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4-[(4-methyl-5-{1-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]morpholine
N-(4-methylphenyl)-4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carboxamide
3-(1-butyl-1H-imidazol-2-yl)-1-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]piperidine
3-hydroxy-S-[2-(1H-pyrrole-2-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]butane-1-sulfonamido
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
2-[3-({3-[benzyl(methyl)amino]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
1-(5-methyl-1,2-oxazole-3-carbonyl)-4-[2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-[(1-methyl-2,3-dihydro-1H-indol-5-yl)methyl]acetamide
4-(cyclopropylmethyl)-1-(6-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
1-[(2-fluorophenyl)methyl]-3-hydroxy-3-({methyl[(4-methylphenyl)methyl]amino}methyl)piperidin-2-one
4-(4-ethoxy-3-methylphenyl)-1-[2-(hydroxymethyl)piperidin-1-yl]butan-1-one
N-[(5-methylthiophen-2-yl)methyl]-3-[2-(propan-2-yl)-2,5-dihydro-1H-pyrrole-1-carbonyl]aniline
2-{1-cyclohexyl-4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
6-ethyl-N4-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-5-methylpyrimidine-2,4-diamine
1-butyl-4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-methyl-2-oxo-6-(propan-2-yl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,2-dihydropyridine-3-carboxamide
8-(4-chlorobenzoyl)-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
4-(5-methylpyridin-2-yl)-1-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidin-4-ol
2-{4-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]morpholin-3-yl}-N-(pyridin-4-ylmethyl)acetamide
1-{4-[(3-fluorophenyl)methyl]-1,4-diazepan-1-yl}-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
3-(1-methylpiperidin-3-yl)-1-[4-(1H-pyrrole-2-carbonyl)piperazin-1-yl]propan-1-one
1-benzyl-6-[(4-chlorophenyl)amino]-1H,4H,5H,8H-imidazo[4,5-e][1,3]diazepine-4,8-dione
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-6-(furan-3-yl)-N-methylpyridine-3-carboxamide
2-ethyl-4-[3-(4-methoxyphenoxymethyl)piperidine-1-carbonyl]pyridine
2-(4-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-(propan-2-yl)piperazin-2-yl)ethan-1-ol
1-{2-[(3-fluorophenyl)methyl]morpholin-4-yl}-2-[methyl(pyridin-2-ylmethyl)amino]ethan-1-one
1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(1H-pyrrol-1-yl)butan-1-one
3-(2-ethyl-1H-1,3-benzodiazol-1-yl)-N-methyl-N-(1H-pyrazol-3-ylmethyl)propanamide
N-(2,5-dimethylphenyl)-N'-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]propanediamide
1-[1'-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
3-cyclopropyl-N-[2-(dimethylamino)ethyl]-N-[(5-methylthiophen-2-yl)methyl]-1H-pyrazole-5-carboxamide
3-(1-ethyl-1H-pyrazol-4-yl)-4-phenyl-4H-1,2,4-triazole
2-(dimethylamino)-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-(3-methylphenyl)acetamide
3-(4-cyano-2-fluorophenyl)-1-(2-methoxyethyl)-1-(1-methylpiperidin-4-yl)urea
2-(1-{[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}pyrrolidin-2-yl)-1-methyl-1H-1,3-benzodiazole
4-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-2-methyl-1,4-oxazepane
1-(furan-3-ylmethyl)-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-4-carboxamide
5-ethyl-3-[(2E)-3-phenylprop-2-en-1-yl]-5-(piperidin-4-yl)imidazolidine-2,4-dione
6-methyl-N-[(1S,3S)-3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}cyclopentyl]pyridine-2-carboxamide
N-[(3S,4R)-4-(propan-2-yl)-1-{thieno[3,2-d]pyrimidin-4-yl}pyrrolidin-3-yl]acetamide
3-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
N-[(3S,4R)-4-methoxyoxolan-3-yl]-3-(2-methyl-1H-indol-1-yl)propanamide
3-[3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]-1-methyl-1-(quinoxalin-2-ylmethyl)urea
6-(1-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)-2-methylpyrimidin-4-ol
3-[2-(4-acetyl-1,4-diazepan-1-yl)-2-oxoethyl]-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidine-2,5-dione
9-(1-ethyl-1H-pyrazole-3-carbonyl)-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-(3-hydroxy-3-methylbut-1-yn-1-yl)benzamide
N-{4-[(2-methoxyethyl)carbamoyl]phenyl}-3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidine-1-carboxamide
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-3-methoxy-4-methylbenzamide
4-ethyl-3-{1-[4-(1H-imidazol-1-yl)benzoyl]piperidin-3-yl}-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one