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2-{4-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1H-1,2,3-triazol-1-yl}-1-(pyrrolidin-1-yl)ethan-1-one
2-(2-hydroxyphenoxy)-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}acetamide
N-cyclohexyl-2-cyclopropyl-4-hydroxy-N-(thiophen-3-ylmethyl)pyrimidine-5-carboxamide
N-(furan-2-ylmethyl)-N-(2-hydroxyethyl)-2-(2-methyl-1H-imidazol-1-yl)propanamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-{1-[3-(1H-pyrazol-4-yl)propanoyl]piperidin-4-yl}propanamide
3-[2-(3,4-difluorophenyl)ethyl]-1-(3-propyl-1H-pyrazole-4-carbonyl)piperidine
(2,1,3-benzoxadiazol-5-ylmethyl)({[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl})amine
{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(2-methoxyethyl)(propan-2-yl)amine
1-[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-[4-(3-methylphenyl)piperazin-1-yl]propan-1-one
1-cyclohexyl-4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
3-[6-hydroxy-4-(3-methoxypropanoyl)-1,4-diazepan-1-yl]pyrazine-2-carbonitrile
2-[(2S,6S)-6-(hydroxymethyl)-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]-1-(piperazin-1-yl)ethan-1-one
[(3R,4R)-1-(dimethyl-1,3-thiazole-5-carbonyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
methyl 2-[({1-[(2-fluorophenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)amino]acetate
N-(2-{[(2-methoxy-6-methylphenyl)carbamoyl]amino}ethyl)-2-methylpropanamide
5-methanesulfonyl-1'-(1,3-thiazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-(1,5-dimethyl-1H-pyrazol-4-yl)-1-methyl-1-[3-(1-methyl-1H-pyrazol-4-yl)propyl]urea
1-[3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-4-(thiophen-2-yl)butan-1-one
2-[(4aR,7aS)-4-[(2-aminopyridin-3-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
5-[(dimethylamino)methyl]-N-{2-methyl-1,1-dioxo-2H,3H,4H-1λ6-thieno[2,3-e][1,2]thiazin-4-yl}furan-2-carboxamide
5-(2-chloro-4-fluorophenyl)-3-(ethoxymethyl)-1-methyl-1H-1,2,4-triazole
2-({2-[2-methyl-1-(morpholin-4-yl)propan-2-yl]-1H-imidazol-1-yl}methyl)-3,4-dihydroquinazolin-4-one
3-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-(quinolin-6-ylmethyl)propanamide
N-[(1-ethyl-1H-indazol-3-yl)methyl]-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
1-(pyridine-4-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
(3S,4S)-1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(morpholin-4-yl)pyrrolidin-3-ol
1-{1-[(2-ethoxyphenyl)methyl]piperidin-3-yl}-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
2-(2,5-dimethoxyphenyl)-1-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
N-[3-(3-methylphenyl)phenyl]-1-[2-(methylsulfanyl)acetyl]piperidine-3-carboxamide
ethyl 4-{1-[3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanoyl]piperidin-3-yl}piperazine-1-carboxylate
(3R,4S)-1-methanesulfonyl-N,N-dimethyl-4-(5-methylfuran-2-yl)pyrrolidin-3-amine
1-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
3-[2-(dimethylsulfamoyl)ethyl]-1-[4-(furan-2-ylmethoxy)phenyl]urea
N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidin-4-ol
2-(4-methylphenyl)-4-[3-(1H-pyrazol-1-yl)azetidine-1-carbonyl]quinoline
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{2-[(dimethylamino)methyl]-1,3-thiazole-4-carbonyl}piperidin-3-ol
N-[1-({[3-(1H-1,2,3-benzotriazol-1-yl)propyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-3-phenoxypropanamide
1-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-2,2-dimethylpropan-1-one
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-6-phenylpyridazin-3-amine
4-[8-methyl-3-(thiomorpholin-4-ylmethyl)imidazo[1,2-a]pyridine-2-carbonyl]morpholine
2-chloro-N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)pyridine-4-carboxamide
3-(3-chloro-1H-1,2,4-triazol-5-yl)-1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
2-(2-methyl-1,3-thiazol-4-yl)-1-{1'-methyl-3,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
N-{[1-(thiophene-3-carbonyl)piperidin-3-yl]methyl}-1H-indazole-3-carboxamide
N-[1-(cyclohexylmethyl)piperidin-3-yl]-3-(pyridin-4-yl)propanamide
2-methoxy-1-(4-{4-[4-(pyridin-2-yl)piperazine-1-carbonyl]phenoxy}piperidin-1-yl)ethan-1-one
ethyl 4-[(2-chlorophenyl)methyl]-1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidine-4-carboxylate
{[3-(3-fluorophenyl)oxolan-3-yl]methyl}({[4-(methylsulfanyl)phenyl]methyl})amine
N-[(1R,3R)-3-aminocyclopentyl]-6-(2-hydroxyethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide