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N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
[(3R,4R)-1-(3-chlorobenzoyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
ethyl 2-(1-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}piperidin-2-yl)acetate
(1S,4S)-2-(3-chloro-4-methoxyphenyl)-5-[(3,4-dimethoxyphenyl)methyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
2-[(3-chlorophenyl)methyl]-N-cyclobutyl-1,3-benzoxazole-6-carboxamide
2-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]quinoxaline
9-(3,4-dimethylbenzoyl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
3-{5-[2-(4-fluorophenoxy)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
(2S,4R)-4-amino-N-ethyl-1-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carbonyl]pyrrolidine-2-carboxamide
(3R,4R)-1-[(3,7-dimethyl-1H-indol-2-yl)methyl]-4-(morpholin-4-yl)piperidin-3-ol
N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
(2R,3R,6R)-5-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(thiophene-2-carbonyl)piperazine
3-{2-[2-(pyridin-2-yl)ethyl]piperidine-1-carbonyl}-1,2-dihydroquinolin-2-one
(2R,3R,6R)-5-(2-fluoro-4-methylbenzoyl)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
[4-(2-methyl-1,3-benzoxazole-6-carbonyl)-1,4-oxazepan-6-yl]methanol
N-[(3-fluorophenyl)methyl]-2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carboxamide
ethyl 4-[(4-chlorophenyl)methyl]-1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]piperidine-4-carboxylate
3-[3-(dimethylamino)propyl]-5-[(3-fluorophenyl)methyl]-5-[1-(thiophene-2-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
1-{imidazo[1,2-a]pyridine-3-carbonyl}-3-(2-methylphenyl)piperidine
N3-cyclooctyl-N5-[2-(3-fluorophenyl)ethyl]-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
2-[5-cyclopropyl-4-(4-ethylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]-5-methyl-4-(thiophen-2-yl)pyrimidine
N-(4-{1-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-1H-imidazol-2-yl}phenyl)acetamide
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(1H-pyrrole-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
1-[(4aR,8aR)-7-cyclobutanecarbonyl-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-3-(5-methyl-1H-pyrazol-1-yl)propan-1-one
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-(2-methylpropyl)acetamide
2-chloro-4-{[3-(2-hydroxyethyl)-4-(3-methylbutyl)piperazin-1-yl]methyl}phenol
1-[1-(2,2-dimethyloxane-4-carbonyl)piperidin-4-yl]-2-(4-methylphenoxymethyl)-1H-1,3-benzodiazole
1-[4-(4-methylphenoxy)piperidin-1-yl]-2-(1-methylpiperidin-2-yl)ethan-1-one
1-(3-ethyl-1,2-oxazole-5-carbonyl)-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-2-carboxamide
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-{thieno[2,3-d]pyrimidin-4-yl}pyrrolidin-3-yl]methanol
(2R,6R)-4-[(4-acetyl-1-methyl-1H-pyrrol-2-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
4-hydroxy-2-phenyl-N-[2-(piperidin-1-yl)butyl]pyrimidine-5-carboxamide
4-ethyl-6-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyrimidine
1-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
(1R,3S)-7-[4-(4-propylphenyl)benzoyl]-7-azaspiro[3.5]nonane-1,3-diol
1-methyl-N-(2-phenylethyl)-5-[(1,3-thiazol-2-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-[2-(2-hydroxyphenyl)acetyl]-1-(2-methoxyphenyl)piperazin-2-one
({4-cyclopropyl-5-[1-(4-methylbenzoyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
N'-[1-(pyridin-4-yl)propan-2-yl]-N-(2,4,6-trimethylphenyl)butanediamide
[(3-{2-[4-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)(thiophen-2-ylmethyl)amine
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1-[(2-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1,2-oxazole-3-carbonyl)piperidine
2-[5-(ethylsulfanyl)thiophene-2-carbonyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one
2-[5-oxo-3-(piperidin-1-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-4-yl]propanoic acid
N-[(1-benzylpiperidin-3-yl)methyl]thiophene-2-carboxamide
N-[3-(cyclopentyloxy)propyl]-2-(dimethylamino)-2-(4-methylphenyl)acetamide
(3R,4R)-3-cyclopropyl-1-{5-[(diethylamino)methyl]-2-methylfuran-3-carbonyl}-4-methylpyrrolidin-3-ol
4-[1-benzyl-5-(1-methoxypropan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine