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3-{3-[({2-[(4-methylpyridin-2-yl)amino]ethyl}amino)methyl]-1H-indol-1-yl}propanamide
4-{1-[(3,4-dimethoxyphenyl)methyl]piperidin-3-yl}-5-phenyl-2-(pyridin-4-yl)pyrimidine
1-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)-3-(3-chloro-1,2-oxazol-5-yl)propan-1-one
4-{[3-(3-methoxybenzoyl)piperidin-1-yl]methyl}phenol
2-[(3-{[2-(1H-imidazol-4-yl)ethyl]carbamoyl}phenyl)amino]acetic acid
4-(3-hydroxy-3-methylbutyl)-N-(3,3,3-trifluoropropyl)benzamide
10-methoxy-5-{[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
6-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyrazine-2-carboxamide
1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(piperidine-1-carbonyl)piperidine
3-{[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]methyl}benzonitrile
2-[4-(3-cyclopropyl-1H-pyrazole-5-carbonyl)piperazin-1-yl]-1,3-benzothiazole
N-[3-(ethylcarbamoyl)-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
[(5-ethylfuran-2-yl)methyl]({[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
7-(cyclopropylmethyl)-2-(2,4-difluorobenzenesulfonyl)-2,7-diazaspiro[4.5]decan-6-one
2-(pyridin-4-yl)-N-[2-(1H-1,2,4-triazol-1-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-(1-benzyl-3-oxopiperazin-2-yl)-N-[2-(2-methoxyphenyl)ethyl]acetamide
1-(2,3-dihydro-1-benzofuran-5-carbonyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
3-(5-methylfuran-2-yl)-N-[(4-methylphenyl)(pyridin-4-yl)methyl]-1H-pyrazole-5-carboxamide
4-methoxy-N-{1-[1-(pent-4-enoyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
1-{1-[(4-methylphenyl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
(3aR,5S,6S,7aS)-2-[(4,5-dichlorothiophen-2-yl)sulfonyl]-octahydro-1H-isoindole-5,6-diol
(4aR,7aS)-1-(2-methoxyacetyl)-4-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2-{[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl][(5-methylthiophen-2-yl)methyl]amino}ethyl)dimethylamine
2-[(1,3-benzothiazol-2-yl)amino]-1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethan-1-one
2-[({1-[3-(3-fluorophenyl)phenyl]piperidin-4-yl}amino)methyl]-6-methyl-3,4-dihydropyrimidin-4-one
3-(4-chlorophenyl)-1-[4-(2-hydroxyethyl)piperazin-1-yl]-3-phenylpropan-1-one
7,7-dimethyl-2-(1-methyl-1H-imidazol-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-ethyl-4-[1-(2-hydroxyethyl)-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
3-methyl-4-{[3-(pentan-3-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-5-phenyl-1,2-oxazole
1-cyclohexyl-N-(2-hydroxyethyl)-N-(1,3-thiazol-2-ylmethyl)piperidine-4-carboxamide
3-{3-[3-(4-fluorophenyl)oxolan-3-yl]-1,2,4-oxadiazol-5-yl}-1,4,6-trimethyl-1,2-dihydropyridin-2-one
N,5-dimethyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-1-benzofuran-2-carboxamide
4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-N-(cyclopropylmethyl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
3-{spiro[azepane-4,2'-chromene]-1-ylmethyl}phenol
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]acetamide
2-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]benzonitrile
1-ethyl-5-[2-(4-fluorophenyl)azetidine-1-carbonyl]-3-(propan-2-yl)-1H-pyrazole
5-methyl-2-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}-1H-indole
N-[(2-{4-[5-(methoxymethyl)furan-2-amido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
4-amino-2-{4-[2-(benzyloxy)ethyl]piperazin-1-yl}pyrimidine-5-carbonitrile
3-({2-[1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
3-(4-fluorophenyl)-3-{[3-(5-methylfuran-2-yl)-1H-pyrazol-5-yl]formamido}propanoic acid
3-{[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]sulfamoyl}-N-(pyridin-4-ylmethyl)benzamide
N-[(4-fluorophenyl)methyl]-N-methyl-2-[1-methyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]acetamide
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-1-(pyridin-2-yl)piperidine-3-carboxamide
(2R,4S)-1-[2-(2-fluorophenyl)benzoyl]-4-hydroxypiperidine-2-carboxylic acid
N-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-[(trimethyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
N-(2,4-dimethoxyphenyl)-3-(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-4-yl)propanamide
(3S,4S)-4-methyl-1-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}piperidine-3,4-diol
methyl({[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}){[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amine