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N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-N-methyl-2-(pyrrolidin-1-yl)-5,6,7,8-tetrahydroquinazoline-4-carboxamide
4-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-3-fluoropyridine
(4-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methanol
(1-methyl-1H-imidazol-2-yl)({1-[2-methyl-2-(morpholin-4-ylmethyl)propyl]piperidin-4-yl})methanol
cyclopentyl 4-({[2-(pyridin-3-yl)ethyl]carbamoyl}amino)benzoate
1-[(3-fluorophenyl)methyl]-3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]urea
(1s,4s)-4-[2-(7-fluoro-2-methyl-1H-indol-3-yl)acetamido]cyclohexane-1-carboxylic acid
N-{4-[2-(1,2-benzoxazol-3-yl)acetamido]-2-methoxyphenyl}-3-methylbutanamide
1-{6-phenylimidazo[2,1-b][1,3]thiazole-3-carbonyl}-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
methyl 3-[(2,6-difluorophenyl)methyl]-7-oxo-9-[2-(pyridin-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
6-[3-(morpholin-4-ylmethyl)phenyl]pyridine-2-carboxamide
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-methyl-N-[(3-methyloxetan-3-yl)methyl]-1H-pyrazole-3-carboxamide
6-methoxy-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]pyrimidin-4-amine
1-{3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}-3,3,3-trifluoropropan-1-one
2-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-N-methylpyridine-3-carboxamide
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[1-(2-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethan-1-one
[(2S,4R,5R)-5-(4-chlorophenyl)-1-ethyl-4-({[(3-methoxyphenyl)methyl]amino}methyl)-2-methylpyrrolidin-2-yl]methanol
4-{1-[1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidin-4-yl]piperidine-4-carbonyl}morpholine
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(2-methyl-1,3-thiazol-4-yl)methyl]benzamide
1-(cyclohexylmethyl)-3-hydroxy-3-({[(3-methyl-1H-pyrazol-5-yl)methyl]amino}methyl)piperidin-2-one
N-[(4-fluorophenyl)(pyridin-4-yl)methyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-6-(3-fluorophenyl)-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
3-(4-chlorophenyl)-1-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
3-[4-methoxy-3-(propan-2-yloxy)phenyl]-6-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridine
(1S,6R)-9-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
3-{1-[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]ethyl}-1-[2-(trifluoromethoxy)phenyl]urea
N-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]oxolane-3-carboxamide
1-(2-methylpropyl)-N-[2-(3-methylpyridin-2-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
3-(but-2-yn-1-yl)-5-[1-(3-methylbutyl)piperidin-4-yl]-5-(2-phenylethyl)imidazolidine-2,4-dione
6-{1-[2-(7-fluoro-2-methyl-1H-indol-3-yl)acetyl]piperidin-3-yl}-3,4-dihydropyrimidin-4-one
N-[2-(4-chlorophenyl)ethyl]-2-{[(dimethyl-1,3-thiazol-5-yl)methyl]amino}acetamide
4-{1-[2-(3,4-dimethoxyphenyl)ethyl]-1H-imidazol-2-yl}-2-methyl-1,3-oxazole
4-(2,6-dimethylpyridin-3-yl)-N-[1-(pyridin-3-yl)propan-2-yl]pyrimidin-2-amine
1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(1H-pyrazol-1-yl)propan-1-one
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[3-(1H-1,2,3-triazol-1-yl)propyl]benzamide
3-[(2-methyl-1,4-oxazepan-4-yl)sulfonyl]-N-[(2-methylpyridin-4-yl)methyl]benzamide
3-{2-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
N'-cycloheptyl-N-[4-(morpholin-4-yl)butan-2-yl]butanediamide
N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
2-(4-methoxyphenyl)-N-[1-(3-phenylpropyl)piperidin-3-yl]acetamide
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-6-(2-hydroxyethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-(thiophen-2-ylmethyl)-5-(thiophen-3-yl)-1H,4H-pyrazolo[3,4-d]imidazole
2-[(4-methanesulfonylphenyl)methyl]-octahydropyrrolo[1,2-a]piperazine
7-{[4-(propan-2-yl)phenyl]methyl}-2-(1,3-thiazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
3-(1-methyl-1H-imidazol-2-yl)-1-[4-(2-methylpropyl)benzoyl]piperidine
(2S)-2-({5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}amino)-4-methylpentan-1-ol
1-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-dihydropyridin-2-one
N-[(1-methylpiperidin-3-yl)methyl]-2-propyl-1,3-thiazole-4-carboxamide
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
N-[(5-methylfuran-2-yl)methyl]-1-[3-(2-methylpyrimidin-4-yl)phenyl]piperidin-4-amine