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7-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-2-oxa-7-azaspiro[4.5]decan-8-one
(1R,2R,6S,7S)-4-[6-(morpholine-4-carbonyl)pyrazin-2-yl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane
1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-3-phenylpiperidine
(2S,4R)-1-[(2,5-difluorophenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]-N,N-dimethylpyrrolidine-2-carboxamide
4-{[(6-methylpyridin-2-yl)methyl]amino}-1-(2-phenylethyl)pyrrolidin-2-one
[(3R,4S)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-3-yl]methanol
1-cyclopentanecarbonyl-N-[4-(3-methoxyphenyl)phenyl]piperidine-3-carboxamide
2-[(2-hydroxyethyl)({3-[5-(1-methyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]propyl})amino]ethan-1-ol
2-(5-fluoro-2-methoxyphenyl)-2-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}acetic acid
1-[2-({[2-(piperidin-1-yl)ethyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
3-(1H-1,3-benzodiazol-1-yl)-N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]propanamide
(4aS,8aR)-6-(3,6-dimethylpyrazin-2-yl)-1-(piperidin-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(3-methyl-1,2-oxazol-5-yl)acetamide
2-amino-8-{4-[3-(1H-imidazol-1-yl)propoxy]phenyl}-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
(4aR,7aS)-1-benzyl-4-{[5-(hydroxymethyl)furan-2-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[4-methyl-2-(piperidin-1-yl)pyrimidine-5-carbonyl]-1-phenylpiperazin-2-one
4-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]-1,4-oxazepane
1-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}-2-(1,2,3,6-tetrahydropyridin-4-yl)ethan-1-one
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
(1S,5R)-6-methyl-3-[4-(methylamino)-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl]-3,6-diazabicyclo[3.2.2]nonan-7-one
4-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]piperazin-2-one
1-(furan-2-ylmethyl)-N-[2-(1H-indol-1-yl)ethyl]-N-methylpiperidine-3-carboxamide
N-[(2R,3R)-1'-(1-ethyl-1H-pyrazole-4-carbonyl)-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
(4aS,8aS)-2-ethyl-7-(6-ethyl-2-methylpyrimidin-4-yl)-decahydro-2,7-naphthyridin-4a-ol
2-({5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)pyridin-3-ol
(5S,9aS,9bS)-5-(5-acetylthiophen-3-yl)-2-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-({3-methoxy-4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]-4-(trifluoromethoxy)benzene-1-sulfonamide
2-(1,2-benzoxazol-3-yl)-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]acetamide
3-(1,2-oxazinan-2-yl)-N-[3-(2-phenylacetamido)phenyl]propanamide
3-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-N-[(4-methoxyphenyl)methyl]propanamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
N-methyl-3-(2-{[({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)carbamoyl]amino}phenyl)propanamide
2-ethyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]pyrimidine-5-carboxamide
2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)acetamide
N-[1-(thian-4-yl)piperidin-4-yl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
3-{[(2S,4S)-4-amino-1-methylpyrrolidin-2-yl]formamido}-N-cyclohexylpropanamide
1-[2-(4-methoxyphenyl)ethyl]-N-[(2-methoxyphenyl)methyl]-N-methyl-6-oxopiperidine-3-carboxamide
4-(2,3-dihydro-1H-inden-5-yloxy)-1-(pyridazin-3-yl)piperidine-4-carboxylic acid
5-(2-fluorophenyl)-N-[(3,4,5-trimethoxyphenyl)methyl]-1,2,4-triazin-3-amine
2-methoxy-1-[1'-(4-methylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
N-{3-[1-(cyclohex-2-en-1-yl)-1,2,5,6-tetrahydropyridin-3-yl]-1-methyl-1H-pyrazol-5-yl}-2-methoxyacetamide
6-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-3-yl)-2-methylpyrimidin-4-ol
3-(piperidine-1-sulfonyl)-N-[2-(pyrazin-2-yl)ethyl]benzamide
(1S,5R)-6-benzyl-3-[(2-methyl-1,3-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl 2-(furan-3-yl)-1H-1,3-benzodiazole-6-carboxylate
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
1-{3-[({[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}amino)methyl]pyridin-2-yl}piperidin-3-ol
2-chloro-4-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]phenol
1-phenoxy-2-(4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)propan-2-ol
[(2S,4R)-4-(dimethylamino)-1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)pyrrolidin-2-yl]methanol