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3-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}-1-(2-methyl-1-benzofuran-5-yl)urea
N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-ethyl-N-methyl-6-[methyl(quinolin-5-ylmethyl)amino]pyridine-3-carboxamide
(1S,5R)-6-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-(2-phenylphenyl)-4-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]piperazin-2-one
(1R,2R,6S,7S)-4-[1-(1-phenylethyl)-1H-1,2,3,4-tetrazol-5-yl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane
3-(2-methoxyethyl)-5-[(3-methoxyphenyl)methyl]-5-{1-[(3-methylthiophen-2-yl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
(2R,3R,6R)-5-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
6-[4-(1-methyl-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]pyrazine-2-carboxamide
N-(2-{[2-(1H-imidazol-2-yl)phenyl]formamido}ethyl)pyridine-3-carboxamide
1-(4-{4-[(2-methoxyphenyl)amino]piperidin-1-yl}phenyl)pyrrolidin-2-one
3-[4-(6-hydroxypyrimidin-4-yl)piperidine-1-carbonyl]-N,N-dimethylpiperidine-1-carboxamide
4-(2-methylpropyl)-3-(2-oxo-2-{4-[(2-oxopyrrolidin-1-yl)methyl]piperidin-1-yl}ethyl)piperazin-2-one
5-(methoxymethyl)-N-[(3-methylpyridin-2-yl)methyl]furan-2-carboxamide
4-[4-(furan-2-yl)butan-2-yl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-(2-{[ethyl(propyl)amino]methyl}phenyl)-3H,4H,5H,6H,7H,8H,9H-cyclohepta[d]pyrimidin-4-one
N-(1,4-dioxan-2-ylmethyl)-N-methyl-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}-N-(2-methylphenyl)piperidine-1-carboxamide
1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(2,2,6,6-tetramethylpiperidin-4-yl)ethan-1-one
(3S,4R)-4-methyl-1-(quinoxaline-6-carbonyl)piperidine-3,4-diol
1-(1-benzothiophen-2-ylmethyl)-N-[3-(1H-pyrazol-5-yl)phenyl]piperidine-4-carboxamide
3-(2-{6-[(3-methoxyphenyl)methoxy]-3-oxo-4-(2-phenylethyl)-1,4-diazepan-1-yl}-2-oxoethyl)-1,3-thiazolidine-2,4-dione
5-ethyl-4-[3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]-2-methylpyrimidine
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-methyl-N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}benzamide
cyclopentyl 4-{2-[5-(1-aminoethyl)-4H-1,2,4-triazol-3-yl]acetamido}benzoate
N-(1,1-dioxo-1λ6-thiolan-3-yl)-3-(5-methylthiophen-2-yl)-N-(prop-2-en-1-yl)-1H-pyrazole-5-carboxamide
N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-5-(3-methoxyphenoxymethyl)-1,2-oxazole-3-carboxamide
3-(1-methyl-1H-pyrrol-2-yl)-N-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)-1H-pyrazole-5-carboxamide
N-[4-(pyrrolidin-1-yl)butyl]-N'-(2,4,6-trimethylphenyl)butanediamide
ethyl 4-{6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-amido}piperidine-1-carboxylate
2-(6-methoxynaphthalen-2-yl)-4-{2-methylthieno[2,3-d]pyrimidin-4-yl}morpholine
2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-N-methyl-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}butanamide
N-[2-(3-ethylphenoxy)ethyl]-N,2-dimethyl-2,8-diazaspiro[4.5]decane-3-carboxamide
[(2S,4R,5R)-5-(4-chlorophenyl)-1-ethyl-2-methyl-4-{[(1-methylpiperidin-4-yl)amino]methyl}pyrrolidin-2-yl]methanol
1-[(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-hydroxypropan-1-one
N-[(2-methoxyphenyl)methyl]-3-methyl-N-(pyridin-3-ylmethyl)furan-2-carboxamide
2-methyl-4-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
3-methyl-6-[3-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]pyridazine
N-methyl-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)-N-(2-phenoxyethyl)acetamide
N-[(1R)-1-(4-methoxyphenyl)ethyl]-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
1-[9-cyclopentyl-1-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
(1R,4S)-2-[2-(6-methoxypyridin-3-yl)pyridine-3-carbonyl]-2-azabicyclo[2.2.1]heptane
ethyl 4-[(3-methoxyphenyl)methyl]-1-[1-(4-methylpyridin-2-yl)propan-2-yl]piperidine-4-carboxylate
1-(1-{3-benzyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}ethyl)-1H-1,2,4-triazole
4-(6-fluoroquinolin-8-yl)-5H,6H,7H-cyclopenta[d]pyrimidin-2-amine
methyl (2S,3R)-2-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-3-hydroxybutanoate
2-(4-methoxyphenoxymethyl)-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]-1,3-oxazole-4-carboxamide
N-{[4-(4-fluorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-2,3-dimethoxybenzamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N,2,2-trimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carboxamide
6-(4-fluorophenyl)-2-[2-(1,4-oxazepan-4-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one