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4-[1-(4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}phenyl)ethyl]morpholine
5-butyl-N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]pyridine-2-carboxamide
N,N-dimethyl-2-[(1S,5R)-6-[(5-phenylthiophen-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
ethyl 4-{6-[4-(morpholin-4-yl)benzoyl]-6-azaspiro[2.5]octane-1-carbonyl}piperazine-1-carboxylate
3-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decane-4-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
N-cyclooctyl-3-[(3S,4R)-4-[4-(2-methoxyphenyl)piperazin-1-yl]-1-(pyridin-2-ylmethyl)piperidin-3-yl]propanamide
N-phenyl-5-[2-(1H-1,2,4-triazol-1-yl)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-phenyl-2-(2-{[3-(trifluoromethyl)phenyl]methyl}morpholin-4-yl)ethane-1,2-dione
N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
2-{2-[4-(oxolan-3-yl)-1H-1,2,3-triazol-1-yl]ethyl}-1,2,3,4-tetrahydrophthalazine-1,4-dione
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
3-(3-methylthiophene-2-carbonyl)-1-[3-(1H-pyrazol-1-yl)propyl]piperidine
N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)-4-oxopentanamide
(2S,4R)-4-amino-1-[(6-chloropyridin-3-yl)methyl]-N,N-diethylpyrrolidine-2-carboxamide
1-(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
methyl 3-(4-fluorobenzamido)-6-{[methyl(propan-2-yl)amino]methyl}thieno[2,3-b]pyridine-2-carboxylate
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N,N-diethylpiperidine-3-carboxamide
3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-(5-methoxyfuran-2-carbonyl)piperidine
N-(4-{4-[(1,4-dioxan-2-ylmethyl)amino]piperidin-1-yl}phenyl)benzenesulfonamide
2-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[2-(dimethylamino)-2-(thiophen-2-yl)ethyl]-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
1-methanesulfonyl-N-[3-(3-methylphenyl)phenyl]pyrrolidine-2-carboxamide
2-methoxy-N-{1-[3-(piperidine-1-carbonyl)phenyl]-1H-pyrazol-4-yl}acetamide
N-{2-[3-(4-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}benzamide
2-amino-N-[3-(benzyloxy)pyridin-2-yl]-6-methylpyrimidine-4-carboxamide
(2S)-1-(1,3-oxazole-5-carbonyl)-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
3-(piperidin-3-yl)-N-(pyrimidin-4-ylmethyl)benzamide
5-[6-amino-5-cyano-4-(thiophen-2-yl)pyridin-2-yl]-2,4-dimethyl-1H-pyrrole-3-carboxylic acid
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(2-methylbenzoyl)pyrrolidin-3-yl]methanol
ethyl 2-[4-(3-methylphenoxy)piperidin-1-yl]-1,3-oxazole-4-carboxylate
2-[(4-chlorophenyl)amino]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-cyclopropyl-5-[3-(oxolan-3-yl)-1-phenyl-1H-1,2,4-triazol-5-yl]-3,4-dihydropyrimidin-4-one
6-(2-hydroxyethyl)-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]acetamide
5-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
1-{1-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
3-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-5-(propan-2-yl)-1,2-oxazole
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
7-(5-chloropyridin-2-yl)-4-(1-methyl-1H-pyrazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-(1H-imidazol-1-yl)-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}benzamide
(4-benzyl-1-cyclooctylpiperidin-4-yl)methanol
(2S,4S)-4-[4-(2-fluoro-4-methylbenzenesulfonamidomethyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
9-(1-methyl-1H-pyrazole-5-carbonyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-{5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-yl}phenol
(1R,5R)-6-methyl-3-[4-(2-methylphenyl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
6-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}pyrazine-2-carboxamide
(2S,4S)-N-ethyl-4-(2-methylfuran-3-amido)-1-[3-(methylsulfanyl)propanoyl]pyrrolidine-2-carboxamide
2-(4-methyl-1H-imidazole-2-carbonyl)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane
3-[(2,6-dichlorophenyl)methyl]-4-(hydroxymethyl)-1,3-oxazolidin-2-one
2-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[4-(2-fluorophenyl)piperazin-1-yl]ethan-1-one