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2-(4-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}morpholin-2-yl)ethan-1-amine
ethyl 4-(3-phenylpropyl)-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]piperidine-4-carboxylate
ethyl 1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-3-[(4-fluorophenyl)methyl]piperidine-3-carboxylate
1-methyl-5-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-({4-[(2-chloroprop-2-en-1-yl)oxy]phenyl}methyl)-4-(4-fluorophenyl)-N-(pyridin-3-ylmethyl)benzamide
N-methyl-5-{[4-(trifluoromethoxy)phenyl]methyl}-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(1R,3S)-3-{[2-(dimethylamino)ethyl][(5-methylthiophen-2-yl)methyl]carbamoyl}cyclopentane-1-carboxylic acid
2-[3-(dimethylamino)propyl]-9-[(2S)-2-hydroxy-3-phenylpropanoyl]-2,9-diazaspiro[5.5]undecan-3-one
3-{5-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
3-fluoro-4-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
(2S)-4-methyl-2-{2-[2,6,6-trimethyl-4-oxo-1-(propan-2-yl)-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamido}pentanamide
N4-({4-[(dimethylamino)methyl]phenyl}methyl)-5-ethyl-6-methylpyrimidine-2,4-diamine
N-[1-(methylcarbamoyl)cyclohexyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-(4-phenylazepan-1-yl)ethan-1-one
4-[3-(2H-1,3-benzodioxol-5-yl)-3-phenylpropanoyl]-3,3-dimethylpiperazin-2-one
2-(2-aminoethyl)-5,6-dimethyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}thieno[2,3-d]pyrimidin-4-amine
N-({1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]pyrrolidin-3-yl}methyl)cyclohexanecarboxamide
2-{2-[2-(cyclopropylcarbamoyl)ethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}-1,3-thiazole-4-carboxamide
5-{1-[(2-phenyl-2H-1,2,3-triazol-4-yl)methyl]-1H-imidazol-2-yl}-2-(pyridin-2-yl)pyrimidine
1-{[(3R,4R)-4-(hydroxymethyl)-1-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}pyrrolidin-3-yl]methyl}piperidin-4-ol
3-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-5-(3-methoxyphenoxymethyl)-1,2-oxazole
N-[(1-cyclopropanecarbonylpiperidin-3-yl)methyl]-6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
{2-[5-(2,4-dimethylphenyl)-1,2,4-oxadiazol-3-yl]ethyl}dimethylamine
1-(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)azocane
{[2-(2-methoxyphenyl)pyrimidin-5-yl]methyl}(methyl)[(3-methylpyridin-4-yl)methyl]amine
(4aS,8aR)-6-(1H-imidazole-2-carbonyl)-1-(2-phenylethyl)-decahydro-1,6-naphthyridin-2-one
1-[5-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine-1-carbonyl)thiophen-2-yl]ethan-1-one
4-{[(4-hydroxy-5,8-dimethylquinolin-2-yl)methyl](methyl)amino}-1λ6-thiane-1,1-dione
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(methylsulfanyl)pyridine-3-carboxamide
ethyl 5-(2,6-dimethylpyrimidine-4-carbonyl)-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-{1-[1-(1-benzothiophen-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopentanecarboxamide
(3R,5S)-1-[(3,4-dimethoxyphenyl)methyl]-5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-[2-(morpholin-4-yl)ethyl]piperidine-3-carboxamide
(3S,9aR)-3-[(benzyloxy)methyl]-8-(naphthalene-1-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(4-methoxyphenyl)-N-({1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]piperidin-3-yl}methyl)acetamide
N-(2-{7-[(3,5-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclohexanecarboxamide
N-methyl-4-{[(3R)-pyrrolidin-3-yl]sulfamoyl}-N-(1,3-thiazol-2-ylmethyl)benzamide
3-[5-(1-carbamoylethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-N-cyclopropylpropanamide
N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
3-[(3R,4S)-1-(2-methoxy-4-methylbenzoyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(methylamino)pyrimidine-5-carboxamide
(1S,5R)-3-cyclobutanecarbonyl-6-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]-2-(2-cyclopropyl-1H-1,3-benzodiazol-1-yl)ethan-1-one
6-methyl-5-[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]-2-(1,2-oxazole-3-carbonyl)-1,2,3,4-tetrahydro-2,7-naphthyridine
1-[4-(6-hydroxypyrimidin-4-yl)piperidin-1-yl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
1-(2-phenylethyl)-3-(pyrimidin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[(2,3-dimethoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(1,3-benzothiazol-6-yl)-4-(6-ethylpyrimidin-4-yl)piperazine-1-carboxamide
9-(6-chloro-2H-chromen-3-yl)-1H,2H,3H,6H,7H,8H,9H-[1,4]oxazino[3,2-g]quinoline-2,7-dione
1-{4-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]phenyl}imidazolidine-2,4-dione
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-hydroxypiperidin-1-yl)methyl]pyrrolidin-1-yl]-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]ethan-1-one