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2-phenyl-N-[1-(1H-pyrazol-1-yl)propan-2-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
5-{2-azabicyclo[2.2.1]heptane-2-carbonyl}-N-(cyclohexylmethyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
N-benzyl{[1-(3-cyanopyridin-2-yl)piperidin-4-yl]amino}sulfonamide
2-[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]-5-methyl-1H-1,3-benzodiazole
5-(3-chlorophenyl)-3-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]-1,2,4-triazine
1-({4-[(4-fluoro-3-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)-4-(pyridin-3-yl)piperidin-4-ol
1-(5-methyl-1,3-oxazole-4-carbonyl)-4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-chloro-4-[6-(cyclopropylamino)pyridazin-3-yl]benzamide
N-methyl-2-(2-oxopiperidin-1-yl)-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]acetamide
N-[(2-aminopyrimidin-5-yl)methyl]-4-(cyclobutylsulfamoyl)-N-methylbenzamide
2-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}acetic acid
N-[2-(1H-indol-1-yl)ethyl]-6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-amine
(1S,5R)-3-(1-benzylpiperidin-4-yl)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-[1-(1H-pyrazol-1-yl)propan-2-yl]pyridin-2-amine
3-{[1-(1-benzofuran-5-ylmethyl)piperidin-4-yl]methyl}-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-methoxypropan-1-one
2-{1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]piperidin-2-yl}acetic acid
6-[4-(benzyloxy)piperidine-1-carbonyl]-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
N-[2-(2,4-dimethylphenoxy)ethyl]-N-methyl-3-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]propanamide
ethyl 4-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]piperazine-1-carboxylate
5-[2-fluoro-6-(propan-2-yloxy)phenyl]-2,3-dihydro-1H-indol-2-one
9-(2-methyl-1H-pyrrole-3-carbonyl)-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1H-indole
(3E)-1-[2-amino-7-methyl-4-(3-methylphenyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pent-3-en-1-one
8-[(4-fluoro-3-methoxyphenyl)methyl]-1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3-propyl-1H-pyrazole-5-carboxamide
1-({3-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]phenyl}methyl)-1H-pyrazole
(3S,9aR)-8-{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-chloro-4-[({[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]-6-methoxyphenol
3-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]pyridin-2-ol
ethyl 4-[5-(4-cyclohexylphenyl)-1,2,4-triazin-3-yl]piperazine-1-carboxylate
(3S,4S)-1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-4-(naphthalen-2-yl)piperidin-3-ol
1-cyclopropanecarbonyl-N-[(2-methylpyridin-4-yl)methyl]piperidine-4-carboxamide
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[2-(oxan-4-yl)ethyl]acetamide
N,N-dimethyl-9-oxo-8-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecane-2-sulfonamide
methyl 3-({5-[2-(4-chlorophenoxy)acetyl]-1-(cyclopropylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}formamido)propanoate
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-(thiophen-2-yl)butanamide
1-{1-[(4-hydroxy-5-methoxypyridin-2-yl)methyl]-4-phenylpiperidin-4-yl}ethan-1-one
N-(1H-indol-4-ylmethyl)-1-(2-methoxyethyl)-6-oxopiperidine-3-carboxamide
1-{1-[2-(carbamoylamino)acetyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
8-[5-(ethoxymethyl)-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl]quinoline
N-[(2-ethoxyphenyl)methyl]-N-ethyl-4-methanesulfonylbenzamide
2-{4-[(2-chloro-3,4-dimethoxyphenyl)methyl]-1-(3-methylbutyl)piperazin-2-yl}ethan-1-ol
3-[3-(4-ethylpiperazin-1-yl)propyl]-8-propanoyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(2-chloro-4-fluorophenyl)-2-(thiomorpholin-4-yl)acetic acid
2-(4-methoxyphenoxymethyl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-1,3-oxazole-4-carboxamide
1-(1-phenyl-1H-1,2,3-triazole-5-carbonyl)-3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
3-{5-[1-(2-phenylethyl)-1H-imidazol-2-yl]thiophen-3-yl}prop-2-yn-1-ol
4-{3-[3-(trimethyl-1H-pyrazol-4-yl)propanamido]propyl}-1,2,5-oxadiazole-3-carboxylic acid
2-(2-hydroxyethyl)-8-(2,3,4-trifluorobenzoyl)-2,8-diazaspiro[5.5]undecan-3-one