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5-fluoro-N,1,3-trimethyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-1H-indole-2-carboxamide
5-[2-(4-methylpentyl)morpholine-4-carbonyl]pyridin-2-ol
2-[2-({4-[2-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
N-({1-[(2-fluorophenyl)methyl]pyrrolidin-3-yl}methyl)-6-oxo-1,6-dihydropyridine-2-carboxamide
5-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidine-1-carbonyl}-2,3-dihydro-1H-pyrazol-3-one
N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)-1,1-dioxo-1λ6-thiane-4-carboxamide
1-(2-methylpropyl)-N-[2-(methylsulfanyl)ethyl]-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(3S,4S)-4-(3-methoxyphenyl)-1-[(2-methoxypyridin-3-yl)methyl]piperidin-3-ol
1-[(4,5-dimethylfuran-2-yl)methyl]-4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine
1-{[1-(4-butylphenyl)-1H-pyrazol-4-yl]methyl}-4-(hydroxymethyl)azepan-4-ol
N-(1-benzylpyrrolidin-3-yl)-3-[1-(2-methoxyacetyl)piperidin-4-yl]propanamide
1-(2-methoxyethyl)-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
N-[(3S,4R)-1-[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
N-ethyl-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-1-(methoxymethyl)cyclobutane-1-carboxamide
1-ethyl-N-(2-methoxyethyl)-7-methyl-4-oxo-N-(thiophen-2-ylmethyl)-1,4-dihydro-1,8-naphthyridine-3-carboxamide
2-cyclopropyl-9-(2,3,4-trifluorobenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(4,8-dimethoxynaphthalen-1-yl)methyl]azetidine-3-carboxylic acid
1-(4-{[2-(hydroxymethyl)phenyl]methyl}piperazin-1-yl)-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]ethan-1-one
(4aS,8aS)-2-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)-7-(propan-2-yl)-decahydro-2,7-naphthyridin-4a-ol
10-methoxy-5-(5-methoxy-1H-indole-2-carbonyl)-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
(5S,9aS,9bS)-2-(pyridin-3-ylmethyl)-5-[3-(trifluoromethyl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[4-(3-methylphenyl)phenyl]-1-(1,2-oxazol-3-ylmethyl)piperidine-4-carboxamide
N-[(1-{6-methylimidazo[2,1-b][1,3]thiazole-3-carbonyl}piperidin-3-yl)methyl]-1-phenylmethanesulfonamide
4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]-1-[(4-methoxyphenyl)methyl]piperazin-2-one
3-{[(6,8-dimethyl-4-oxo-1,4-dihydroquinolin-2-yl)methyl](ethyl)amino}-1λ6-thiolane-1,1-dione
N-(cyclohexylmethyl)-5-(2,6-dimethylphenoxymethyl)-1,2-oxazole-3-carboxamide
1-[5-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]-3-phenylpropan-2-ol
ethyl 4-(2-{4-[3-(hydroxymethyl)piperidin-1-yl]piperidin-1-yl}-6-(2-methoxyphenyl)pyridine-3-carbonyl)piperazine-1-carboxylate
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-(pyrazin-2-yl)piperazin-2-yl}ethan-1-ol
1-[1-oxo-1-(piperidin-1-yl)propan-2-yl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-(5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)-4-(propan-2-yl)piperazine
N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
N,6-dimethyl-2-oxo-N-(quinoxalin-2-ylmethyl)-1,2-dihydropyridine-4-carboxamide
1-{1-[1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-ol
3-[4-(3-methylpiperidine-1-carbonyl)phenyl]-1-(2-phenoxyethyl)urea
1-(1H-indole-6-carbonyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
methyl 4-({3-[ethyl(pyridin-4-ylmethyl)amino]piperidin-1-yl}methyl)benzoate
1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide
4-[(1-{1-[(4,5-dimethylfuran-2-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methyl]piperazin-2-one
N-[(5-{[(4-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]-9-methyl-9H-carbazole-3-carboxamide
1-{3-[3-({[2-(dimethyl-1,3-thiazol-2-yl)ethyl]amino}methyl)phenoxy]-2-hydroxypropyl}piperidin-4-ol
2-[3-(2-methoxyethyl)-5-(2-phenylphenyl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
methyl 8-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
1-(4-{[(3-phenylpropyl)amino]methyl}phenoxy)-3-(piperidin-1-yl)propan-2-ol
5-ethyl-5-{1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidin-4-yl}-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]imidazolidine-2,4-dione
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[(2-ethylphenyl)methyl]pyrrolidin-3-yl]-1H-imidazole-2-carboxamide
N-(2-{[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]methyl}propyl)-2-(methylamino)pyrimidine-5-carboxamide
5-({4-oxo-3H,4H-pyrido[4,3-d]pyrimidin-3-yl}methyl)pyrrolidin-2-one
6-methyl-3-[(4-phenylpiperazin-1-yl)methyl]-1-(prop-2-en-1-yl)-1,2-dihydroquinolin-2-one
1-(4-cyclopentylpyrimidin-2-yl)-4-(5-methylpyridin-2-yl)piperidin-4-ol