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1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-3-[2-(methylsulfanyl)benzoyl]piperidine
N-[3-(1H-imidazol-1-yl)propyl]-3-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]-N-(pyridin-3-ylmethyl)propanamide
1-[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]-2-(propan-2-ylsulfanyl)ethan-1-one
N-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-methyl-1,2,3,4-tetrahydronaphthalen-1-amine
1-{2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-3-[(methylsulfanyl)methyl]piperidine
1-(2-cyclohexylethyl)-N-methyl-N-{[1-(2-methylpropyl)piperidin-4-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methyl-2-oxo-1,3-oxazolidine-4-carboxamide
N-({7-[(2E)-3-(2,3-difluorophenyl)prop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1-phenylmethanesulfonamide
methyl (2S,4R)-1-methyl-4-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamido}pyrrolidine-2-carboxylate
2-(2-hydroxyethyl)-9-(quinoline-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl 4-(5-methyl-4-{[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methyl}-1,3-oxazol-2-yl)benzoate
1-[(6-fluoro-4-hydroxyquinolin-2-yl)methyl]-N-(3-hydroxypropyl)piperidine-3-carboxamide
1-[2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)acetyl]piperidine-4-carbonitrile
2-ethyl-N-[(5-methoxy-1H-indol-2-yl)methyl]-4-methyl-1,3-oxazole-5-carboxamide
1-(3-methoxy-1,5-dimethyl-1H-pyrazol-4-yl)-3-(2-{[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]methyl}propyl)urea
(1S,4S)-2-(2-methoxy-5-methylphenyl)-5-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
N-(5-cyclobutyl-1,3,4-thiadiazol-2-yl)-2-(1,3-thiazol-2-yl)piperidine-1-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1-methyl-1H-pyrazole-4-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-N-methyl-N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)acetamide
8-fluoro-N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-N-methyl-4-oxo-1,4-dihydroquinoline-2-carboxamide
N-[2-(2-chlorophenyl)ethyl]-1-cycloheptyl-6-oxopiperidine-3-carboxamide
1-(furan-2-ylmethyl)-N-methyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)piperidine-4-carboxamide
1-[4-(2-methylphenoxy)piperidin-1-yl]-3-(methylsulfanyl)propan-1-one
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[2-(1H-imidazol-1-yl)-1-phenylethyl]propanamide
(1R,3S,5S)-8-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octane
N-[4-({7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}methyl)phenyl]acetamide
1-[(3aR,6aR)-3a-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]-octahydropyrrolo[3,4-c]pyrrol-2-yl]-2-methoxyethan-1-one
[(3R,4R)-4-[({[2-(naphthalen-2-yl)pyrimidin-5-yl]methyl}amino)methyl]pyrrolidin-3-yl]methanol
N-[(3R,5S)-1-cyclopentyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]-4-methylpyrimidine-5-carboxamide
4-[(5-methoxy-1,3,4-thiadiazol-2-yl)methyl]-1-(2-methoxyphenyl)piperazin-2-one
(3aR,7aS)-5-methyl-2-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
2-(morpholin-4-yl)-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)pyrimidine-5-carboxamide
3-chloro-N-[2-(dimethylamino)ethyl]-4-({1-[4-(methylsulfanyl)butan-2-yl]piperidin-4-yl}oxy)benzamide
2-[4-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-N,N-bis(prop-2-en-1-yl)acetamide
(1R,2R,4R)-N-(2H-1,3-benzodioxol-5-ylmethyl)-N-(pentan-3-yl)bicyclo[2.2.1]hept-5-ene-2-carboxamide
4-[4-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-6-(propan-2-yl)pyrimidin-2-amine
3-[3-(1-benzylazetidin-2-yl)-4H-1,2,4-triazol-4-yl]pyridine
7-(3-chlorophenyl)-4-(2-fluoroethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-2-(2-methyl-1H-1,3-benzodiazol-5-yl)acetamide
1-{5H,6H,7H-cyclopenta[b]pyridin-3-ylmethyl}-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
1-(2-methoxyethyl)-4-{4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]-1H-imidazol-2-yl}pyrrolidin-2-one
4-(1-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}piperidin-3-yl)benzoic acid
N-[2-(4-fluorophenyl)ethyl]-2-methyl-N-(pyridin-3-ylmethyl)imidazo[1,2-a]pyrimidine-3-carboxamide
3-[5-(1H-imidazol-4-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-1-(morpholin-4-yl)propan-1-one
1-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-4-[5-(2-methylpropyl)-1H-pyrazol-3-yl]-1H-1,2,3-triazole
N-{[2-(3-hydroxypiperidin-1-yl)-8-methylquinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]-3-(3-methyl-1H-pyrazol-1-yl)propanamide
5-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-1H-1,2,3-benzotriazole
[(2-chlorophenyl)methyl][(6-{octahydropyrrolo[1,2-a]piperazin-2-yl}-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl)methyl]amine
5-{[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]carbamoyl}-1H-imidazole-4-carboxylic acid
{2-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-oxoethyl}urea