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6-{1-oxaspiro[4.4]nonan-3-yl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
6-ethyl-2-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]quinoline-4-carboxamide
butyl 3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxylate
3-({[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)-2,2-dimethylpropan-1-ol
N-benzyl{[3-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]amino}sulfonamide
4-(2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-1,3-oxazole-4-carbonyl)-1,4-diazepan-2-one
8-[4-(1H-imidazol-1-yl)butanoyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
5-{[(4aS,8aR)-2-oxo-1-(2-phenylethyl)-decahydro-1,6-naphthyridin-6-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
N-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
1-(2-methoxyphenyl)-4-[3-(2-methoxyphenyl)propanoyl]piperazin-2-one
(2S,4S)-N,N-diethyl-4-{4-[(2-hydroxyethyl)(methyl)amino]benzamido}-1-methylpyrrolidine-2-carboxamide
2-{4-[(2-chlorophenyl)methyl]-1-[(4-ethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-4-methyl-N-(oxolan-2-ylmethyl)-1,2,3-thiadiazole-5-carboxamide
2-(cyclopropylmethyl)-8-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
N-{2-[3-(ethylsulfanyl)-5-oxo-4,5-dihydro-1,2,4-triazin-6-yl]phenyl}-6-oxopiperidine-3-carboxamide
2-(2H-1,2,3-benzotriazol-2-yl)-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)acetamide
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
3-(but-2-ynoyl)-9-methoxy-N-[(4-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-[2-(2,6-difluorophenyl)ethyl]-1-[(2-methyl-1,3-thiazol-4-yl)methyl]piperidine
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-9-oxo-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraene-10-carboxamide
3-phenyl-1-[4-(piperidin-1-ylmethyl)benzoyl]piperazine
N-cyclopropyl-3-[5-(3-phenyl-1,2,4-oxadiazol-5-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanamide
3-methyl-8-({2-phenylimidazo[1,2-a]pyrimidin-3-yl}methyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3S,4R)-4-(2-methylphenyl)-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}pyrrolidine-3-carboxylic acid
6-methyl-N-[(5-methyl-2-{3-[2-(4-methylphenoxy)acetamido]phenyl}-1,3-oxazol-4-yl)methyl]pyridine-2-carboxamide
N-[4-fluoro-3-({[3-(pyrrolidin-1-yl)propyl]carbamoyl}amino)phenyl]propanamide
(3S,9aR)-3-(4-aminobutyl)-8-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N3-[3-(dimethylamino)-2,2-dimethylpropyl]-N5-(furan-2-ylmethyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-N-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}propanamide
3-cyclopropyl-1-{4-[4-(1-hydroxycyclopentyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}propan-1-one
N-(1-{[2-(ethylamino)pyrimidin-5-yl]methyl}piperidin-4-yl)methanesulfonamide
3-[4-(2-methylphenyl)-3-oxopiperazin-1-yl]propanoic acid
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[(1s,4s)-4-hydroxycyclohexanecarbonyl]pyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
N-{imidazo[1,2-a]pyridin-2-ylmethyl}-6-methyl-4-oxo-2-(2-phenylethyl)-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
2-{4-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-cyclopentylpiperazin-2-yl}ethan-1-ol
6-(2-methoxyphenyl)-N-[2-(1H-pyrazol-1-yl)ethyl]pyridazin-3-amine
(4-{[1-(2,3-dihydro-1-benzofuran-5-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
3-(2-cyclopropyl-1,3-dioxo-2,3-dihydro-1H-isoindol-5-yl)-1-[1-(3-methylpyridin-2-yl)propan-2-yl]urea
1-(1-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
(3aS,6aS)-2-acetyl-5-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-methyl-1-[(4-phenyl-1,3-thiazol-2-yl)methyl]-N-[2-(pyridin-2-yl)ethyl]piperidin-3-amine
3-[2-(dimethylamino)ethyl]-5-(3-methylbutyl)-5-(1-{2-[4-(methylsulfanyl)phenyl]acetyl}piperidin-4-yl)imidazolidine-2,4-dione
5-(3-acetylphenoxymethyl)-N-[4-(1H-pyrazol-1-yl)butan-2-yl]-1,2-oxazole-3-carboxamide
({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)({[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl})(pyridin-3-ylmethyl)amine
2,5-difluoro-N-[1-(7-{[4-(propan-2-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]benzamide
N-(2-hydroxybutyl)-5-(3-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-chloro-N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-4-fluoro-1-benzothiophene-2-carboxamide
6-(2,5-dimethylphenyl)-N-(6-hydroxy-6-methylheptan-2-yl)imidazo[2,1-b][1,3]thiazole-3-carboxamide