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N-(1-hydroxy-2-methylpropan-2-yl)-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide
ethyl 4-(2-{[2-(ethoxycarbonyl)piperidin-1-yl]methyl}-8-methylquinazolin-4-yl)piperazine-1-carboxylate
3-(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)-1-ethyl-1-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]urea
4-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-2-{[3-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindole-1,3-dione
2-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]imidazo[1,2-a]pyrimidine-3-carboxamide
4-(4-methylphthalazin-1-yl)benzamide
3-[4-({2-methyl-2,8-diazaspiro[4.5]decan-8-yl}methyl)-1H-pyrazol-1-yl]propanoic acid
N,N-dimethyl-6-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}pyrazin-2-amine
N-methyl-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
4-{1-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-1H-imidazol-2-yl}-2,1,3-benzoxadiazole
N-[(1-ethylpyrrolidin-2-yl)methyl]-1-[4-(furan-2-yl)pyrimidin-2-yl]-5-(propan-2-yl)-1H-pyrazole-4-carboxamide
3-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methoxy}pyridin-2-amine
1-[7-(1-benzothiophen-3-yl)-9-ethoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(thiophen-3-yl)ethan-1-one
ethyl 4-[(3R,4R)-3-hydroxy-4-(pyridine-3-amido)piperidin-1-yl]piperidine-1-carboxylate
2-ethyl-8-{2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]acetyl}-2,8-diazaspiro[4.5]decan-3-one
3-ethyl-8-[3-(morpholin-4-yl)benzoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-4-(2-propyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-1,3-oxazole
2-(morpholin-4-yl)-8-[4-(prop-2-en-1-yloxy)phenyl]-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
1-[1-ethyl-3-(4-phenylpiperazine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(thiophen-2-yl)ethan-1-one
1-{1-[(2-chlorophenyl)methyl]piperidin-4-yl}-3-(1-ethyl-1H-1,2,4-triazol-3-yl)urea
2-[4-(5-methyl-1,3,4-oxadiazol-2-yl)piperazin-1-yl]-1-(morpholin-4-yl)ethan-1-one
N-cyclopentyl-3-{5-[(3E)-pent-3-enoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
N-(5-methyl-2,1,3-benzothiadiazol-4-yl)-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
(1S,6R)-9-[3-(pyrazin-2-yl)propanoyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[1-(thiophen-2-yl)ethyl]benzamide
6-(3-chloro-4-fluorobenzoyl)-1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-azaspiro[2.5]octane
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-1,2,5-thiadiazole-3-carboxamide
2-[4-(4-fluorophenyl)-2-[(4-methylpiperazin-1-yl)methyl]phenoxy]-N-(2-methoxy-2-methylpropyl)acetamide
4-{2-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]pyridine-4-carbonyl}morpholine
1-[1-(5-phenoxyfuran-2-carbonyl)piperidin-4-yl]-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
N-{[3-methyl-7-(oxolane-2-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(phenylsulfanyl)acetamide
methyl 2-[(cyclohexylmethyl)sulfamoyl]-6-[3-(methylsulfanyl)propanoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N-(propan-2-yl)pyridine-4-carboxamide
2-[4-(2H-1,3-benzodioxol-4-ylmethyl)-1-[(2-fluoro-4-methoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
3-[2-(4-methyl-1,3-thiazol-2-yl)ethyl]-1-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}urea
7-cyclohexyl-2-(pyridin-4-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
(2S,4S)-4-amino-N-methyl-1-[4-(thiophen-2-yl)butanoyl]pyrrolidine-2-carboxamide
N-(1-{1-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-4-yl}-2-(3-methoxyphenyl)ethyl)-N,1-dimethyl-1H-pyrazole-3-carboxamide
5-[methyl(2-phenylethyl)amino]-2-[2-(1,4-oxazepan-4-yl)-2-oxoethyl]-2,3-dihydropyridazin-3-one
3-(4-methoxy-3,5-dimethylbenzoyl)-1-(5-methyl-1,2-oxazole-3-carbonyl)piperidine
5-ethyl-4-methyl-6-{3-[(4-methylpiperazin-1-yl)methyl]piperidin-1-yl}pyrimidin-2-amine
(4aR,7aS)-1-cyclobutanecarbonyl-4-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[2-(4-chlorophenyl)ethyl]-N-methyl-6-oxo-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
1-(1-methylpiperidine-4-carbonyl)-3,3-diphenylpiperidine
N-(2-{[(3-{3-[benzyl(methyl)amino]-2-hydroxypropoxy}-4-methoxyphenyl)methyl]amino}ethyl)acetamide
N-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
4-methoxy-2-({3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)phenol
1-[2-(4-fluorophenyl)piperidin-1-yl]-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
N-[2-(4-methoxyphenyl)ethyl]-N-[(1-methylpiperidin-4-yl)methyl]-5-[(methylsulfanyl)methyl]furan-2-carboxamide
1-[3-({methyl[1-(pyridin-3-yl)ethyl]amino}methyl)phenyl]ethan-1-one