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(2-methoxyethyl)(methyl){[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}amine
N-(furan-2-ylmethyl)-1-methyl-N-(2-phenylethyl)piperidine-2-carboxamide
3-(3,4-dimethoxyphenyl)-1-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}propan-1-one
1-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)ethan-1-one
1-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
[(5-methoxy-1,3-benzoxazol-2-yl)methyl]({[5-(pyrimidin-2-ylsulfanyl)furan-2-yl]methyl})amine
2-{4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl}pyridine-3-carbonitrile
{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(oxan-4-ylmethyl)amine
[(3R,4R)-1-[(4-fluoro-3-methylphenyl)methyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
2,2-dimethyl-N-{1-[1-(4-oxo-4-phenylbutanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}propanamide
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-[(1r,4r)-4-hydroxycyclohexyl]piperidine-3-carboxamide
N-[2-(6-hydroxypyrimidin-4-yl)ethyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
2-{1-[2-(3-methylpyridin-2-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}benzoic acid
2-[2-(pyrrolidine-1-sulfonyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]pyridine
2-chloro-4-{[7-(cyclobutylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]methyl}-6-methoxyphenol
2-(ethylsulfanyl)-5-{1-[1-(furan-2-yl)ethyl]-1H-imidazol-2-yl}pyrimidine
4,6-dimethoxy-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}pyrimidin-2-amine
5-methyl-5-[1-(5-phenoxyfuran-2-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
ethyl 4-[3-(diphenylmethyl)-1,2-oxazole-5-amido]piperidine-1-carboxylate
5-(1-benzyl-1H-pyrazol-3-yl)-N-[(4-methoxyphenyl)methyl]-4-methyl-1,3-thiazol-2-amine
4-(cyclopropylmethyl)-1-(2-methyl-1H-1,3-benzodiazole-4-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
N-[3-(3-methyl-2,5-dioxoimidazolidin-1-yl)phenyl]-3-(1H-pyrazol-3-yl)piperidine-1-carboxamide
2-(3-chloro-4-fluorophenoxy)-1-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}ethan-1-one
2-[3-methyl-5-(3-methyl-1-propyl-1H-pyrazol-4-yl)-1H-1,2,4-triazol-1-yl]pyridine
1-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-hydroxypropan-1-one
3-methyl-1-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-3-ol
1-[(4-hydroxy-3,5-dimethylphenyl)methyl]-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol
(5S,9aS,9bS)-2-(1-methylpiperidin-4-yl)-5-[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[(1-cyclopentylpiperidin-4-yl)methyl]-N-(pyridin-3-ylmethyl)but-3-enamide
4-(3-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}pyrrolidine-1-carbonyl)pyridazine
(1R,5S,8S)-3-[(3-chloro-4-methoxyphenyl)methyl]-8-methoxy-3-azabicyclo[3.2.1]octane
N-(pyridin-4-ylmethyl)-4-{[1-(1,3-thiazol-2-ylmethyl)piperidin-4-yl]oxy}benzamide
2-[5-(3,3,3-trifluoropropyl)-1,2,4-oxadiazol-3-yl]pyridine
(1S,5R)-N-(2,4-dichlorophenyl)-7-oxo-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
5-[1-(2-chlorophenyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]-2-methyl-3,4-dihydropyrimidin-4-one
1-{[5-(3-methoxyphenyl)-1,2-oxazol-3-yl]methyl}-5-oxopyrrolidine-3-carboxylic acid
N,N-dimethyl-5-{[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]methyl}pyridin-2-amine
3-[({1-[4-(propan-2-yl)-1,3-thiazole-2-carbonyl]piperidin-4-yl}oxy)methyl]pyridine
N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
3-(dimethyl-1,2-oxazol-4-yl)-1-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]propan-1-one
5-(3-cyclopropyl-1H-pyrazole-4-carbonyl)-N-phenyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
6-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-1-methyl-1H-indole
5-({1-tert-butyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)-2-ethyl-4-methyl-1H-imidazole
3-methyl-1-{1-[4-methyl-2-(pyridin-3-yl)pyrimidine-5-carbonyl]piperidin-4-yl}butan-1-ol
(2R,6R)-11-methoxy-4-(4-methylpiperazine-1-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-(1-ethyl-1H-pyrazol-4-yl)-3-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)urea
5-{[2-(2,3-dimethoxyphenyl)-1H-imidazol-1-yl]methyl}-1,3-dimethyl-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-{3-[(pyridin-3-yl)amino]propyl}pyrazine-2-carboxamide
3-[2-(furan-2-yl)azepane-1-carbonyl]-1-methyl-1,2,5,6,7,8-hexahydroquinolin-2-one
(3S,4S)-4-cyclopropyl-1-(2-methylpyrimidin-4-yl)pyrrolidine-3-carboxylic acid