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6-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3-oxo-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
2-methoxy-1-[9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
{4-[(2-chlorophenyl)methyl]-1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-4-yl}methanol
1-[3-(phenylamino)piperidin-1-yl]-2-(phenylsulfanyl)ethan-1-one
4-(3,5-dimethyl-1H-indole-2-carbonyl)-1-phenylpiperazin-2-one
{[2-(4-ethylpiperazin-1-yl)-7-methoxyquinolin-3-yl]methyl}[2-(3-methoxyphenyl)ethyl]amine
(4aS,7aR)-1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
propan-2-yl 4-[(5-ethylpyridin-2-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.5]undecane-9-carboxylate
1-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-(2-methylphenyl)piperazine
3-(2-ethylbutyl)-8-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(4-fluorophenyl)-1-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl}methyl)(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)methylamine
9-(4-fluoro-2-methylbenzenesulfonyl)-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
3-{[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]amino}-2,3-dihydro-1λ6-thiophene-1,1-dione
1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-[5-methyl-2-(propan-2-yl)phenoxy]propan-1-one
5-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-2,1,3-benzoxadiazol-1-ium-1-olate
3-[3-(3-methoxyphenoxy)azetidine-1-carbonyl]-1-methyl-5-phenyl-1H-pyrazole
methyl 1-[(3S,5S)-5-[(furan-2-ylmethyl)carbamoyl]-1-(3-phenylpropyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
{4-[(1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}pyrrolidin-3-yl)methyl]phenyl}methanol
N-benzyl-2-(thiophen-2-yl)azetidine-1-sulfonamide
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[2-(3,4-dimethoxyphenyl)ethyl]propanamide
4-ethyl-3-(piperidin-4-ylmethyl)-1-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{imidazo[1,2-a]pyrimidine-2-carbonyl}-2-(2-methylphenyl)pyrrolidine
2-[3-(naphthalene-1-carbonyl)piperidin-1-yl]acetamide
9-(4-methanesulfonylbenzoyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
2-methyl-3-[(pyridin-2-ylmethyl)amino]-N-[1-(thiophen-3-yl)propan-2-yl]benzamide
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(1,3-thiazol-4-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-[3-(dimethylamino)phenyl]-1-(1-hydroxybutan-2-yl)-1-(pyridin-4-ylmethyl)urea
{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}({5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl})amine
N-(3,4-dimethylphenyl)-1-(thiophene-2-carbonyl)piperidin-3-amine
8-[(4-methoxyphenyl)methyl]-1-(2-phenylethyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
8-(2-aminopyridine-4-carbonyl)-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-{[4-(dimethylamino)oxan-4-yl]methyl}-3-[3-fluoro-5-(trifluoromethyl)phenyl]urea
[1-({[2-(2-aminoethyl)-5,6-dimethylthieno[2,3-d]pyrimidin-4-yl](methyl)amino}methyl)cyclobutyl]methanol
8-(2-aminopyridine-4-carbonyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
6-methyl-2-(oxan-4-ylmethyl)-5-[5-(1H-pyrazol-3-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)amine
3-{5-[1-(cyclopent-3-en-1-yl)-4-phenyl-1H-imidazol-5-yl]thiophen-3-yl}prop-2-yn-1-ol
1-{1-[(2-fluoro-5-methoxyphenyl)methyl]piperidin-3-yl}-4-(4-methoxyphenyl)piperazine
9-(cyclopropylmethyl)-4-(4,6-dimethylpyrimidin-2-yl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-{[3-(2-chloro-4-fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
3-(1-{[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-3-(4-fluorophenoxymethyl)piperidine
4-[2-methyl-7-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-1,4-oxazepane
N-[3-(4-{[4-(2-chlorophenyl)piperazin-1-yl]methyl}phenoxy)propyl]thiophene-2-carboxamide
1-[4-(4-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazin-1-yl)phenyl]ethan-1-one
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-(2-methyl-1H-indol-1-yl)propanamide