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1-[1'-(2,4-difluorobenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
3-{1-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]piperidin-3-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-benzyl-3-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-N-methyl-6-phenylpyridin-2-amine
2-(1-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)-1,3-benzoxazole
N-(1-hydroxy-2-methylpropan-2-yl)-5-methyl-4-{[(3S)-2-oxoazepan-3-yl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
(4aS,7aR)-N-butyl-4-[2-(dimethylamino)acetyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
4-[4-(4-cyclohexylpiperazin-1-yl)piperidin-1-yl]-5-propylpyrimidine
1-(3-phenylpropyl)-4-(1H-pyrrole-3-carbonyl)-1,4-diazepane
2-(3,4-dimethoxyphenyl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-cyclobutanecarbonyl-4'-(4-methylpentyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-butyl-N-methyl-3-[(4-methyl-3-phenylpiperazin-1-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide
(4aR,8aS)-N,N-dimethyl-1-(2-methylbenzoyl)-decahydro-1,6-naphthyridine-6-sulfonamide
(4aS,7aR)-1-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]-2-(trimethyl-1H-pyrazol-1-yl)ethan-1-one
{1-[1-(2-methylpentyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methanol
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[2-(3-methoxyphenyl)pyrrolidin-1-yl]ethan-1-one
4-(1-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-3-carbonyl)morpholine
4-[3-(propan-2-yl)-1H-pyrazol-5-yl]-1-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}piperidine
8-(5-carboxypyridin-2-yl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
5-[methyl(pyrimidin-4-ylmethyl)amino]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-benzyl-N-(cyclobutylmethyl)-4-hydroxy-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N'-(3-fluorophenyl)-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]ethanediamide
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
6-(2-chlorophenyl)-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-benzyl-8-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
5-methyl-4-(1-methyl-1H-pyrazol-4-yl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrimidin-2-amine
1-[(4aR,8aS)-6-[4-(trifluoromethyl)benzoyl]-decahydro-1,6-naphthyridin-1-yl]-3-(2H-1,3-benzodioxol-5-yl)propan-1-one
3-cyclohexyl-N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N-methyl-1H-pyrazole-4-carboxamide
(3R)-1-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)pyrrolidin-3-ol
1-(2-{[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]amino}ethyl)-1,2,3,6-tetrahydropyridazine-3,6-dione
2-(2H-1,3-benzodioxol-5-yl)-1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
(2S,4R)-4-amino-1-[3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)propanoyl]-N-methylpyrrolidine-2-carboxamide
3-[4-chloro-2-(trifluoromethyl)phenyl]-1-{[4-(hydroxymethyl)oxan-4-yl]methyl}-1-methylurea
N-{1-[7-(5-acetylthiophene-2-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-3-methylbutyl}-2-(dimethylamino)acetamide
methyl 3-(3-fluorobenzoyl)-9-[3-(1-methyl-1H-pyrazol-4-yl)propoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-[(2-{[3-(azepan-1-yl)propyl](methyl)carbamoyl}phenyl)amino]acetic acid
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(1S,5R)-3-(4-methylpent-3-en-1-yl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{9-methyl-3,9-diazaspiro[5.6]dodecan-3-yl}quinoline-4-carboxylic acid
9-[(3-methylpyridin-4-yl)methyl]-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
(1S,5R)-6-(cyclobutylmethyl)-3-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
4-{[2-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]methyl}-1-methylpiperidin-4-ol
4-phenoxy-1-(3-phenylpropyl)piperidine-4-carboxylic acid
1-(diphenylmethyl)-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
3-[1-cyclohexyl-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-5-yl]-N,N-dimethylpropanamide
[(1,3-dimethylpyrrolidin-3-yl)methyl][(2-fluoro-4-methoxyphenyl)methyl]methylamine
4-benzyl-3-[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(1,3-benzothiazol-2-ylmethyl)-1-(1,3,4-thiadiazol-2-yl)urea
1-(2-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-2-yl}ethyl)-4-methylpiperazine
2-cyclopropyl-8-(2-methyl-6-oxo-1,6-dihydropyrimidine-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one