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N-cyclopentyl-9-(cyclopropylmethyl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
N-[2-methyl-5-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-4-(oxan-4-yl)piperazine-1-carboxamide
N-[(5-carbamoyl-1,2,4-oxadiazol-3-yl)methyl]-4-hydroxy-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
(1S,5R)-N-(4-fluorophenyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
(3-{[1-(8-methoxy-4-methylquinolin-2-yl)pyrrolidin-3-yl]methyl}phenyl)methanol
N-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-amine
4-[3-fluoro-5-(2-methylpropoxy)phenyl]-6-(morpholin-4-yl)pyrimidin-2-amine
N-[1-(pyrimidin-2-yl)piperidin-3-yl]-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
2-[(1S,5R)-3-(3-methoxybenzoyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
N-ethyl-5-(1H-imidazol-2-ylmethyl)-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-(2,4-dimethoxyphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-[(3R,4S)-4-cyclopropyl-1-(2-methoxyacetyl)pyrrolidin-3-yl]-1,3-benzothiazole-6-carboxamide
3-(5-methylfuran-2-yl)-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]-1H-pyrazole-5-carboxamide
1-[5-({[(2-chlorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
4-[1-(4-fluorophenyl)-1H-pyrazol-4-yl]-N-[1-(pyridin-4-yl)propan-2-yl]pyrimidin-2-amine
3-({1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}oxy)pyridine
1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-4-carboxamide
(3S,4R)-1-[2-(2-hydroxyphenyl)acetyl]-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
3-(4-chloro-2-methoxy-5-methylphenyl)-1-{[4-(hydroxymethyl)oxan-4-yl]methyl}-1-methylurea
4-{3-[1-(dimethylamino)ethyl]phenyl}-6-methyl-2,3-dihydropyridazin-3-one
[(3R,4R)-4-[(dimethylamino)methyl]-1-[(4-phenoxyphenyl)methyl]pyrrolidin-3-yl]methanol
N-[(3,4-difluorophenyl)methyl]-3-(morpholine-4-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-{3-[2-(4-fluorophenoxy)ethyl]phenyl}-5-methyl-1,3,4-oxadiazole
(4aS,7aR)-1-(1H-imidazol-2-ylmethyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-chloro-N,N-diethyl-3-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)acetamido]benzamide
N-butyl-5-{4-[(ethylcarbamoyl)amino]-3-methoxyphenyl}furan-2-carboxamide
N-[1-({[2-hydroxy-3-(3-methoxyphenoxy)propyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-2-methylfuran-3-carboxamide
2-[({5-[1-(3-chloropyridin-2-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)(methyl)amino]ethan-1-ol
1-(4-{4-[(2,2-dimethylpyrrolidin-1-yl)methyl]-1H-1,2,3-triazol-1-yl}piperidin-1-yl)hexan-1-one
6-(2-chloro-4-fluorobenzoyl)-N-[3-(pyridin-4-yl)propyl]-6-azaspiro[2.5]octane-1-carboxamide
[(3aS,6aS)-2-(3,4,7-trimethyl-1H-indole-2-carbonyl)-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
2-methyl-1-(1-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}azetidin-3-yl)piperidine
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
2-{3-[4-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]piperidin-1-yl}acetamide
(2R,3R)-3-(dimethylamino)-1'-(5-nitropyridin-2-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-(4-hydroxyphenyl)-N-(thiophen-2-ylmethyl)-1H-pyrazole-5-carboxamide
(1S,6R)-9-[2-(4-methylphenoxymethyl)furan-3-carbonyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(pyrazin-2-yl)pyrrolidin-3-yl]methanol
N-cyclopentyl-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxamide
6-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-N-ethylpyridine-3-carboxamide
1-[(2-fluorophenyl)methyl]-4-(thiophen-3-ylmethyl)-1,4-diazepane
N-benzyl-1-[1-(3-methylfuran-2-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
6-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carboxylic acid
methyl 9-(cyclopentyloxy)-3-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-methyl-3-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1-(1-oxo-2,3-dihydro-1H-inden-5-yl)urea
3-(dimethyl-1H-1,2,4-triazol-1-yl)-N,2-dimethyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}propanamide
(2R,4R)-N-[1-(4-chlorophenyl)cyclobutyl]-4-hydroxypyrrolidine-2-carboxamide
[(3R,4S)-1-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
4-[2-(3,4-dichlorophenyl)morpholin-4-yl]-6-methylpyrimidin-2-amine