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4-(5-{[3-(2-chlorophenyl)pyrrolidin-1-yl]methyl}-1,3-thiazol-2-yl)morpholine
2-(4-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)pyrimidine
2-ethyl-9-[(4-methoxy-3-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(2-acetamidophenyl)-2-{methyl[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]amino}acetamide
2-({[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]amino}methyl)-6-fluoroquinolin-4-ol
3-[(1-cyclopentylpiperidin-4-yl)oxy]-N-[2-(1H-pyrazol-4-yl)ethyl]benzamide
1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
2-{5-methyl-[1,2,4]triazolo[4,3-a]pyridin-3-yl}quinolin-4-ol
1-[4-(dimethylamino)azepan-1-yl]-2-(2-hydroxyphenyl)ethan-1-one
2-(cyclopropylmethyl)-7-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-N-(pyridin-3-ylmethyl)butanamide
(3S,4R)-4-methyl-1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidine-3,4-diol
N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
ethyl 1-{[2-(furan-2-yl)phenyl]methyl}-4-(2-methoxyethyl)piperidine-4-carboxylate
6-ethyl-N-(2-methanesulfonylethyl)-2-(piperidin-1-yl)pyrimidin-4-amine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetamide
(4aR,8aS)-6-(pyridin-4-ylmethyl)-1-[(3,4,5-trimethoxyphenyl)methyl]-decahydro-1,6-naphthyridin-2-one
N-{2-[1-(1,1-dioxo-1λ6-thiolan-3-yl)-3-methyl-1H-1,2,4-triazol-5-yl]ethyl}-2-fluorobenzamide
1-{3-[4-(3-hydroxypiperidin-1-yl)piperidine-1-carbonyl]phenyl}ethan-1-one
1-(2,4-dimethylphenyl)-4-{5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}piperazine
(3S,5S)-5-[(4-fluorophenyl)carbamoyl]-1-(pyridin-2-ylmethyl)piperidine-3-carboxylic acid
N-{[7-(2-cyclopentyl-2-phenylacetyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}pyrazine-2-carboxamide
N-(1-{7-[(2-chlorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)furan-3-carboxamide
N-[(2S,4R,6S)-2-(2-methylpropyl)-6-(1,3-thiazol-2-yl)oxan-4-yl]benzamide
N-[2-(2,2-dimethyl-4-phenyloxan-4-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
(1R,9aR)-1-(1H-indazol-1-ylmethyl)-octahydro-1H-quinolizin-1-ol
2-methyl-4-[3-(1,2-oxazinane-2-carbonyl)phenyl]but-3-yn-2-ol
1-[2-(piperidin-2-yl)ethyl]-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}-1H-1,2,3-triazole-4-carboxamide
3-[5-(4-methylbenzoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
3-(4-fluorophenyl)-6-(3-methyl-1H-pyrazol-4-yl)pyridazine
1-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]butan-2-ol
2-{[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}-4-(pyrazin-2-yl)phenol
N-[2-(2-fluorophenyl)ethyl]-1-[(2-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
(3aS,6aS)-2-cyclopentyl-5-[2-(3,5-difluorophenyl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-(2-ethylpyridine-4-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
(5S,9aS,9bS)-2-[(4-methoxyphenyl)methyl]-5-(thiophen-3-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-{2-[3-(benzyloxy)piperidin-1-yl]-2-oxoethyl}-3-methoxy-1,2-dihydropyridin-2-one
N-[(2-fluorophenyl)methyl]-5-methylpyrazolo[1,5-a]pyrimidin-7-amine
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-(2-methylpropyl)pyrrolidin-2-one
1-{3-[7-(2,2-dimethylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-oxopropyl}azepan-2-one
N-(4-cyanonaphthalen-1-yl)-4-cyclohexyl-3-oxopiperazine-1-carboxamide
3-[(3R,4S)-4-(dimethylamino)-1-[(trimethyl-1H-pyrazol-4-yl)sulfonyl]piperidin-3-yl]propanoic acid
1-{4-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl}-4-(1H-pyrazol-4-yl)butan-1-one
2-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyrazine
2-{3-[3-(4-methoxy-2-methylphenyl)phenyl]-1H-pyrazol-1-yl}ethan-1-ol
2-(4-chloro-1H-pyrazol-1-yl)-N-[2-(4-phenylpyrimidin-2-yl)ethyl]propanamide
(3R,4R)-1-(2,4-difluorobenzenesulfonyl)-3,4-dimethylpyrrolidin-3-ol
5-[1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1H-1,2,3-triazol-4-yl]-3-propyl-1,2,4-oxadiazole
N-(2-hydroxyethyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-2,3-dihydro-1H-indene-1-carboxamide
2-(2-ethyl-1H-imidazol-1-yl)-1-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]ethan-1-one