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N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
phenyl({1-[1-(1,3-thiazol-2-ylmethyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl})methanol
1,3-dimethyl-N-[1-(4-methylpyridin-2-yl)propyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-[(1S,3R)-1-(2-aminoethoxy)-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-2-(2,3-difluorophenyl)ethan-1-one
(2-methylpropyl)[(3-methylthiophen-2-yl)methyl](pyridin-3-ylmethyl)amine
2,6-difluoro-N-{1-[1-(2-hydroxyethyl)-1,2,5,6-tetrahydropyridin-3-yl]propyl}benzamide
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetamide
3-{[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]methyl}-1H-indole
7-chloro-3,5-dimethyl-N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]-1-benzofuran-2-carboxamide
2-[(2-{1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidin-4-yl}-1H-imidazol-1-yl)methyl]pyridine
N-(5-{1H-pyrazolo[3,4-b]pyridin-1-yl}quinolin-8-yl)acetamide
1-(4-chloro-3-methylphenoxy)-3-[(thian-4-yl)amino]propan-2-ol
methyl (2S,4S)-1-[(2-chlorophenyl)methyl]-4-[4-(1H-pyrazol-1-yl)benzamido]pyrrolidine-2-carboxylate
N-[1-(butan-2-yl)-1H-pyrazol-5-yl]-3-(5-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)propanamide
1-(3-{[3-(morpholin-4-yl)piperidin-1-yl]methyl}phenyl)ethan-1-one
1-[(3-fluorophenyl)methyl]-5-(2-{[(3-methoxyphenyl)methyl]amino}ethyl)pyrrolidin-2-one
7-chloro-2-methyl-4-(quinolin-6-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3,5-dimethyl-4-oxo-N-{1-[2-(trifluoromethyl)phenyl]ethyl}-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
N-{2-[4-(dimethylamino)phenyl]ethyl}-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
N,6-dimethyl-2-(4-methylphenoxymethyl)-1-[2-(morpholin-4-yl)ethyl]-4-oxo-N-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
(3S)-3-{[1,3-dimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}azepan-2-one
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-(1H-pyrazol-3-ylmethyl)acetamide
N-tert-butyl-3-(4-methyl-1,4-diazepane-1-carbonyl)-5-[(thiophen-2-ylmethyl)amino]benzene-1-sulfonamide
4-{6-[(piperidin-4-yl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phthalazin-1-ol
7-fluoro-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
(3S)-4-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-1,3-dimethylpiperazin-2-one
4-(piperidin-3-yl)-N-(pyridin-2-ylmethyl)benzamide
N-(1,3-benzothiazol-5-yl)-1H-indazole-3-carboxamide
4-[3-(azepane-1-carbonyl)-1-ethyl-4,5,6,7-tetrahydro-1H-indazol-5-yl]-7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepine
7-[(3-methylthiophen-2-yl)methyl]-3-(oxolan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
4-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepane-1-carbonyl}-2-methylphenol
1-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-4-(1,3-thiazol-2-yl)-1H-1,2,3-triazole
N-cyclopropyl-3,5-dimethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]adamantane-1-carboxamide
2-(cyclohex-1-en-1-ylmethyl)-6-(1-methylpiperidin-4-yl)-3,4-dihydropyrimidin-4-one
3-[({[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}amino)methyl]pyrrolidin-3-ol
6-(2-chlorophenyl)-N-(dicyclopropylmethyl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-propyl-1,3-thiazole-4-carboxamide
N-{[2-(4-acetylpiperazin-1-yl)-7-methylquinolin-3-yl]methyl}-N-cyclopropyl-2H-1,3-benzodioxole-5-carboxamide
2-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-5-ethyl-1H-pyrrole
1-[5-(2-chlorophenyl)furan-2-carbonyl]-2-(1-methyl-1H-pyrazol-3-yl)piperidine
3,5-dimethyl-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1,2-oxazole-4-carboxamide
7-cyclohexyl-2-(4-methoxybenzoyl)-2,7-diazaspiro[4.5]decan-6-one
N-methyl-N-[(1-methylpyrrolidin-2-yl)methyl]-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-(3-fluorophenyl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
N-methyl-2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-[(4-phenoxyphenyl)methyl]acetamide
1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-4-(5-methylpyridin-2-yl)piperidin-4-ol
2-[3-(2-phenyl-1H-imidazol-1-yl)phenoxy]propanamide
N-cyclopropyl-N-[(2-ethoxyphenyl)methyl]-2-ethylpyrimidine-5-carboxamide
{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
7-(2-cyclohexylethyl)-2-[3-(methylsulfanyl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one