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6-{4-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperazin-1-yl}pyridine-3-carbonitrile
(1H-indol-4-ylmethyl)(methyl){[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}amine
1-{2-[(5-chloropyridin-2-yl)oxy]hex-5-en-1-yl}piperidine-4-carboxylic acid
N-[2-(cyclohex-1-en-1-yl)ethyl]-4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide
1,4,6-trimethyl-2-oxo-N-{[5-(pyridin-2-yl)thiophen-2-yl]methyl}-1,2-dihydropyridine-3-carboxamide
3-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-1-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)urea
methyl 3-(1,4-dioxan-2-ylmethyl)-1-[(4-fluorophenyl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylate
N-cyclopropyl-N-({4-[3-(1,3-dioxo-2,3-dihydro-1H-isoindol-2-yl)propoxy]phenyl}methyl)-2H-1,3-benzodioxole-5-carboxamide
4-(prop-2-en-1-yl)-1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-1,4-diazepan-5-one
2-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-4-(pyridin-3-ylmethyl)piperazine
2-[4-(2-phenoxyethyl)piperazin-1-yl]pyrazine
5-{1-[(2-chloro-6-fluorophenyl)methyl]-4-hydroxypiperidin-4-yl}-N-(oxolan-2-ylmethyl)-1-benzofuran-2-carboxamide
N-(1H-1,3-benzodiazol-5-yl)-2-{4-[(6-methylpyridin-2-yl)methyl]morpholin-3-yl}acetamide
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(5-methylthiophen-2-yl)methyl]piperidine
N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-4-(morpholin-4-yl)benzamide
(3S,4S)-4-(pyridin-2-yl)-1-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}pyrrolidine-3-carboxylic acid
6-(4-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperazin-1-yl)pyridine-3-carboxamide
2-[1-methyl-4-(2-methyl-1,3-thiazole-4-carbonyl)-10-oxo-1,4,9-triazaspiro[5.6]dodecan-9-yl]acetic acid
N-{[5,8-dimethoxy-2-(4-methylphenyl)quinolin-3-yl]methyl}-N-[2-(dimethylamino)ethyl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-2-(methylamino)pyrimidine-5-carboxamide
2-{[(5-fluoro-2-methoxyphenyl)formamido]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
N-(5-tert-butyl-2-methoxyphenyl)thiomorpholine-4-carboxamide
2-(3-fluorophenyl)-N-[(7-{[3-(trifluoromethyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]acetamide
2-[(3-fluorophenyl)methyl]-N-(1-methoxypropan-2-yl)-6-methyl-1-[3-(morpholin-4-yl)propyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
2-(5-{[3-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}furan-2-yl)benzonitrile
N-(5-tert-butyl-2-methoxyphenyl)-2-(2-hydroxyethyl)-3-oxopiperazine-1-carboxamide
(3S)-4-{1-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-3-methyl-1-(2-methylpropyl)piperazin-2-one
N3-cyclooctyl-N5-(2,2-dimethyloxan-4-yl)-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
1-ethyl-N-(2-{2-methyl-1-azatricyclo[6.3.1.04,12]dodeca-2,4,6,8(12)-tetraen-3-yl}ethyl)-5-oxopyrrolidine-3-carboxamide
1-ethyl-6,7,8-trifluoro-3-(1-methyl-1H-1,2,4-triazol-5-yl)-1,4-dihydroquinolin-4-one
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
6-[(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)methyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
2,6-difluoro-3-methyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]benzamide
1-ethyl-N-{[1-(3-methylbut-2-en-1-yl)piperidin-4-yl]methyl}-1H-pyrazole-5-carboxamide
1-[4-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)phenyl]-1H-imidazole
5-[4-(aminomethyl)piperidin-1-yl]-2-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-2,3-dihydropyridazin-3-one
1-(2-{[methyl(1H-pyrazol-5-ylmethyl)amino]methyl}phenoxy)-3-(thiomorpholin-4-yl)propan-2-ol
6-{methyl[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(15),3(8),6,11,13-pentaen-4-one
6-({[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}amino)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
methyl 4-(5-chloro-2-{[(1,3-dimethyl-1H-pyrazol-5-yl)formamido]methyl}-2,3-dihydro-1-benzofuran-7-yl)benzoate
N-(2-fluorophenyl)-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
1-[(3-methoxyphenyl)methyl]-6-oxo-N-[2-(1H-pyrazol-4-yl)ethyl]piperidine-3-carboxamide
1-(2-methylpyridin-4-yl)-4-(trimethylpyrimidin-4-yl)-1,4-diazepane
3-(4-chloro-1H-pyrazol-1-yl)-1-{4-[(3-fluorophenyl)methyl]-1,4-diazepan-1-yl}propan-1-one
4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]methyl}-2,1,3-benzoxadiazole
2-(2-{1-[4-(1H-imidazol-1-yl)benzoyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
N'-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N,N-dimethylbutanediamide
1-{[(1,3-dimethyl-1H-pyrazol-4-yl)carbamoyl]methyl}-1,4-diazepane-6-carboxylic acid
(1s,4s)-4-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}cyclohexan-1-ol