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3-(2-fluorophenyl)-1-(2-methoxyethyl)-3-{2-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
methyl 5-{[(2-chloro-4,5-dimethoxyphenyl)methyl]amino}-3-cyclobutaneamido-1-[2-(pyridin-2-yl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]-N-phenylpyrimidin-2-amine
N-[(2-chloropyridin-3-yl)methyl]-1-cyclopentyl-N-methyl-5-oxopyrrolidine-3-carboxamide
5-acetyl-N-[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-({[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]amino}methyl)piperidin-2-one
8-methoxy-2-(morpholin-4-ylmethyl)quinoline
4-(4-methyl-1,3-oxazole-5-carbonyl)-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine
1-[3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-3-phenoxypropan-1-one
2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}butanamide
7-(3-chlorophenyl)-4-(1,4-dioxane-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-{[5-(2-methylpropyl)thiophen-2-yl]methyl}-4-(pyrrolidine-1-sulfonyl)piperazine
2-(4-fluorophenoxymethyl)-N-methyl-N-[(1-methylpyrrolidin-2-yl)methyl]-1,3-oxazole-4-carboxamide
N-[(3R,4S)-1-(2-methoxyethyl)-4-(propan-2-yl)pyrrolidin-3-yl]-2-(4H-1,2,4-triazol-4-yl)acetamide
3-{2-[(2,1,3-benzoxadiazol-5-ylmethyl)amino]propyl}-3,4-dihydroquinazolin-4-one
2-[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-(5-cyclopropyl-1,3,4-thiadiazol-2-yl)-1-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}urea
N-{2-[7-(2H-1,3-benzodioxol-5-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}oxolane-2-carboxamide
2-{4-[(2,3-dimethoxyphenyl)methyl]-1-(3-methylbutyl)piperazin-2-yl}ethan-1-ol
2-methyl-N-[(2S)-oxolan-2-ylmethyl]-7-(1,3-thiazol-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-[2-(3-fluorophenyl)ethyl]-11-{[(5-methylpyrazin-2-yl)methyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-(3-benzyl-1H-1,2,4-triazol-5-yl)-4-(pyridin-2-yl)piperazine-1-carboxamide
1-[2-(1H-imidazol-4-yl)ethyl]-2-(4-methoxy-2,3-dimethylphenyl)-1H-imidazole
methyl (2S,4S)-4-{4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-amido}-1-methylpyrrolidine-2-carboxylate
2-(cyclopropylmethyl)-8-(4-hydroxy-3-methoxybenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(2-aminoethyl)-5,6-dimethyl-N-[3-(pyridin-4-yl)propyl]thieno[2,3-d]pyrimidin-4-amine
3-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-2,2-dimethylpropan-1-ol
9-[2-(3-fluorophenyl)acetyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-methyl-1H-imidazole-5-carboxamide
2-(2,6-dimethoxypyridin-3-yl)-2-[4-(pyridin-2-yl)piperazin-1-yl]acetic acid
2-[benzyl({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)amino]ethan-1-ol
5-phenyl-N-[3-(pyridin-3-yloxy)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-(cyclopropylmethyl)-N-ethyl-5-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-[3-(4-ethoxyphenoxymethyl)-5-(methoxymethyl)-1H-1,2,4-triazol-1-yl]-4-methylpyridine
7-(cyclobutylmethyl)-2-[3-oxo-3-(pyrrolidin-1-yl)propyl]-2,7-diazaspiro[4.5]decan-6-one
1-[(2-methylphenyl)methyl]-N-(2-phenoxyethyl)-1H-1,2,3-triazole-4-carboxamide
2-[2-(3-methoxypropyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]pyridine-3-carboxamide
1-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)-6-methoxyhexan-1-one
1-(4-{3-[methyl(2-phenylethyl)amino]piperidine-1-carbonyl}phenyl)pyrrolidin-2-one
1-methyl-1-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}urea
1-(4-hydroxy-1,2-oxazolidin-2-yl)-3-(3-hydroxyquinoxalin-2-yl)propan-1-one
N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-4-(pyridin-2-yl)pyrimidin-2-amine
5-[(cyclopentylamino)methyl]-N-methyl-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-benzyl-4-[1-(pyrrolidin-1-yl)cyclopentanecarbonyl]-1,4-diazepan-6-ol
N-[(3R,5S)-5-(ethylcarbamoyl)-1-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl]-6-oxo-1,6-dihydropyridine-3-carboxamide
1-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-N-ethyl-N-(pyridin-4-ylmethyl)piperidin-3-amine
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-(3-methylfuran-2-carbonyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
(2S,4S)-4-({[4-(benzyloxy)phenyl]methyl}amino)-N-ethyl-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
N-cyclopropyl-1-[1-(naphthalen-2-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
(1R,3S)-3-(2-hydroxyethoxy)-7-(2-methoxy-3-methylbenzoyl)-7-azaspiro[3.5]nonan-1-ol