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3-({2-[1-(2,5-dimethylbenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
methyl(2-phenylethyl)[(3-{1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-1,2-oxazol-5-yl)methyl]amine
(2S,4R)-N-ethyl-4-[(2E)-3-phenylprop-2-enamido]-1-(pyridin-4-ylmethyl)pyrrolidine-2-carboxamide
2-(2-aminopyrimidin-5-yl)-7,8-dimethyl-N-[1-(pyrimidin-4-yl)ethyl]quinoline-4-carboxamide
(1S,5R)-6-methyl-3-[2-(pyridin-4-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[1-(3-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-6-(pyridin-4-yl)-1,2-dihydropyridin-2-one
N-[2-(cyclohex-1-en-1-yl)ethyl]-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
5-[(4-{4-cyclopropyl-5-[(dimethylamino)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]-N-ethylpyrimidin-2-amine
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-{[3-(2-methoxyphenyl)-1,2-oxazol-5-yl]methyl}acetamide
N-{[5-methyl-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
4-(4-chloro-2-methoxybenzoyl)-2-(4-chlorophenyl)morpholine
1-cyclohexyl-4-[1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperazin-2-one
3-[2-(dimethylamino)ethyl]-5-(3-methylbutyl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
ethyl 4-(2-methoxyethyl)-1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidine-4-carboxylate
ethyl 4-(4-phenyl-1H-imidazol-5-yl)-1H-pyrazole-3-carboxylate
N-[4-(furan-2-yl)phenyl]-1-[(4-oxo-4H-chromen-3-yl)methyl]piperidine-3-carboxamide
3-[4-(cyclobutylmethyl)piperazine-1-carbonyl]-1-phenylpyrrolidin-2-one
N-methyl-N-(quinolin-5-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[2-(2-ethylphenoxy)ethyl]-N-methyl-3-(1H-1,2,4-triazol-1-yl)propanamide
2-(4-acetyl-4-phenylpiperidin-1-yl)-1-(azepan-1-yl)ethan-1-one
N-ethyl-N-[(3-methoxyphenyl)methyl]quinoxaline-5-carboxamide
3-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-9-methoxy-N-[(4-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-(furan-2-ylmethyl)piperidine-3-carboxamide
4-{3-[3-(4-fluorophenyl)oxolan-3-yl]-1,2,4-oxadiazol-5-yl}-6-(propan-2-yl)pyrimidin-2-amine
1-ethyl-4-[({[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)methyl]pyrrolidin-2-one
N-{2-methyl-3-[(1,3-thiazol-2-yl)carbamoyl]phenyl}-5-(2-methylpropyl)-1,2-oxazole-3-carboxamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
4-[2-(3-phenyl-1,2-oxazol-5-yl)-1H-imidazol-1-yl]benzene-1-sulfonamide
1-(2-{1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl](methyl)[1-(pyrimidin-4-yl)ethyl]amine
2-{3-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]phenoxy}acetamide
4-benzyl-3-ethyl-1-(1H-indole-2-carbonyl)-1,4-diazepan-5-one
[(3S,4S)-1-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]-4-(hydroxymethyl)pyrrolidin-3-yl]methanol
3-(4-fluorophenoxymethyl)-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine
5-(2-{2-[4-(methylsulfanyl)phenyl]-1H-imidazol-1-yl}ethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-[2-(8-chloro-2-ethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-oxoethyl]-6-methoxy-2,3-dihydro-1H-indol-2-one
(2-ethoxy-5-{1-phenyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenyl)methanol
3-{[(2R)-2-(hydroxymethyl)pyrrolidin-1-yl]sulfonyl}-N-(2,2,2-trifluoroethyl)benzamide
[(1-cyclopentylpiperidin-3-yl)methyl][(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl][2-(piperidin-1-yl)ethyl]amine
[(3R,4R)-1-[(3-chloro-4-methoxyphenyl)methyl]-4-{[ethyl(methyl)amino]methyl}pyrrolidin-3-yl]methanol
N-[(4-hydroxy-3,5-dimethylpyridin-2-yl)methyl]-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
1-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-3-(2-methoxyphenoxy)azetidine
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-chloro-N-cyclopentyl-1-methyl-1H-pyrazole-3-carboxamide
methyl (2S,4S)-4-(3,5-dimethoxybenzamido)-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxylate
3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]propan-1-one
6-(3-acetylphenyl)-5-cyano-2-methylpyridine-3-carboxylic acid
N3-tert-butyl-1-cyclohexyl-N5-[2-methyl-2-(morpholin-4-yl)propyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-(4-{1-[methyl(pyridin-4-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)propan-1-one