-ol
methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl][(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]amine
2-[({[(1R,2R)-2-hydroxy-2-methylcyclohexyl]methyl}amino)methyl]-6-methylquinolin-4-ol
4-({2-[2-(dimethylamino)ethyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}sulfonyl)benzonitrile
6-[4-hydroxy-4-(hydroxymethyl)piperidine-1-carbonyl]-3,5-dimethyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
1-(morpholin-2-ylmethyl)-3-(1-{[2-(trifluoromethyl)phenyl]methyl}-1H-pyrazol-5-yl)urea
ethyl 1-[3-(2-oxopyrrolidin-1-yl)propanoyl]-3-(3-phenylpropyl)piperidine-3-carboxylate
[(2S,6S)-4-[(3,4-dimethoxypyridin-2-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
N-({7-[1-(4-chlorophenyl)cyclobutanecarbonyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(1H-imidazol-1-yl)acetamide
ethyl[(1-ethyl-1H-pyrazol-4-yl)methyl][(6-methoxypyridin-3-yl)methyl]amine
2-[3-(3-fluorophenyl)-2,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]acetamide
1-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)-3-(morpholin-4-yl)propan-1-one