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2-[3-benzyl-1-(4-methoxyphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(2-methylprop-2-en-1-yl)acetamide
6-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-N,N-dimethylpyrazin-2-amine
(1R,7S)-3-(3,4-dimethylphenyl)-6-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-phenoxypropanamide
[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]({[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-2-(thiophen-3-yl)acetamide
N-(5-{3-[methyl(2-phenylethyl)amino]piperidine-1-carbonyl}-1,3-thiazol-2-yl)acetamide
3-{2-[(3,5-dimethyl-1H-indol-2-yl)formamido]acetamido}propanoic acid
N-{[4-(dimethylamino)oxan-4-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-[(4-{[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]amino}piperidin-1-yl)methyl]phenol
6-[(3-fluorophenyl)methyl]-2-{3-[(3-oxopiperazin-1-yl)methyl]phenyl}-3,4-dihydropyrimidin-4-one
2-[3-(methoxymethyl)pyrrolidin-1-yl]-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridine
N-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-2,2-dimethylcyclopropane-1-carboxamide
1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
N-(1-{7-[(2E)-3-(2,4-difluorophenyl)prop-2-enoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)propanamide
5-(2,6-dimethoxyphenyl)-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-1,2,4-triazin-3-amine
(3aR,5R,6S,7aS)-2-[(8-methoxyquinolin-2-yl)methyl]-octahydro-1H-isoindole-5,6-diol
5-[(3S,4S)-3-carboxy-4-propylpyrrolidine-1-carbonyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxylic acid
1-[(3,4-difluorophenyl)methyl]-3-(5-fluoro-2-methoxybenzoyl)piperidine
(1R,5S,8S)-8-methoxy-N-{3-[(E)-2-(pyridin-2-yl)ethenyl]phenyl}-3-azabicyclo[3.2.1]octane-3-carboxamide
N-[2-methyl-3-(pyrrolidin-1-yl)phenyl]-4-(2-oxo-1,3-oxazolidin-3-yl)piperidine-1-carboxamide
1-(3-chlorophenyl)-4-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]piperazin-2-one
5-(2-chloro-4-methoxyphenoxymethyl)-N,N-dimethyl-1H-pyrazole-3-carboxamide
4-[1-(1-cyclohexylpiperidin-4-yl)piperidine-3-carbonyl]morpholine
N-(1,3-benzothiazol-2-ylmethyl)-2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-methylacetamide
2-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-9-oxa-2-azaspiro[5.5]undecane
N-(1,4-dioxan-2-ylmethyl)-N-methyl-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
N-[2-(2-chlorophenyl)-1-[1-(quinolin-5-ylmethyl)piperidin-4-yl]ethyl]-N-methylfuran-2-carboxamide
7-(azepane-1-sulfonyl)-2-(dimethylamino)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-(5-acetylthiophen-3-yl)-N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
3-(2-chlorophenyl)-1-methyl-3-[2-oxo-2-(3-oxo-4-phenylpiperazin-1-yl)ethyl]pyrrolidine-2,5-dione
1-(propan-2-yl)-4-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]piperidine
{1-[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidin-3-yl}methanol
2-(1,3-thiazol-2-yl)-1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperidine
1-cyclohexyl-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)piperidine-4-carboxamide
4-{[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]methyl}-N-methylbenzamide
4-ethyl-5-[3-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine-1-carbonyl]-1,3-thiazol-2-amine
3-(4-chlorophenyl)-1-[4-(2-hydroxyethyl)piperidin-1-yl]-3-phenylpropan-1-one
7-methyl-2-(2-{methyl[(4-methylphenyl)methyl]amino}acetyl)-2,7-diazaspiro[4.5]decan-6-one
N-(2-{[(2-fluorophenyl)methyl]sulfanyl}phenyl)-1-(methoxymethyl)cyclobutane-1-carboxamide
1-methyl-9-[2-(1H-pyrazol-1-yl)benzoyl]-1,4,9-triazaspiro[5.5]undecan-5-one
4-benzyl-1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(4-fluorobenzoyl)piperidine
7-[1-(2H-1,3-benzodioxol-5-yl)-3-methyl-1H-1,2,4-triazol-5-yl]-3-methyl-3,4-dihydroquinazolin-4-one
N-[(1-phenylcyclopentyl)methyl]-6-(quinolin-8-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
(3aR,7aS)-2-[4-(pyridin-2-yl)pyrimidin-2-yl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
1-{6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carbonyl}-2-methyl-1,4-diazepan-5-one
2-[3-(4-methylpiperidine-1-carbonyl)phenyl]-2-(thiomorpholin-4-yl)acetic acid
3-chloro-4-fluoro-N-[3-(1H-1,2,3-triazol-1-yl)propyl]-1-benzothiophene-2-carboxamide
(5S,9aS,9bS)-5-(2,4-dimethoxyphenyl)-2-[(3-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one